MedPath

Next Generation Rocklatan

Phase 2
Not yet recruiting
Conditions
Open Angle Glaucoma
Ocular Hypertension
Interventions
Registration Number
NCT06441643
Lead Sponsor
Alcon Research
Brief Summary

The purpose of this two-stage clinical trial is to assess the safety and hypotensive efficacy of AR-17043 and PG043 ophthalmic solutions in subjects with open-angle glaucoma (OAG) or ocular hypertension (OHT).

Detailed Description

During Stage 1, approximately 100 adult subjects with OAG or OHT will be randomized to 5 arms: 3 different concentrations of AR-17043, placebo comparator, or netarsudil 0.02% (Rhopressa®) for a treatment duration of 7 days.

During Stage 2, approximately 350 adult subjects with OAG or OHT will be randomized to 5 arms: low and high concentrations of PG043 (AR-17043/latanoprost 0.005%), AR-17043 high concentration, latanoprost, or netarsudil 0.02%/latanoprost 0.005% (Rocklatan®) for a treatment duration of 28 days.

Recruitment & Eligibility

Status
NOT_YET_RECRUITING
Sex
All
Target Recruitment
450
Inclusion Criteria
  • Diagnosis of OAG or OHT in both eyes.
  • High unmedicated IOP measurements in the study eye as specified in the protocol.
  • Corrected visual acuity equal to or better than +0.7 logMAR (Snellen equivalent equal to or better than 20/100) in the study eye.
  • Other protocol-specified inclusion criteria may apply.

Stage 1 and Stage 2 Key

Exclusion Criteria
  • Current use of more than 2 ocular hypotensive medications within 30 days (either eye).
  • Intraocular pressure greater than 36 millimeters mercury (mmHg) at Screening.
  • Glaucoma other than OAG.
  • Previous glaucoma surgery.
  • Any abnormality preventing reliable measurements.
  • Unable to demonstrate proper eyedrop instillation.
  • Other protocol-specified exclusion criteria may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
AR-17043 low concentration (Stage 1)AR-17043 Ophthalmic SolutionAR-17043 Ophthalmic Solution, one drop in each eye in the morning on Day 1, followed by one drop in each eye in the evening on Days 2-7.
AR-17043 medium concentration (Stage 1)AR-17043 Ophthalmic SolutionAR-17043 Ophthalmic Solution, one drop in each eye in the morning on Day 1, followed by one drop in each eye in the evening on Days 2-7.
AR-17043 high concentration (Stage 1)AR-17043 Ophthalmic SolutionAR-17043 Ophthalmic Solution, one drop in each eye in the morning on Day 1, followed by one drop in each eye in the evening on Days 2-7.
AR-17043 vehicle (Stage 1)AR-17043 VehicleAR-17043 Vehicle, one drop in each eye in the morning on Day 1, followed by one drop in each eye in the evening on Days 2-7.
Rhopressa (Stage 1)Netarsudil 0.02% Ophthalmic SolutionNetarsudil 0.02% Ophthalmic Solution, one drop in each eye in the morning on Day 1, followed by one drop in each eye in the evening on Days 2-7.
PG043 low concentration (Stage 2)PG043 Ophthalmic SolutionPG043 Ophthalmic Solution, one drop in each eye in the evening on Days 1-28.
PG043 high concentration (Stage 2)PG043 Ophthalmic SolutionPG043 Ophthalmic Solution, one drop in each eye in the evening on Days 1-28.
AR-17043 high concentration (Stage 2)AR-17043 Ophthalmic SolutionAR-17043 Ophthalmic Solution, one drop in each eye in the evening on Days 1-28.
Latanoprost (Stage 2)Latanoprost 0.005% Ophthalmic SolutionLatanoprost 0.005% Ophthalmic Solution, one drop in each eye in the evening on Days 1-28.
Rocklatan (Stage 2)Netarsudil 0.02%/Latanoprost 0.005% Ophthalmic SolutionNetarsudil 0.02%/Latanoprost 0.005% Ophthalmic Solution, one drop in each eye in the evening on Days 1-28.
Primary Outcome Measures
NameTimeMethod
Mean diurnal IOP at Day 29 (Stage 2)Day 29 (8:00, 10:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer. Diurnal IOP will be calculated as the average of the three measurements.

Mean diurnal IOP at Day 8 (Stage 1)Day 8 (8:00, 10:00, 12:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer. Diurnal IOP will be calculated as the average of the four measurements.

Secondary Outcome Measures
NameTimeMethod
Mean change from the diurnally adjusted baseline IOP at each post-treatment timepoint (Stage 1)Baseline (8:00, 10:00, 12:00, 16:00), Day 1 (8:00, 10:00, 12:00), Day 8 (8:00, 10:00, 12:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer at each post-treatment timepoint and compared to the time-relevant (corresponding) baseline measurement. Baseline is defined as the last visit prior to initiation of treatment.

Mean percent change from baseline mean diurnal IOP at each post-treatment timepoint (Stage 1)Baseline (8:00, 10:00, 12:00, 16:00); Day 1 (8:00, 10:00, 12:00), Day 8 (8:00, 10:00, 12:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer. The baseline mean diurnal IOP will be calculated as the average of the four baseline measurements. Baseline is defined as the last visit prior to initiation of treatment.

Mean percent change from diurnally adjusted baseline IOP at each post-treatment timepoint (Stage 2)Baseline (8:00, 10:00, 16:00); Day 8 (8:00, 10:00, 16:00); Day 15 (8:00, 10:00, 16:00); Day 29 (8:00, 10:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer at each post-treatment timepoint and compared to the time-relevant (corresponding) baseline measurement. Baseline is defined as the last visit prior to initiation of treatment.

Mean change from baseline mean diurnal IOP at each post-treatment timepoint (Stage 2)Baseline (8:00, 10:00, 16:00); Day 8 (8:00, 10:00, 16:00); Day 15 (8:00, 10:00, 16:00); Day 29 (8:00, 10:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer. The baseline mean diurnal IOP will be calculated as the average of the three baseline measurements. Baseline is defined as the last visit prior to initiation of treatment.

Mean percent change from baseline mean diurnal IOP at each post-treatment timepoint (Stage 2)Baseline (8:00, 10:00, 16:00); Day 8 (8:00, 10:00, 16:00); Day 15 (8:00, 10:00, 16:00); Day 29 (8:00, 10:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer. The baseline mean diurnal IOP will be calculated as the average of the three baseline measurements. Baseline is defined as the last visit prior to initiation of treatment.

Mean IOP at each post-treatment timepoint (Stage 1)Day 1 (8:00, 10:00, 12:00), Day 8 (8:00, 10:00, 12:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer at each post-treatment timepoint.

Mean change from baseline mean diurnal IOP at each post-treatment timepoint (Stage 1)Baseline (8:00, 10:00, 12:00, 16:00), Day 1 (8:00, 10:00, 12:00), Day 8 (8:00, 10:00, 12:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer. The baseline mean diurnal IOP will be calculated as the average of the four baseline measurements. Baseline is defined as the last visit prior to initiation of treatment.

Mean IOP at each post-treatment timepoint (Stage 2)Day 8 (8:00, 10:00, 16:00); Day 15 (8:00, 10:00, 16:00); Day 29 (8:00, 10:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer at each post-treatment timepoint.

Mean change from the diurnally adjusted baseline IOP at each post-treatment timepoint (Stage 2)Baseline (8:00, 10:00, 16:00); Day 8 (8:00, 10:00, 16:00); Day 15 (8:00, 10:00, 16:00); Day 29 (8:00, 10:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer at each post-treatment timepoint and compared to the time-relevant (corresponding) baseline measurement. Baseline is defined as the last visit prior to initiation of treatment.

Mean percent change from diurnally adjusted baseline IOP at each post-treatment timepoint (Stage 1)Baseline (8:00, 10:00, 12:00, 16:00), Day 1 (8:00, 10:00, 12:00), Day 8 (8:00, 10:00, 12:00, 16:00)

Intraocular pressure (IOP) will be measured with a Goldmann tonometer at each post-treatment timepoint and compared to the time-relevant (corresponding) baseline measurement. Baseline is defined as the last visit prior to initiation of treatment.

Trial Locations

Locations (12)

Orange County Ophthalmology Medical Group

🇺🇸

Garden Grove, California, United States

United Medical Research Institute

🇺🇸

Inglewood, California, United States

Eye Research Foundation

🇺🇸

Newport Beach, California, United States

North Bay Eye Associates

🇺🇸

Petaluma, California, United States

Eye Center of Northern Colorado, PC

🇺🇸

Fort Collins, Colorado, United States

Coastal Research Associates

🇺🇸

Roswell, Georgia, United States

Rochester Ophthalmological Group

🇺🇸

Rochester, New York, United States

James D. Branch Ophthalmology

🇺🇸

Winston-Salem, North Carolina, United States

Scott & Christie and Associates, PC

🇺🇸

Cranberry Township, Pennsylvania, United States

University Eye Specialists

🇺🇸

Maryville, Tennessee, United States

Total Eye Care PA

🇺🇸

Memphis, Tennessee, United States

Piedmont Eye Center

🇺🇸

Lynchburg, Virginia, United States

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