MedPath

Ibudilast in the Treatment of Medication Overuse Headache

Phase 1
Conditions
Medication Overuse Headache
Interventions
Drug: Placebo
Registration Number
NCT01317992
Lead Sponsor
University of Adelaide
Brief Summary

The purpose of this study is to determine if ibudilast is effective in reverting patients with medication overuse headache suffering chronic daily headache back to their original episodic headache pattern.

Detailed Description

It has been established that excessive intake of medications used to treat primary headaches, particularly those containing opioids, can induce a form of secondary headache, known as medication overuse headache (MOH). Despite the significant clinical impact of this condition the mechanisms behind MOH remain poorly understood, guidelines for treatment are lacking, and relapse is common.

Recently, it has been recognised that repeated opioid exposure can facilitate pain by activating glia, the immunocompetent cells of the central nervous system, resulting in opioid-induced hyperalgesia (OIH).

The investigators hypothesise that MOH represents a form of OIH in this susceptible patient group - repeated activation of nociceptive pathways by frequent headaches interacts with the opioid induced pro-inflammatory actions of activated glia to produce chronic daily headache (CDH).

This double-blind, randomised, placebo controlled pilot study will investigate the use of ibudilast, a know attenuator of glial activation, in the treatment of medication overuse headache.

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
40
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
IbudilastIbudilastTo receive ibudilast 40mg twice daily for 8 weeks.
PlaceboPlaceboTo receive placebo twice daily for 8 weeks.
Primary Outcome Measures
NameTimeMethod
Headache Index2, 4, 8, 24 weeks

Headache Index as calculated by the summation of headache duration (hours) X headache intensity (11-point numerical rating scale), over the final two weeks of treatment.

Secondary Outcome Measures
NameTimeMethod
Medication frequency2, 4, 8, 24 weeks

Defined as number of days acute headache medication taken over the previous month.

Headache frequency2, 4, 8, 24 weeks

Defined as number of days with headache over the previous month

Duration of headache2, 4, 8, 24 weeks

Average duration of headache in hours over previous 2 weeks

Intensity of headache2, 4, 8, 24 weeks

Average intensity of headache assessed by numerical rating scale over previous 2 weeks

Frequency of probable migraine attacks2, 4, 8, 24 weeks

Defined as number of probable migraine attacks (using International Classification of Headache Disorders, second edition, criteria for diagnosis of migraine/migraine with aura) over previous month

Headache related impact on quality of life2, 4, 8, 24 weeks

As assessed via the six-item the Headache Impact Test

Allodynia symptom checklist score2, 4, 8, 24 weeks

Assesses presence of cutaneous allodynia during activities of daily living

Von Frey filament test2, 4, 8, 24 weeks

To assess sensitivity to static mechanical cutaneous allodynia

Brush allodynia test2, 4, 8, 24 weeks

To assess sensitivity to dynamic mechanical cutaneous allodynia

Response rate2, 4, 8, 24 weeks

Response defined as ≥ 30% reduction in headache days/month or headache index from baseline. Expressed as percentage of patients who saw a ≥ 30% reduction in headache index after ibudilast treatment (at week 8) and NNT, number of patients treated to see 1 patient "respond".

Relapse rate2, 4, 8, 24 weeks

Expressed as the percentage of patients who were initially classed as responders (at weeks 8) who no longer meet the criteria for responders at 6 months

Trial Locations

Locations (1)

Pain and Anaesthesia Research Clinic, Royal Adelaide Hospital

🇦🇺

Adelaide, South Australia, Australia

© Copyright 2025. All Rights Reserved by MedPath