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Phase 3 Study of Daraxonrasib (RMC-6236) in Patients With Previously Treated Metastatic Pancreatic Ductal Adenocarcinoma (PDAC)

Phase 3
Recruiting
Conditions
Pancreatic Cancer
PDAC
PDAC - Pancreatic Ductal Adenocarcinoma
Interventions
Registration Number
NCT06625320
Lead Sponsor
Revolution Medicines, Inc.
Brief Summary

The purpose of this study is to evaluate the safety and efficacy of a novel RAS(ON) inhibitor compared to standard(s) of care (SOC) treatment.

Detailed Description

This is a global, randomized, open-label, Phase 3 study designed to evaluate whether treatment with RMC-6236 will improve progression free survival (PFS) or overall survival (OS) compared to Investigator's choice of standard of care chemotherapy in patients with metastatic PDAC who were previously treated with one prior line of therapy with 5-fluorouracil (5-FU) based or gemcitabine-based regimen.

Patients will be randomized in a 1:1 ratio to receive RMC-6236 (Arm A) or Investigator's choice of standard of care chemotherapy (Arm B).

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
460
Inclusion Criteria
  • At least 18 years old and has provided informed consent.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
  • Histologically or cytologically confirmed PDAC with metastatic disease.
  • Measurable disease per RECIST 1.1.
  • Adequate organ function (bone marrow, liver, kidney, coagulation)
  • Documented RAS mutation status, either mutant or wild-type. RAS mutations defined as nonsynonymous mutations in KRAS, NRAS, or HRAS at codons 12, 13, or 61 (G12, G13, or Q61).
  • Able to take oral medications.
Exclusion Criteria
  • Prior therapy with direct RAS-targeted therapy (eg. degraders and/or inhibitors).
  • History of or known central nervous system metastatic disease.
  • Any conditions that may affect the ability to take or absorb study treatment
  • Major surgery within 4 weeks prior to randomization.
  • Patient is unable or unwilling to comply with protocol-required study visits or procedures

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
RMC-6236RMC-6236Study drug
Investigator's choice of standard of care therapyGemcitabinePatients randomized to Investigator's choice of standard of care chemotherapy will receive one of the following four treatments: * Gemcitabine and nab-paclitaxel (GnP) * Oxaliplatin, leucovorin, irinotecan, and 5-FU (Modified FOLFIRINOX: mFOLFIRINOX) * Liposomal irinotecan (Nal-IRI + 5-FU/LV) * Oxaliplatin, leucovorin and 5-FU IV (FOLFOX)
Investigator's choice of standard of care therapynab-paclitaxelPatients randomized to Investigator's choice of standard of care chemotherapy will receive one of the following four treatments: * Gemcitabine and nab-paclitaxel (GnP) * Oxaliplatin, leucovorin, irinotecan, and 5-FU (Modified FOLFIRINOX: mFOLFIRINOX) * Liposomal irinotecan (Nal-IRI + 5-FU/LV) * Oxaliplatin, leucovorin and 5-FU IV (FOLFOX)
Investigator's choice of standard of care therapyIrinotecanPatients randomized to Investigator's choice of standard of care chemotherapy will receive one of the following four treatments: * Gemcitabine and nab-paclitaxel (GnP) * Oxaliplatin, leucovorin, irinotecan, and 5-FU (Modified FOLFIRINOX: mFOLFIRINOX) * Liposomal irinotecan (Nal-IRI + 5-FU/LV) * Oxaliplatin, leucovorin and 5-FU IV (FOLFOX)
Investigator's choice of standard of care therapyLiposomal irinotecanPatients randomized to Investigator's choice of standard of care chemotherapy will receive one of the following four treatments: * Gemcitabine and nab-paclitaxel (GnP) * Oxaliplatin, leucovorin, irinotecan, and 5-FU (Modified FOLFIRINOX: mFOLFIRINOX) * Liposomal irinotecan (Nal-IRI + 5-FU/LV) * Oxaliplatin, leucovorin and 5-FU IV (FOLFOX)
Investigator's choice of standard of care therapy5-fluorouracilPatients randomized to Investigator's choice of standard of care chemotherapy will receive one of the following four treatments: * Gemcitabine and nab-paclitaxel (GnP) * Oxaliplatin, leucovorin, irinotecan, and 5-FU (Modified FOLFIRINOX: mFOLFIRINOX) * Liposomal irinotecan (Nal-IRI + 5-FU/LV) * Oxaliplatin, leucovorin and 5-FU IV (FOLFOX)
Investigator's choice of standard of care therapyOxaliplatinPatients randomized to Investigator's choice of standard of care chemotherapy will receive one of the following four treatments: * Gemcitabine and nab-paclitaxel (GnP) * Oxaliplatin, leucovorin, irinotecan, and 5-FU (Modified FOLFIRINOX: mFOLFIRINOX) * Liposomal irinotecan (Nal-IRI + 5-FU/LV) * Oxaliplatin, leucovorin and 5-FU IV (FOLFOX)
Investigator's choice of standard of care therapyleucovorinPatients randomized to Investigator's choice of standard of care chemotherapy will receive one of the following four treatments: * Gemcitabine and nab-paclitaxel (GnP) * Oxaliplatin, leucovorin, irinotecan, and 5-FU (Modified FOLFIRINOX: mFOLFIRINOX) * Liposomal irinotecan (Nal-IRI + 5-FU/LV) * Oxaliplatin, leucovorin and 5-FU IV (FOLFOX)
Primary Outcome Measures
NameTimeMethod
Progression free survival (PFS) in the RAS G12-mutant populationUp to approximately 3 years

PFS is defined as the time from randomization until disease progression or death from any cause, whichever occurs first. Progression is per response evaluation criteria in solid tumors (RECIST) v1.1 and as assessed by blinded independent central review (BICR)

Overall survival (OS) in the RAS G12-mutant populationUp to approximately 3 years

OS is defined as the time from randomization until death from any cause.

Secondary Outcome Measures
NameTimeMethod
PFS in the all-patient populationUp to approximately 3 years

PFS is defined as the time from randomization until disease progression or death from any cause, whichever occurs first. Progression is per RECIST v1.1 and as assessed by BICR.

Objective response in the RAS G12 and all-patient populationsUp to approximately 3 years

Objective response is defined as partial response (PR) or completed response (CR) per RECIST v1.1, assessed by BICR.

OS in the all-patient populationUp to approximately 3 years

OS is defined as the time from randomization until death from any cause.

Time to deterioration (TTD) in European Organization for Research and Treatment of Cancer Quality of Life Questionnaire Pancreatic Cancer Module (EORTC QLQ-PAN26) in the RAS G12 and all-patient populationsUp to approximately 3 years

TTD is defined as the time from randomization to the first occurrence of deterioration as defined by a change of at least 10 points, or death, whichever occurs first, in each subscale in EORTC QLQ-PAN26.

Time to deterioration (TTD) in European Organization for Research and Treatment of Cancer Quality of Life Questionnaire Core 30 (EORTC QLQ-C30) in the RAS G12 and all-patient populationsUp to approximately 3 years

TTD is defined as the time from randomization to the first occurrence of deterioration as defined by a change of at least 10 points, or death, whichever occurs first, in each subscale and global QoL score in EORTC QLQ-C30.

Objective response per investigator in RAS G12 and all- patient populationsUp to approximately 3 years

Objective response is defined as PR or CR per Response Evaluation Criteria in Solid Tumors (RECIST) v1.1, as assessed by the investigator.

Duration of response (DOR) in RAS G12 and all-patient populationsUp to approximately 3 years

DOR is defined as time from first evidence of objective response (PR or CR) to disease progression or death due to any cause, whichever occurs first, as assessed by BICR and by the investigator.

Time to response (TTR) in RAS G12 and all-patient populationsUp to approximately 3 years

TTR is defined as time from randomization to first evidence of objective response (PR or CR), as assessed by BICR and by the investigator.

Percentage of patients with adverse events (AEs)Up to approximately 3 years
Pharmacokinetics of RMC-6236 in RAS G12 and all-patient populationsUp to approximately 3 years

Pharmacokinetics are defined by blood concentrations of RMC-6236 over time.

Trial Locations

Locations (47)

Hospital 12 de Octubre

🇪🇸

Madrid, Spain

City of Hope-Duarte

🇺🇸

Duarte, California, United States

University of Miami Sylvester Comprehensive Cancer Center

🇺🇸

Miami, Florida, United States

The University of Chicago Medical Center

🇺🇸

Chicago, Illinois, United States

Roswell Park Cancer Institute

🇺🇸

Buffalo, New York, United States

Stephenson Cancer Center

🇺🇸

Oklahoma City, Oklahoma, United States

Osaka International Cancer

🇯🇵

Osaka, Japan

Hospital Unversitari

🇪🇸

Barcelona, Spain

Hospital Clinico de Valencia

🇪🇸

Valencia, Spain

Banner MD Anderson Cancer Center

🇺🇸

Gilbert, Arizona, United States

Mayo Clinic

🇺🇸

Phoenix, Arizona, United States

Cedars-Sinai Medical Center

🇺🇸

Los Angeles, California, United States

UCLA

🇺🇸

Los Angeles, California, United States

UC San Diego Health Moores Cancer Center

🇺🇸

San Diego, California, United States

Mission Hall UCSF

🇺🇸

San Francisco, California, United States

Rocky Mountain Cancer

🇺🇸

Aurora, Colorado, United States

Mayo Clinic Cancer Center

🇺🇸

Jacksonville, Florida, United States

Cancer Care Centers of Brevard Inc

🇺🇸

Palm Bay, Florida, United States

Johns Hopkins

🇺🇸

Baltimore, Maryland, United States

Dana Farber Cancer Institute

🇺🇸

Boston, Massachusetts, United States

Karmanos Cancer Institute

🇺🇸

Detroit, Michigan, United States

Mayo Clinic Rochester

🇺🇸

Rochester, Minnesota, United States

Washington University

🇺🇸

Saint Louis, Missouri, United States

NYU Lagone Health

🇺🇸

New York, New York, United States

Memorial Sloan Kettering Cancer Center

🇺🇸

New York, New York, United States

Columbia University Medical Center

🇺🇸

New York, New York, United States

Duke University Medical Center

🇺🇸

Durham, North Carolina, United States

University of Cincinnati Medical Center

🇺🇸

Cincinnati, Ohio, United States

Abramson Cancer Center Clinical Research Unit

🇺🇸

Philadelphia, Pennsylvania, United States

Sarah Cannon Research Institute (Tennessee)

🇺🇸

Nashville, Tennessee, United States

Texas Oncology Sammons

🇺🇸

Dallas, Texas, United States

MD Anderson Cancer Center

🇺🇸

Houston, Texas, United States

Texas Oncology - Central South

🇺🇸

Irving, Texas, United States

Huntsman Cancer Institute

🇺🇸

Salt Lake City, Utah, United States

Virginia Cancer Specialists

🇺🇸

Fairfax, Virginia, United States

Institut Paoli Calmettes

🇫🇷

Marseille, France

Centre Eugene Marquis

🇫🇷

Rennes, France

Hopital Paul Brousse

🇫🇷

Villejuif, France

Gustave Roussy

🇫🇷

Villejuif, France

Fondazione IRCCS Istituto Nazionale dei Tumori

🇮🇹

Milan, Italy

IEO-Istituto Europeo di Oncologia

🇮🇹

Milan, Italy

Azienda Ospedaliera

🇮🇹

Pisa, Italy

National Cancer Center Hospital

🇯🇵

Tokyo, Japan

Cancer Institute Hospital of JFCR

🇯🇵

Tokyo, Japan

Kanagawa Cancer Center

🇯🇵

Yokohama, Japan

Pan-American Center for Oncology Trials

🇵🇷

San Juan, Puerto Rico

Clinica Universidad de Navarra

🇪🇸

Pamplona, Spain

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