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Tigulixostat, Phase 3 Study, Placebo Controlled in Gout Patients

Phase 3
Completed
Conditions
Gout
Hyperuricemia
Gout Flare
Tophi
Interventions
Drug: Placebo
Registration Number
NCT05586958
Lead Sponsor
LG Chem
Brief Summary

The aim of this 6-month randomized multi-regional double-blind parallel group placebo-controlled phase 3 study is to assess the efficacy and safety of three different doses of Tigulixostat in gout patients with hyperuricemia.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
354
Inclusion Criteria
  • Male or female subjects between the ages of 18 85 years, inclusive.
  • Subjects with hyperuricemia and a history or presence of gout per American College of Rheumatology/European League Against Rheumatism (ACR/EULAR) 2015 criteria.
  • Subjects who are currently on urate-lowering therapies (ULT) with an sUA level ≥6.0 mg/dL at screening (Visit 1); or subjects who are currently not on ULT with an sUA level ≥7.0 mg/dL at screening (Visit 1). Subjects currently on ULT will undergo washout and must have an sUA level ≥7.0 mg/dL at Visit 3 to be randomized and participate in the study.
  • Subjects with a Body Mass Index ≤50 kg/m2 and estimated glomerular filtration rate (eGFR) ≥30 mL/min/1.73 m2 at screening (Visit 1).
Exclusion Criteria
  • Subjects with secondary hyperuricemia, enzymatic defects.
  • Subjects experiencing an acute gout attack (intense pain, swelling, or/and tenderness in the joint area) within 2 weeks prior to screening (Visit 1).
  • Subjects who have received pegloticase to treat gout which has not responded to the usual treatments.
  • Subjects who have not been receiving stable doses of drugs known to affect sUA levels for the last 3 weeks prior to screening (Visit 1).
  • Subjects with a history of xanthinuria (elevated levels of xanthine in the urine) and rheumatoid arthritis

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Tigulixostat 100mgTigulixostatTigulixostat 100mg, Once a day (QD) for up to 6 months
Tigulixostat 200mgTigulixostatTigulixostat 200mg, Once a day (QD) for up to 6 months
Tigulixostat 300mgTigulixostatTigulixostat 300mg (100mg + 200mg), Once a day (QD) for up to 6 months
PlaceboPlaceboPlacebo, Once a day (QD) for up to 6 months
Primary Outcome Measures
NameTimeMethod
The proportion of subjects with sUA levels <6.0 mg/dL sustained at months 4, 5, and 6Up to Month 6

Serum uric acid (sUA) level will be measured at Month 4,5, and 6

Secondary Outcome Measures
NameTimeMethod
The proportion of subjects with sUA levels <5.0 mg/dL sustained at months 4, 5, and 6Up to Month 6

Serum uric acid (sUA) level will be measured at Month 4,5, and 6

The proportion of subjects reporting a gout flare up to each visit.Up to Month 6

Gout flare (intense pain, swelling, or/and tenderness in the joint area) will be assessed from baseline up to 6 months

Incidence rate of adverse eventUp to Month 6

Safety assessment

Trial Locations

Locations (50)

Allied Biomedical Research Institute

🇺🇸

Miami, Florida, United States

LTD "Clinic LJ"

🇬🇪

Kutaisi, Georgia

Aleksandre Aladashvili Clinic LLC

🇬🇪

Tbilisi, Georgia

LTD Israel-Georgian Medical Research Clinic Helsicore

🇬🇪

Tbilisi, Georgia

JSC "Vian"

🇬🇪

Tbilisi, Georgia

LTD MediClub Georgia

🇬🇪

Tbilisi, Georgia

LTD Multiprofile Clinic Consilium Medulla

🇬🇪

Tbilisi, Georgia

Angeles University Foundation Medical Center

🇵🇭

Angeles, Philippines

Davao Doctors Hospital

🇵🇭

Davao, Philippines

Lipa Medix Medical Center

🇵🇭

Lipa, Philippines

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Allied Biomedical Research Institute
🇺🇸Miami, Florida, United States

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