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Nintedanib in Patients With Bronchiolitis Obliterans Syndrome Following Hematopoietic Stem Cell Transplantation

Phase 2
Recruiting
Conditions
Bronchiolitis Obliterans Syndrome (BOS)
Bronchiolitis Obliterans (BO)
Interventions
Registration Number
NCT03805477
Lead Sponsor
University Hospital, Basel, Switzerland
Brief Summary

This study investigates the safety and tolerability of Nintedanib in patients with bronchiolitis obliterans syndrome (BOS) following allogeneic hematopoietic cell transplantation. All study patients with BOS will be treated with the study drug Nintedanib (300 mg/day) as an add-on therapy to their basic immunosuppressive treatment over a 12-months treatment period.

Detailed Description

Allogeneic hematopoietic stem cell transplantation (HCT) is an established treatment option for several malignant and non-malignant disorders. An important limitation of long-term survival after HCT is chronic graft-versus-host disease (cGvHD). The manifestation of cGvHD in the lungs, bronchiolitis obliterans (BO - if proven by lung biopsy) or bronchiolitis obliterans syndrome (BOS - clinical diagnosis), has a reported incidence between 5 and 20%. Despite different treatment approaches, prognosis of BO remains poor, with an overall 3-year mortality of up to 65%. Nintedanib is an orally available indolinone derivate that competitively binds to the vascular endothelial growth factor (VEGF) receptors, fibroblast growth factor (FGF) receptors, and platelet derived growth factor (PDGF) receptors. The anti-fibrotic activities of Nintedanib may impact the progressive course of fibrotic lung diseases like BO. This study investigates the safety and tolerability of Nintedanib in patients with bronchiolitis obliterans syndrome following allogeneic hematopoietic cell transplantation.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
20
Inclusion Criteria
  • Time interval from transplant </= 5 years at the time of inclusion

  • BOS as defined per the National Institute of Health (NIH) criteria:

    1. FEV1/vital capacity < 0.7 or the fifth percentile of predicted.
    2. FEV1 < 75% of predicted with ≥ 10% decline over less than 2 years.
    3. Absence of infection in the respiratory tract, documented with investigations directed by clinical symptoms, such as chest radiographs, computed tomographic (CT) scans, or microbiologic cultures (sinus aspiration, upper respiratory tract viral screen, sputum culture, and broncho-alveolar lavage).
    4. One of the 2 supporting features of BOS: 1. Evidence of air trapping by expiratory CT or small airway thickening or bronchiectasis by high-resolution chest CT, or 2. Evidence of air trapping by PFTs: residual volume > 120% of predicted or residual volume/total lung capacity elevated outside the 90% confidence interval and prior or current diagnosis of cGvHD per NIH criteria or histologically proven BO
  • Diagnosis of BOS within 6 months before enrollment or prior diagnosis of BOS with an absolute decline of the percentage of predicted forced expiratory volume in 1 second (FEV1) by >/= 10% within the past 12 months before inclusion

Exclusion Criteria

  • Known intolerance to Nintedanib or any of its component
  • Pregnancy or nursing
  • Serum ALT > 5 x upper limit of normal (ULN) unless explained entirely by liver GvHD or total bilirubin > 3x ULN unless explained entirely by liver GvHD
  • Any acute pulmonary infection with viruses, bacteria or fungi within four weeks before study inclusion
  • Chronic oxygen therapy; non-invasive ventilation
  • Inability to give informed consent or to perform repeated pulmonary function tests (PFT)
  • Life expectancy < 1 year at the time of enrolment as suggested by the treating physician
  • Hematologic malignancy in hematologic relapse
  • Symptomatic angina pectoris
  • Therapeutic anticoagulation (primary or secondary prophylactic platelet anti-aggregation allowed)
  • Recent abdominal surgery or untreated gastric ulcer
Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
NintedanibNintedanibNintedanib 150 mg Kps bid (oral)
Primary Outcome Measures
NameTimeMethod
adverse event rate leading to interruption/ discontinuation of study treatmentfrom screening to month 12 after screening

adverse events of the following severity according to Common terminology criteria for adverse events(CTCAE): Diarrhoea ≥ grade 3; Nausea ≥ grade 3; Vomiting ≥ grade 3; Abdominal pain ≥ grade 3; Elevation of liver enzymes (AST, ALT) ≥ grade 2; Elevation of total bilirubin ≥ 2

Secondary Outcome Measures
NameTimeMethod
change in total lung capacity (TLC)Pulmonary function tests will be performed at screening, after 1, 2, 3, 6, 9, 12 and after 13 months

the volume in the lungs at maximal Inflation (measured in liters)

change of the percent of predicted forced expiratory volume in 1 second (FEV1)Pulmonary function tests will be performed at screening, after 1, 2, 3, 6, 9, 12 and after 13 months

absolute change of the percent of predicted FEV1 by ≥10% from FEV1 before enrolment (eg, 50% to 40% predicted FEV1), confirmed by 2 pulmonary function tests (PFT) performed at least two weeks apart and after exclusion of infections and extra pulmonary causes

change in forced vital capacity (FVC)Pulmonary function tests will be performed at screening, after 1, 2, 3, 6, 9, 12 and after 13 months

volume of air that can forcibly be blown out after full inspiration, (measured in Liters)

Change in exhaled nitric oxide (eNO)Pulmonary function tests will be performed at screening, after 1, 2, 3, 6, 9, 12 and after 13 months

Change in exhaled nitric oxide (eNO) (measured in parts per Billion)

changes in St. George's Respiratory Questionnaire (SGRQ)assessed at screening, after 1, 2, 3, 6, 9, 12, and after 13 months

The SGRQ is designed to measure health impairment in patients with asthma and chronic obstructive pulmonary disease (COPD); 3 component scores are calculated: symptoms; activity; impacts. Each questionnaire response has a unique empirically derived 'weight'. The lowest possible weight is zero and the highest is 100.

changes in NIH GvHD grading scoreassessed at screening, after 1, 2, 3, 6, 9, 12, and after 13 months

NIH symptom-based lung score (score 0: no symptoms, score 1: shortness of breath with stairs, score 2: shortness of breath on flat ground, score 3: shortness of breath at rest or requiring oxygen)

Change in diffusion capacity of the lung for carbon monoxide (DLCO)Pulmonary function tests will be performed at screening, after 1, 2, 3, 6, 9, 12 and after 13 months

extent to which oxygen passes from the air sacs of the lungs into the blood (measured in "ml/min/kPa)

Nitrogen (N2)-washoutPulmonary function tests will be performed at screening, after 1, 2, 3, 6, 9, 12 and after 13 months

The following describes a single-breath nitrogen test: A subject takes a breath of 100% oxygen and exhales through a one-way valve measuring nitrogen content and volume. A plot of the nitrogen concentration (as a % of total gas) vs. expired volume is obtained by increasing the nitrogen concentration from zero to the percentage of nitrogen in the alveoli. The nitrogen concentration is initially zero because the subject is exhaling the dead space oxygen they just breathed in (does not participate in alveolar exchange), and climbs as alveolar air mixes with the dead space air. The dead space can be determined from this curve by drawing a vertical line down the curve such that the areas below the curve (left of the line) and above the curve (right of the line) are equal

changes in Functional Assessment of Cancer Therapy-Bone Marrow Transplant (FACT-BMT) questionnaireassessed at screening, after 1, 2, 3, 6, 9, 12, and after 13 months

specific HSCT-patients validated self-report questionnaire using a 5 point Likert scale and covering 4 specific domains that include physical, social and family, emotional and functional well-being. Scoring produces a range from 0-148, the higher the score, the better the Quality of Life (QOL).

changes in in 6 minutes walking distance (6-MWD)6-MWD will be performed at screening, after 6, after 12 months

standardized 6-minute walk test will be performed breathing room air and performed according to the guidelines of the American Thoracic Society. Significant drop of transcutaneous measured arterial oxygen Saturation (SaO2) is defined as a ΔSaO2 ≥ 4% or SaO2 \< 90%. A significant change in walking distance will be Δ distance = 40 metre.

cumulative steroid dosesassessed at screening, after 1, 2, 3, 6, 9, 12, and after 13 months

steroid doses per month (in mg)

overall survivalassessed at screening, after 1, 2, 3, 6, 9, 12, and after 13 months

overall survival

occurrence of GvHD in other organsassessed at screening, after 1, 2, 3, 6, 9, 12, and after 13 months

occurrence of GvHD in other organs

disease-free survival of underlying hematologic diseaseassessed at screening, after 1, 2, 3, 6, 9, 12, and after 13 months

disease-free survival of underlying hematologic disease

Trial Locations

Locations (3)

King Faisal Specialist Hospital & Research Centre

🇸🇦

Riyadh, Saudi Arabia

Clinic of Hematology, University Hospital Basel

🇨🇭

Basel, Switzerland

Clinic of Respiratory Medicine, University Hospital Basel

🇨🇭

Basel, Switzerland

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