MedPath

Belatacept Early Steroid Withdrawal Trial

Phase 4
Completed
Conditions
Renal Transplantation
Interventions
Registration Number
NCT01729494
Lead Sponsor
University of Cincinnati
Brief Summary

The study purpose is to determine the safety and efficacy of a belatacept-based immunosuppressive regimen (calcineurin inhibitor free) with alemtuzumab or rabbit antithymocyte globulin (rATG) induction and early glucocorticoid withdrawal (CSWD) and a belatacept-based immunosuppressive regimen with tacrolimus-based regimen with rabbit antithymocyte globulin induction and early glucocorticoid withdrawal in renal transplant recipients.

The hypothesis is that a belatacept-based immunosuppressive regimen with alemtuzumab induction, mycophenolate mofetil (MMF)/mycophenolic acid (MPA), and early glucocorticoid withdrawal (Group A) in renal transplant recipients or Belatacept-based immunosuppressive regimen with rabbit antithymocyte globulin induction, MMF/MPA and early glucocorticoid withdrawal (Group B) will lead to less risk of graft loss, patient death, or reduced renal function at 12 months as compared to a tacrolimus-based immunosuppressive regimen with rabbit antithymocyte globulin, MMF/MPA, and early glucocorticoid withdrawal in renal transplant recipients (Group C).

Detailed Description

Renal transplant is the most effective treatment for end-stage renal disease. It provides improved survival and quality of life. Maintenance of a functioning renal transplant mandates lifelong immunosuppressive therapy to prevent immune destruction of the graft. Current immunosuppressive regimens yield 1-year survival rates of 89% for cadaveric and 94% for living-donor grafts. Over time, however, there is progressive loss of both subjects and grafts. Five-year graft survival for cadaveric and living related donor renal transplants is 67% and 80%, respectively.

The most common causes of long-term subject and graft loss in kidney transplant recipients are cardiovascular disease and chronic allograft nephropathy (CAN), respectively. Paradoxically, the principal immunosuppressive therapies for renal transplant, the calcineurin inhibitors (CNIs), cyclosporine (CsA) and tacrolimus, directly contribute to long-term allograft loss and subject death, since they are inherently nephrotoxic and can cause or exacerbate cardiovascular risks including hypertension, hypercholesterolemia, and diabetes mellitus.

There is, therefore, a substantial unmet medical need for new therapies in renal transplant that can provide short-term subject and graft survival comparable to the CNIs without their long-term nephrotoxic, cardiovascular, and metabolic effects. Because belatacept can be administered at the time of engraftment rather than in a delayed fashion, as is frequently necessary with CNIs - especially in those allografts with initial impaired renal function-- it affords immunosuppression in a timely manner. Unlike CNIs, the targeted mechanism of action of belatacept should provide immunosuppression without nephrotoxicity or adverse effects on the cardiovascular/metabolic profile.

Glucocorticoids have been a cornerstone of immunosuppressive therapy for six decades. Although glucocorticoids provide potent suppression of allo-immune responses in humans, their adverse effects including infection, diabetes, weight gain, hypertension, hyperlipidemia, bone disease, dermal thinning, collagen loss in multiple tissues, and cataracts, combined with a lack of available therapeutic monitoring all argue against their continued use in transplantation.

Belatacept represents a potential new treatment option for renal transplant recipients, which addresses the current unmet need for an immunosuppressive treatment that provides short-term outcomes comparable to calcineurin inhibitors (CNIs) with the potential to avoid their renal, cardiovascular, and metabolic toxicities. However, the initial Phase 3 studies exhibited in higher rate of acute rejection and malignancy. The malignancies were associated with recipients who were EBV negative at the time of transplant. All EBV negative patients are precluded from treatment with Belatacept. Due to the limitations of Phase 3 trial designs and the required use of basilixumab induction, it is intuitive that the addition of a potent t cell depleting induction agent may decrease the overall acute rejection rate in patients treated with belatacept.

The current study tests these assumptions with the following immunosuppressive regimens. Group A and B consist of potent T-cell depleting induction agents combined with belatacept. Group C represents the most common immunosuppressive regimen currently utilized in the United States. Each of these regimens include early withdrawal of glucocorticoids along with maintenance mycophenolate mofetil.

Based upon the totality of available evidence, the current study offers a favorable benefit/risk profile to study subjects, and the potential to continue to provide important data for the development of new immunosuppressive regimens that address important unmet needs.

The proposed Phase 4 study is designed to determine whether belatacept, in combination with other immunosuppressive agents (rabbit antithymocyte globulin or alemtuzumab, mycophenolate mofetil/EC mycophenolate sodium), may provide acceptable efficacy and safety in de novo kidney transplant recipients, in a regimen that provides simultaneous CNI freedom and early CSWD.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
316
Inclusion Criteria
  1. Male and female patients > 18 years of age.
  2. Patient who is receiving a renal transplant from a living or deceased donor.
  3. Female patients of child bearing potential must have a negative urine or serum pregnancy test within the past 48 hours prior to study inclusion.
  4. The patient has given written informed consent to participate in the study.
Exclusion Criteria
  1. Patient has previously received an organ transplant other than a kidney.

  2. Patient is receiving an human leucocyte antigen (HLA) identical living donor transplant.

  3. Patient who is a recipient of a multiple organ transplant.

  4. Patient has a most recent cytotoxic panel reactive antibody (PRA) of >25% or calculated PRA of > 50% where multiple moderate level HLA antibodies exist and in the opinion of the PI represents substantial HLA sensitization.

  5. Patient with a positive T or B cell crossmatch that is primarily due to HLA antibodies.

  6. Patient with a donor specific antibody (DSA) as deemed by the local PI to be associated with significant risk of rejection.

  7. Patient has received a blood group (ABO) incompatible donor kidney.

  8. The donor and/or donor kidney meet any of the following extended criteria for organ donation (ECD):

    • Donor age >/= 60 years OR

    • Donor age 50-59 years and 1 of the following:

      • Cerebrovascular accident (CVA) + hypertension + serum creatinine (SCr) > 1.5 mg/dL OR
      • CVA + hypertension OR
      • CVA + SCr > 1.5 mg/dL OR
      • Hypertension + SCr > 1.5 mg/dL OR
    • Cold ischemia time (CIT) > 24 hours, donor age > 10 years OR

    • Donation after cardiac death (DCD)

  9. Recipients will be receiving a dual or en bloc kidney transplant.

  10. Donor anticipated cold ischemia is > 30 hours.

  11. Recipient that is seropositive for hepatitis C virus (HCV) with detectable Hepatitis C viral load are excluded. HCV seropositive patients with a negative HCV viral load testing may be included.

  12. Recipients who are Hepatitis B core antibody seropositive are eligible if their hepatitis B viral loads are negative. After transplant, their hepatitis B viral loads will be monitored every three months for the first year after transplant. If hepatitis B viral loads become positive, patients will be treated per institutional standard of care.

  13. Patients who are Hepatitis B surface antibody seropositive and who receive a kidney from a Hepatitis B core surface antibody positive donor may be included.

  14. Recipient or donor is known to be seropositive for human immunodeficiency virus (HIV).

  15. Recipient who is seronegative for Epstein Barr virus (EBV).

  16. Patient has uncontrolled concomitant infection or any other unstable medical condition that could interfere with the study objectives.

  17. Patients with thrombocytopenia (PLT < 75,000/mm3), and/or leucopoenia (WBC < 2,000/mm3), or anemia (hemoglobin < 6 g/dL) prior to study inclusion.

  18. Patient is taking or has been taking an investigational drug in the 30 days prior to transplant.

  19. Patient who has undergone desensitization therapy within 6 months prior to transplant.

  20. Patient has a known hypersensitivity to belatacept, tacrolimus, mycophenolate mofetil, alemtuzumab, rabbit anti-thymocyte globulin, or glucocorticoids.

  21. Patient is receiving chronic steroid therapy at the time of transplant.

  22. Patients with a history of cancer (other than non-melanoma skin cell cancers cured by local resection) within the last 5 years, unless they have an expected disease free survival of > 95%.

  23. Patient is pregnant, where pregnancy is defined as the state of a female after conception and until the termination of gestation, confirmed by positive human Chorionic Gonadotropin (hCG) laboratory test.

  24. Women of childbearing potential must use reliable contraception simultaneously, unless they are status post bilateral tubal ligation, bilateral oophorectomy, or hysterectomy.

  25. Patient has any form of substance abuse, psychiatric disorder or a condition that, in the opinion of the investigator, may invalidate communication with the investigator.

  26. Inability to cooperate or communicate with the investigator.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Group Bearly cessation of steroidsRabbit antithymocyte globulin + belatacept + mycophenolate mofetil /Enteric coated (EC) mycophenolate sodium + early cessation of steroids
Group Aearly cessation of steroidsAlemtuzumab + belatacept + mycophenolate mofetil /Enteric coated mycophenolate sodium + early cessation of steroids
Group AAlemtuzumabAlemtuzumab + belatacept + mycophenolate mofetil /Enteric coated mycophenolate sodium + early cessation of steroids
Group Cearly cessation of steroidsRabbit antithymocyte globulin + tacrolimus + mycophenolate mofetil /Enteric coated (EC) mycophenolate sodium + early cessation of steroids
Group AMycophenolate mofetilAlemtuzumab + belatacept + mycophenolate mofetil /Enteric coated mycophenolate sodium + early cessation of steroids
Group Brabbit antithymocyte globulinRabbit antithymocyte globulin + belatacept + mycophenolate mofetil /Enteric coated (EC) mycophenolate sodium + early cessation of steroids
Group BMycophenolate mofetilRabbit antithymocyte globulin + belatacept + mycophenolate mofetil /Enteric coated (EC) mycophenolate sodium + early cessation of steroids
Group Crabbit antithymocyte globulinRabbit antithymocyte globulin + tacrolimus + mycophenolate mofetil /Enteric coated (EC) mycophenolate sodium + early cessation of steroids
Group CTacrolimusRabbit antithymocyte globulin + tacrolimus + mycophenolate mofetil /Enteric coated (EC) mycophenolate sodium + early cessation of steroids
Group CMycophenolate mofetilRabbit antithymocyte globulin + tacrolimus + mycophenolate mofetil /Enteric coated (EC) mycophenolate sodium + early cessation of steroids
Group ABelataceptAlemtuzumab + belatacept + mycophenolate mofetil /Enteric coated mycophenolate sodium + early cessation of steroids
Group BBelataceptRabbit antithymocyte globulin + belatacept + mycophenolate mofetil /Enteric coated (EC) mycophenolate sodium + early cessation of steroids
Primary Outcome Measures
NameTimeMethod
# Patients With Composite Endpoint of Experiencing Either Death, Graft Loss, or eGFR < 45ml/Min12 months

Number of Patients that experienced patient Death or Graft Loss or had an estimated GFR (eGFR) (MDRD) \< 45 mL/min

Secondary Outcome Measures
NameTimeMethod
Mean eGFR (MDRD) (ml/Min/1.73m2)24 months

Mean eGFR (MDRD) (ml/min/1.73m2) measured for all patients reaching 2 year endpoint

eGFR (MRDRD) < 45 ml/Min/1.73m224 months

Patients with reduced Renal function measured by estimated GFR MDRD \< 45 ml/min at 24 months

Biopsy Proven Acute Cellular Rejection24 months

Biopsy proven acute cellular rejection (BPACR)

Proteinuria UPC Ratio > 0.824 months

Number of Patients with a Urine protein/creatinine (UPC) ratio \> 0.8

# Patients Experiencing a Graft Loss But Not Including Patients Who Died With Functioning Graft (Death-censored Graft Loss)24 months

Number of patient who experienced Graft loss, not including (censored) patients who lost graft due to death

# Patients With Composite Endpoint of Either Experiencing Death, Graft Loss, or eGFR < 45ml/Min at 24 Months24 months

Composite Endpoint of number of patients who experienced either patient death, allograft loss, or had an eGFR \< 45 ml/min/1.73m2

Biopsy Proven Acute Rejection24 months

Incidence of all biopsy proven acute rejection whether clinically relevant or clinically silent.

Patient Death24 months

Number of Patients who experienced death, all causes

Biopsy Proven Acute Antibody Mediated Rejection24 months

Incidence of patients experiencing a Biopsy proven acute antibody mediated rejection (BPAMR)

Biopsy Proven Mixed Acute Rejection24 months

Incidence of patients experiencing a Biopsy proven acute cellular rejection with either DSA positive or C4d staining positive indicating antibody rejection

# of Patients Developing Denovo Donor Specific Antibody (DSA) Post-transplant24 months

Number of patients (%) with development of denovo DSA after transplant

Trial Locations

Locations (8)

University of Wisconsin-Madison

🇺🇸

Madison, Wisconsin, United States

Tampa General Hospital

🇺🇸

Tampa, Florida, United States

The Christ Hospital

🇺🇸

Cincinnati, Ohio, United States

University of Colorado Denver

🇺🇸

Denver, Colorado, United States

California Pacific Medical Center

🇺🇸

San Francisco, California, United States

University of Illinois Medical Center at Chicago

🇺🇸

Chicago, Illinois, United States

University of Cincinnati

🇺🇸

Cincinnati, Ohio, United States

University of Minnesota

🇺🇸

Minneapolis, Minnesota, United States

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