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A Single-Dose Pilot Study of Radiolabeled Amatuximab (MORAb-009) in Mesothelin Over Expressing Cancers

Phase 1
Completed
Conditions
Mesothelioma
Ovarian Cancer
Non-small Cell Lung Cancer
Pancreatic Cancer
Interventions
Registration Number
NCT01521325
Lead Sponsor
Morphotek
Brief Summary

This research is being conducted to determine the biodistribution of radiolabeled amatuximab in tumor and non-tumor tissues in subjects with mesothelin over expressing cancer including mesothelioma, pancreatic, ovarian or non small cell lung cancer.

Detailed Description

The primary objective is to determine the biodistribution of radiolabeled amatuximab in tumor and nontumor tissues in subjects with mesothelin over-expressing cancers including mesothelioma, pancreatic, ovarian, and non small cell lung cancer. This is a single-center, single-dose, open-label, pilot study of amatuximab in approximately 20 subjects with mesothelin expressing tumors. 111Indium-radiolabeled amatuximab (5 mCi) will be administered. Serial SPECT imaging (at 3 specific time points up to 196 hours after cold infusion) will be performed to determine binding to tumor and nontumor tissue. Subjects will be observed closely for safety and possible development of anti-amatuximab antibodies. Pharmacokinetics of radiolabeled antibody will be determined with imaging over time.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
6
Inclusion Criteria
  • Female and Male subjects > or = 18 years of age
  • Histologically confirmed mesothelin-expressing cancer
  • Measurable disease that has progressed through prior therapy and that includes a non-hepatic lesion for imaging that is > or = 1.5cm, as defined by RECIST v1.1 and disease location, at discretion of the physician, or evaluable by clinical symptoms supported by biomarker, radiological or pathological studies conducted within 4 weeks prior to study entry
Exclusion Criteria
  • Known allergy or hypersensitivity to monoclonal antibodies
  • Known to develop HACA
  • Prior treatment with amatuximab
  • Prior treatment with SS1 (dsFv)PE38 (ss1P)
  • Prior treatment with another test article within previous 30 days
  • Known brain metastasis
  • Known prosthetic devices that would prohibit imaging ow lesion of interest due to radiographic artifact
  • Chemotherapy, biological therapy, radiation therapy or immunotherapy within 3 weeks prior to dosing with amatuximab

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Amatuximab infusionAmatuximabSubjects will receive one infusion of radiolabeled amatuximab.
Primary Outcome Measures
NameTimeMethod
Primary Objective: determine biodistribution of radiolabeled amatuximab in tumor and nontumor tissue1 year

To determine the biodistribution of radiolabeled amatuximab in tumor and nontumor tissue in subjects with mesothelin over expressing cancer including mesothelioma, pancreatic, ovarian or nonsmall cell lung cancer by performing SPECT imaging to determine binding to tumor and non-tumor tissue.

Secondary Outcome Measures
NameTimeMethod
Secondary objectives: determine the safety of a single IV of Indium-CHX-A amatuximab1 year

To determine the safety of a single IV of Indium-CHX-A amatuximab by collecting safety data during/ after the infusions as well as obtain any potential drug-related AEs 30 days post infusion

Pharmacokinetic and serum levels1 year

To determine the PK parameters of the Indium-CHX-A amatuximab with imaging, and serum levels collected over time

uptake of Indium-CHX-A amatuximab1 year

To explore the uptake of Indium-CHX-A amatuximab with mesothelin tumor expression as determined by ICH

occurrence of HACA1 year

To tabulate the occurrence of HACA which will be measured through serum samples collected over time

correlate shed serum mesothelin to imaging1 year

To correlate shed serum mesothelin to imaging obtained after antibody administration.

Trial Locations

Locations (1)

National Cacner Institue

🇺🇸

Bethesda, Maryland, United States

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