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Safety and Immunogenicity of the Na-APR-1 Hookworm Vaccine in Healthy Adults

Phase 1
Completed
Conditions
Hookworm Infection
Hookworm Disease
Interventions
Biological: Na-APR-1 (M74)/Alhydrogel®
Biological: Gluco-Pyranosylphospho-Lipid A Aqueous Formulation
Registration Number
NCT01717950
Lead Sponsor
Baylor College of Medicine
Brief Summary

Hookworms digest hemoglobin from erythrocytes for use as an energy source via a proteolytic cascade that begins with the aspartic protease, APR-1. Vaccination with recombinant APR-1 has protected animals from infection in challenge studies. This study will evaluate the safety and immunogenicity of two formulations of Na-APR-1 (M74) in healthy adult volunteers when co-administered with different concentrations of the immunostimulant GLA-AF.

Detailed Description

Open-label, dose-escalation phase 1 clinical trial in healthy, hookworm-naïve adults:

* Study site: George Washington Medical Faculty Associates, Washington, DC

* Number of participants: 40 in 2 cohorts of 20.

In Cohort 1 five (5) volunteers will receive 30 µg Na-APR-1 (M74) /Alhydrogel®, five (5) will receive 30 µg Na-APR-1 (M74)/Alhydrogel® plus 2.5 µg GLA-AF, and ten (10) will receive 30 µg Na-APR-1 (M74) /Alhydrogel® plus 5 µg GLA-AF. In Cohort 2 five (5) volunteers will receive 100 µg Na-APR-1 (M74)/Alhydrogel®, five (5) will receive 100 µg Na-APR-1 (M74) /Alhydrogel® plus 2.5 µg GLA-AF, and ten (10) will receive 100 µg Na-APR-1 (M74)/Alhydrogel® plus 5 µg GLA-AF.

The cohorts will be enrolled in a staggered fashion with safety data assessed prior to the Na-APR-1 dose escalation from 30 to 100 µg. In addition, within each cohort, vaccinations will be staggered such that formulations containing 0, 2.5, and 5 µg GLA-AF will be tested sequentially: for example, those receiving Na-APR-1 (M74)/Alhydrogel® in combination with 2.5 µg GLA-AF will be vaccinated no sooner than 3 days after the last volunteer is vaccinated with the formulation containing no GLA-AF, whereas those vaccinated with Na-APR-1 (M74)/Alhydrogel® plus 5 µg GLA-AF will be vaccinated no sooner than 7 days after the last one receives the 2.5 µg GLA-AF formulation.

* Immunization schedule: Study days 0, 56 and 112.

* Route: IM in the deltoid muscle.

* Doses of Na-APR-1 (M74) to be tested: 30 and 100 µg.

* Doses of Alhydrogel®: 240 and 800 µg for the 30 and 100 µg doses of Na-APR-1 (M74), respectively.

* Doses of GLA-AF to be tested: 2.5 µg and 5 µg.

* Study duration: 44 weeks (10 months) per study participant; total duration of the study estimated at approximately 13 months.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
40
Inclusion Criteria
  • Males or females between 18 and 50 years, inclusive.
  • Good general health as determined by means of the screening procedure.
  • Available for the duration of the trial (44 weeks).
  • Willingness to participate in the study as evidenced by signing the informed consent document.
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Exclusion Criteria
  • Pregnancy as determined by a positive urine human choriogonadotropin (hCG) (if female).
  • Participant unwilling to use reliable contraception methods up until one month following the third immunization (if female and not surgically sterile, abstinent or at least 2 years post-menopausal).
  • Currently lactating and breast-feeding (if female).
  • Evidence of clinically significant neurologic, cardiac, pulmonary, hepatic, rheumatologic, autoimmune, diabetes, or renal disease by history, physical examination, and/or laboratory studies.
  • Known or suspected immunodeficiency.
  • Laboratory evidence of liver disease (alanine aminotransferase [ALT] greater than 1.25-times the upper reference limit).
  • Laboratory evidence of renal disease (serum creatinine greater than 1.25-times the upper reference limit, or more than trace protein or blood on urine dipstick testing).
  • Laboratory evidence of hematologic disease (hemoglobin <11.5 g/dl [females] or <12.5 g/dl [males]; absolute leukocyte count <3600/mm3 or >10.7 x 103/mm3; absolute neutrophil count [ANC] <1700/ mm3; absolute lymphocyte count <700/mm3; or platelet count <140,000/mm3).
  • Laboratory evidence of a coagulopathy (PTT or PT INR greater than 1.1-times the upper reference limit).
  • Serum glucose (random) greater than 1.2-times the upper reference limit.
  • Other condition that in the opinion of the investigator would jeopardize the safety or rights of a volunteer participating in the trial or would render the subject unable to comply with the protocol.
  • Participation in another investigational vaccine or drug trial within 30 days of starting this study.
  • Volunteer has had medical, occupational, or family problems as a result of alcohol or illicit drug use during the past 12 months.
  • History of a severe allergic reaction or anaphylaxis.
  • Severe asthma as defined by the need for daily use of inhalers or emergency clinic visit or hospitalization within 6 months of the volunteer's expected first vaccination in the study.
  • Positive ELISA for hepatitis B surface antigen (HBsAg).
  • Positive confirmatory test for HIV infection.
  • Positive confirmatory test for hepatitis C virus (HCV) infection.
  • Use of corticosteroids (excluding topical or nasal) or immunosuppressive drugs within 30 days of the volunteer's expected first vaccination in this study.
  • Receipt of a live vaccine within 4 weeks or a killed vaccine within 2 weeks prior to the volunteer's expected first vaccination in the study.
  • History of a surgical splenectomy.
  • Receipt of blood products within the past 6 months.
  • History of previous infection with hookworm or residence for more than 6 months in a hookworm-endemic area.
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Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
30 µg Na-APR-1 (M74)/Alhydrogel®Na-APR-1 (M74)/Alhydrogel®-
30 µg Na-APR-1 (M74)/Alhydrogel® plus 5.0 µg GLA-AFGluco-Pyranosylphospho-Lipid A Aqueous Formulation-
30 µg Na-APR-1 (M74)/Alhydrogel® plus 2.5 µg GLA-AFGluco-Pyranosylphospho-Lipid A Aqueous Formulation-
100 µg Na-APR-1 (M74)/Alhydrogel® plus 2.5 µg GLA-AFGluco-Pyranosylphospho-Lipid A Aqueous Formulation-
30 µg Na-APR-1 (M74)/Alhydrogel® plus 5.0 µg GLA-AFNa-APR-1 (M74)/Alhydrogel®-
100 µg Na-APR-1 (M74)/Alhydrogel® plus 5.0 µg GLA-AFGluco-Pyranosylphospho-Lipid A Aqueous Formulation-
30 µg Na-APR-1 (M74)/Alhydrogel® plus 2.5 µg GLA-AFNa-APR-1 (M74)/Alhydrogel®-
100 µg Na-APR-1 (M74)/Alhydrogel® plus 2.5 µg GLA-AFNa-APR-1 (M74)/Alhydrogel®-
100 µg Na-APR-1 (M74)/Alhydrogel®Na-APR-1 (M74)/Alhydrogel®-
100 µg Na-APR-1 (M74)/Alhydrogel® plus 5.0 µg GLA-AFNa-APR-1 (M74)/Alhydrogel®-
Primary Outcome Measures
NameTimeMethod
Vaccine-related Adverse EventsDay 290

The frequency of immediate, systemic, and local injection site adverse events will be summarized. Adverse events will be assessed by study team members at 1 hour post-vaccination as well as 3, 7, 14, and 28 days following each vaccination. In addition, study participants will be asked to complete symptom diaries for the 7 days after each vaccination.

Secondary Outcome Measures
NameTimeMethod
B cell response to Na-APR-1Study Days 14, 70, 126, 140 and 290

Dose and formulation of the Na-APR-1 (M74) vaccine that results in the highest production of Na-APR-1 (M74) specific B cells and subtypes (memory or plasma).

Exploratory cellular immune response to Na-APR-1Study Days 14, 70, 126, 140 and 290

Exploratory studies of the cellular immune responses to the Na APR-1 (M74) antigen both before and after immunization.

IgG antibody response to Na-APR-114 days after final vaccination

Dose and formulation of Na-APR-1 that generates the highest IgG antibody response at Day 126 (14 days after final vaccination), as determined by an indirect enzyme-linked immunosorbent assay (ELISA).

Trial Locations

Locations (1)

George Washington University Medical Faculty Associates

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Washington, District of Columbia, United States

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