MedPath

A Study of Single Doses of RO4998452 in Patients With Type 2 Diabetes

Phase 1
Completed
Conditions
Diabetes Mellitus Type 2
Interventions
Drug: Placebo
Registration Number
NCT01044017
Lead Sponsor
Hoffmann-La Roche
Brief Summary

This randomized, double-blind, placebo-controlled, cross-over study will evaluate the glucose concentration and other glycemic parameters of efficacy, and the safety and tolerability and pharmacokinetics of single oral doses of RO4998452 in patients with diabetes mellitus type 2. On 3 treatment days a week apart, patients will each receive orally one of 2 dose levels of RO4998452 or placebo. Anticipated time of study treatment is 3 weeks. Target sample size is \<50.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
22
Inclusion Criteria
  • Adult patients, 18-75 years of age
  • Type 2 diabetes mellitus, diagnosed for at least 3 months at screening
  • Treatment with diet and exercise
  • BMI between 27 and 40 kg/m2
Exclusion Criteria
  • Type 1 diabetes
  • History of ketoacidosis, hyperosmolar coma, or lactic acidosis
  • Renal disease or renal dysfunction
  • Evidence of significant diabetic complication
  • Currently or within 3 months prior to screening treated with any oral or injectable anti-diabetic agents (exception: insulin injection in emergency situation)
  • History of anti-diabetic triple therapy

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
ARO4998452-
BRO4998452-
CPlacebo-
Primary Outcome Measures
NameTimeMethod
Effect on postprandial plasma glucose concentrationFollowing meal 13 hours after dosing
Secondary Outcome Measures
NameTimeMethod
Mean postprandial daily plasma glucose concentration (3 consecutive meals)25 hours
Mean daily blood glucose concentration, pre-meal plasma glucose concentration, plasma insulin concentrationAssessments up to 25 hours after dosing
Safety and tolerability: AEs, laboratory parametersAEs throughout study, laboratory assessments on 3 treatment days and on follow-up
Urinary glucose excretionAssessments up to 25 hours after dosing
© Copyright 2025. All Rights Reserved by MedPath