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Use of the Cardioprotectant Dexrazoxane During Congenital Heart Surgery

Phase 1
Conditions
Heart Defects, Congenital
Interventions
Registration Number
NCT04997291
Lead Sponsor
University of Texas at Austin
Brief Summary

Cardiopulmonary bypass and arrest of the heart during cardiac surgery are necessary to allow the surgeon to perform heart operations. However, these processes can cause injury to the heart which may worsen post-operative outcomes. In fact, the effects of these injuries may continue after surgery, and lead to a long-term decrease in heart function. Neonates and young infants are at particular risk for this occurrence.

While much research has been done in adults looking for medicines that might protect the heart during surgery, few studies have been conducted in neonates and young infants. The investigators are testing Dexrazoxane, which has proven to be cardio-protective in pediatric cancer patients, in the hope that it may lessen cardiac injury during and after congenital heart surgery, and thereby improve outcomes in the neonatal and young infant population.

In order to accomplish this, the investigators must first determine how Dexrazoxane can be safely administered to young children with congenital heart disease.

Detailed Description

Neonates and infants undergoing heart surgery with cardiopulmonary bypass and cardioplegic arrest experience both inflammation and myocardial ischemia-reperfusion \[IR\] injury. These processes provoke myocardial apoptosis and oxygen free radical formation which result in cardiac injury and dysfunction. Dexrazoxane \[DRZ\] is a derivative of EDTA that is approved for prevention of anthracycline-related cardiotoxicity. It provides cardioprotection through reduction of toxic reactive oxygen species \[ROS\], and suppression of apoptosis.

The investigators propose a 12-patient pilot to determine DRZ pharmacokinetics, and to collect additional safety data in the neonatal and infant population. Efficacy of cardioprotection will not be evaluated in this preliminary investigation, though the investigators will determine postoperative time to resolution of organ failure, development of low cardiac output syndrome, length of cardiac ICU and hospital stays, laboratory indices of myocardial injury and systemic inflammation, and echocardiographic cardiac dysfunction for safety purposes, and as a run-in to the larger, randomized, placebo controlled trial. Conducting this pilot could optimize team execution of the study protocol. In addition, results could further establish the safety of DRZ in the neonatal and infant populations.

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
12
Inclusion Criteria
  • age ≤ 1 year
  • open heart surgery requiring CPB and use of cardioplegia
  • parent/guardian consent for study obtained
  • surgery planned Monday-Friday
Exclusion Criteria
  • gestational age <36 weeks at time of enrollment
  • known syndrome or genetic abnormality, except Trisomy 21
  • single ventricle physiology
  • concurrent enrollment in another research protocol

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
DexrazoxaneDexrazoxane-
Primary Outcome Measures
NameTimeMethod
Peak Plasma Concentration (Cmax)24 hours
Area under the plasma concentration vs time curve (AUC)24 hours
Minimum plasma concentration (Cmin)24 hours
Time to resolution of organ failure14 days

defined as hours to the point of being off invasive mechanical ventilation, without significant renal dysfunction \[cystatin C within normal range for age, and UOP \> 1 cc/kg/hr\], and off significant inotropic support \[defined as milrinone \>0.3 mcg/kg/min, dopamine \>3 mcg/kg/min, dobutamine \>3 mcg/kg/min, any combination of these inotropes, or any epinephrine, norepinephrine, phenylephrine or vasopressin)\] with a serum lactate \<2 mmol/L. One point will be awarded for each postoperative hour of continued organ dysfunction up to postoperative hour 336 (day 14). A score of 360 will be assigned if organ failure is not resolved by postoperative day 14, or if the patient requires mechanical circulatory support or experiences mortality. This variable has been chosen to allow for recognition of early drug effects, and those which might be delayed beyond the immediate postoperative period.

Secondary Outcome Measures
NameTimeMethod
Oxidative Stress3 days

measured by lipoperoxidation (serum F2 isoprostane)

Myocardial Injury7 days

determined by elevated serum cardiac troponin

Inflammatory activation (IL-6 and IL-10)3 days
Neurologic IR injury3 days

measured by serum activin A concentration

ICU Length of Stay60 days
Hospital Length of Stay60 days
Tei Index (via echocardiogram)60 days

the sum of the isovolumic contraction and relaxation times divided by the ejection time

Ventricular ejection fraction (via echocardiogram)60 days

the volumetric fraction of fluid ejected from a chamber with each contraction

Tissue doppler E/E' ratio (via echocardiogram)60 days

calculated as E wave divided by e' velocities

Composite outcome for neonatal cardiac surgery60 days

(per Graham, EM, et al) - binary variable defined as death, use of mechanical circulatory support, cardiac arrest requiring chest compressions, hepatic injury \[2 times the upper limit of normal for AST or ALT\], renal injury \[Cr \>1.5 mg/dL\], or lactic acidosis \[an increasing lactate \>5 mmol/L in the postoperative period\]

Trial Locations

Locations (1)

Dell Children's Medical Center of Central Texas

🇺🇸

Austin, Texas, United States

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