MedPath

Efficacy, Safety, and Tolerability of E2007 in Levodopa Treated Parkinson's Disease Patients With Motor Fluctuations

Phase 3
Completed
Conditions
Parkinson's Disease
Interventions
Drug: placebo comparator
Drug: 2 mg perampanel
Drug: 4 mg perampanel
Registration Number
NCT00368108
Lead Sponsor
Eisai Inc.
Brief Summary

This is a multi-center, randomized, double-blind, placebo-controlled, parallel-group study of E2007 in levodopa treated Parkinson's disease patients with motor fluctuations.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
752
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
placeboplacebo comparatorThe placebo dosage was a fixed dosage for the entire double-blind study. Subjects receiving the placebo were to take one dose orally once every day in the evening.
2 mg perampanel2 mg perampanelThe Perampanel 2mg dosage was fixed for the entire double-blind study. Subjects taking perampanel 2mg were to take the dose orally once every day in the evening.
4 mg perampanel4 mg perampanelThe Perampanel 4mg group first were subjected to a 4 week titration period, followed by a maintenance period for the remaining weeks. Subjects taking perampanel 4mg had a titration period of 4 weeks, starting at 2mg per day adding 1mg of perampel every two weeks up to 4mg. The dosages were to be taken orally once every day in the evening.
Primary Outcome Measures
NameTimeMethod
Mean Change From Baseline in Total Daily OFF Time (Hours) to Week 20 (Including Last Observation Carried Forward [LOCF] Data)Baseline and Week 20

Patients described themselves in home diaries as "OFF", "ON" without dyskinesias, "ON" with non troublesome dyskinesias, "ON" with troublesome dyskinesias, or Asleep, every 30 minutes during waking hours for 3 consecutive days prior to Baseline, Weeks 8, 10, 18, and 20. OFF state is when medication has worn off and is no longer providing benefits with regard to stiffness, slowness, and tremor.

Secondary Outcome Measures
NameTimeMethod
Mean Change From Baseline in Scale UPDRS Part II (ADL) Score in Total Daily OFF Time to Week 20 (Including LOCF Data)Baseline and Week 20

Patients described themselves in home diaries every 30 minutes during waking hours for 3 consecutive days prior to Baseline, Weeks 8, 12, 16, and 20. Unified Parkinson's Disease (PD) Rating Scale (UPDRS) is a standardized assessment of the symptoms and signs of PD. Part II assesses Activities of Daily Living (ADL) based on 13 items, such as speech, hygiene, and falling. Participants receive a score of 0-4 points per item, with a higher score indicating more severe symptoms. Range of possible total scores, 0 to 52. ON state is when medication is providing benefits to mobility, slowness, and stiffness. OFF state is when medication has worn off and is no longer providing benefits with regard to stiffness, slowness, and tremor.

Mean Change From Baseline in UPDRS Part III (Motor) Score in ON State (Hours) to Week 20 (Including LOCF Data)Baseline and Week 20

Patients described themselves in home diaries every 30 minutes during waking hours for 3 days prior to Baseline, Weeks 8, 12, 16, and 20. UPDRS is a standardized assessment of the symptoms and signs of PD. Part III assesses motor activity, based on 14 items, such as gait, facial expression, and rigidity. Participants receive a score of 0-4 points per item, with a higher score indicating more severe symptoms. ON state is when medication is providing benefits to stiffness, slowness, and tremor.

Mean Change From Baseline in Total Daily ON Time (Without Dyskinesias or With Non-troublesome Dyskinesias) (Hours) to Week 20 (Including LOCF Data)Baseline and Week 20

Patients described themselves in home diaries every 30 minutes during waking hours for 3 days prior to Baseline, Weeks 8, 12, 16, and 20. ON state is when medication is providing benefits to stiffness, slowness, and tremor.

Trial Locations

Locations (114)

Lehigh Valley Hospital

🇺🇸

Allentown, Pennsylvania, United States

Emory University

🇺🇸

Atlanta, Georgia, United States

Ohio State University Medical Center

🇺🇸

Columbus, Ohio, United States

Rush University Medical Center

🇺🇸

Chicago, Illinois, United States

Harvard Vanguard Medical Associates

🇺🇸

Boston, Massachusetts, United States

Baylor College of Medicine

🇺🇸

Houston, Texas, United States

University of Kansas

🇺🇸

Kansas City, Kansas, United States

University of Southern California

🇺🇸

Los Angeles, California, United States

Mayo Clinic Arizona

🇺🇸

Scottsdale, Arizona, United States

Dartmouth-Hitchcock Medical Center

🇺🇸

Lebanon, New Hampshire, United States

Pacific Parkinson Research Centre

🇨🇦

Vancouver, British Columbia, Canada

University Of Kentucky

🇺🇸

Lexington, Kentucky, United States

University of California San Francisco Medical Center

🇺🇸

San Francisco, California, United States

Duke University

🇺🇸

Durham, North Carolina, United States

University of Oklahoma - Health Sciences Center

🇺🇸

Oklahoma City, Oklahoma, United States

Neurology Associates

🇺🇸

San Antonio, Texas, United States

Mile High Research Center

🇺🇸

Denver, Colorado, United States

University Of Colorado

🇺🇸

Denver, Colorado, United States

Creighton University - Department of Neurology

🇺🇸

Omaha, Nebraska, United States

Medical College of Wisconsin

🇺🇸

Milwaukee, Wisconsin, United States

Wisconsin Institute for Neurologic and Sleep Disorders

🇺🇸

Milwaukee, Wisconsin, United States

Associated Neurologists, PC - Danbury

🇺🇸

Danbury, Connecticut, United States

Clinical Trials Inc.

🇺🇸

Little Rock, Arkansas, United States

North Alabama Neuroscience Research Associates

🇺🇸

Huntsville, Alabama, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

The Parkinson's and Movement Disorder Institute

🇺🇸

Fountain Valley, California, United States

Margolin Brain Institute

🇺🇸

Fresno, California, United States

Pivotal Research Centers

🇺🇸

Peoria, Arizona, United States

The Parkinson's Institute

🇺🇸

Sunnyvale, California, United States

Hartford Hospital

🇺🇸

Hartford, Connecticut, United States

Suncoast Neuroscience Associates, Inc.

🇺🇸

St. Petersburg, Florida, United States

Medical College of Georgia

🇺🇸

Augusta, Georgia, United States

Brain Matters Research

🇺🇸

Delray Beach, Florida, United States

Pacific Neuroscience Medical Group, Inc.

🇺🇸

Oxnard, California, United States

Georgetown University Hospital

🇺🇸

Washington, District of Columbia, United States

Parkinson's Disease and Movement Disorder Center of Boca Raton

🇺🇸

Boca Raton, Florida, United States

Sunrise Clinical Research

🇺🇸

Hollywood, Florida, United States

Cleveland Clinic Florida - Weston

🇺🇸

Weston, Florida, United States

Dekalb Neurology Associates, LLC/DNA Research

🇺🇸

Decatur, Georgia, United States

LSUHSC-Shreveport

🇺🇸

Shreveport, Louisiana, United States

Indiana University

🇺🇸

Indianapolis, Indiana, United States

OSF Saint Francis Medical Center

🇺🇸

Peoria, Illinois, United States

Fort Wayne Neurological Center

🇺🇸

Fort Wayne, Indiana, United States

University of Maryland Medical Center

🇺🇸

Baltimore, Maryland, United States

Boston University Medical Center

🇺🇸

Boston, Massachusetts, United States

Parkinson's and Movement Disorders Center of Maryland

🇺🇸

Elkridge, Maryland, United States

Quest Research Institute

🇺🇸

Bingham Farms, Michigan, United States

Albany Medical College

🇺🇸

Albany, New York, United States

The Clinical Neurosciences Center

🇺🇸

Southfield, Michigan, United States

Northern Michigan Neurology

🇺🇸

Traverse City, Michigan, United States

Struthers Parkinson's Center

🇺🇸

Golden Valley, Minnesota, United States

Columbia University

🇺🇸

New York, New York, United States

Pennsylvania Hospital

🇺🇸

Philadelphia, Pennsylvania, United States

Royal University Hospital

🇨🇦

Saskatoon, Saskatchewan, Canada

North Shore Medical Center

🇺🇸

Manhasset, New York, United States

University of Minnesota

🇺🇸

Minneapolis, Minnesota, United States

Northwest NeuroSpecialists, PLLC

🇺🇸

Tucson, Arizona, United States

University of Miami

🇺🇸

Miami, Florida, United States

Miami Research Associates

🇺🇸

Miami, Florida, United States

Palm Beach Neurological Center

🇺🇸

Palm Beach Gardens, Florida, United States

Coastal Neurological Group

🇺🇸

La Jolla, California, United States

University of California Medical Center - Irvine

🇺🇸

Irvine, California, United States

Scripps Clinic

🇺🇸

La Jolla, California, United States

University of California at San Diego - Department of Neurology

🇺🇸

La Jolla, California, United States

Loma Linda University

🇺🇸

Loma Linda, California, United States

UAMS Department of Neurology

🇺🇸

Little Rock, Arkansas, United States

Colorado Neurology

🇺🇸

Englewood, Colorado, United States

University of Florida - Department of Neurology

🇺🇸

Jacksonville, Florida, United States

Mayo Clinic Jacksonville

🇺🇸

Jacksonville, Florida, United States

Gil, Ramon A.

🇺🇸

Port Charlotte, Florida, United States

Northwestern University Medical School

🇺🇸

Chicago, Illinois, United States

University Of Iowa

🇺🇸

Iowa City, Iowa, United States

Southern Illinois University School of Medicine

🇺🇸

Springfield, Illinois, United States

Washington University

🇺🇸

St. Louis, Missouri, United States

University of Nevada School of Medicine

🇺🇸

Las Vegas, Nevada, United States

University of Medicine and Dentistry of New Jersey

🇺🇸

New Brunswick, New Jersey, United States

Parkinson's Disease and Movement Disorder Center of Long Island

🇺🇸

Commack, New York, United States

Columbia University Medical Center

🇺🇸

New York, New York, United States

New York University Medical Center

🇺🇸

Forest Hills, New York, United States

Asheville Neurology Specialists

🇺🇸

Asheville, North Carolina, United States

University of Rochester - Neurology Clinic

🇺🇸

Rochester, New York, United States

The Mount Sinai Medical Center

🇺🇸

New York, New York, United States

Asheville Neurology Specialists. PA

🇺🇸

Asheville, North Carolina, United States

Raleigh Neurology Associates, P.A.

🇺🇸

Raleigh, North Carolina, United States

The University of Toledo College of Medicine

🇺🇸

Toledo, Ohio, United States

Lankenau Hospital

🇺🇸

Wynnewood, Pennsylvania, United States

Neurology Specialists, Inc.

🇺🇸

Dayton, Ohio, United States

Radiant Research - Dallas North

🇺🇸

Dallas, Texas, United States

Agape' Medical Center, Inc.

🇺🇸

Lubbock, Texas, United States

Crozer Medical Center

🇺🇸

Upland, Pennsylvania, United States

Semmes Murphey Neurology and Spine Institute

🇺🇸

Memphis, Tennessee, United States

Bhupesh Dihenia, MD, PA

🇺🇸

Lubbock, Texas, United States

Fletcher Allen Health Care

🇺🇸

Burlington, Vermont, United States

Capitol Neurology

🇺🇸

Charleston, West Virginia, United States

Neurology and Neurosurgery Associates of Tacoma, PLLC

🇺🇸

Tacoma, Washington, United States

University of Alberta

🇨🇦

Edmonton, Alberta, Canada

University of Calgary

🇨🇦

Calgary, Alberta, Canada

Centre For Movement Disorders

🇨🇦

Markham, Ontario, Canada

David King, MD

🇨🇦

Halifax, Nova Scotia, Canada

Parkinson's and Neurodegenerative Disorders Clinic

🇨🇦

Ottawa, Ontario, Canada

Saint John Regional Hospital, 5DN

🇨🇦

Saint John, New Brunswick, Canada

Torotnto Western Hospital-University Health Network

🇨🇦

Toronto, Ontario, Canada

The Ottawa Hospital - Civic Campus

🇨🇦

Ottawa, Ontario, Canada

CHUM- Hotel-Dieu

🇨🇦

Montreal, Quebec, Canada

Montreal General Hospital

🇨🇦

Montreal, Quebec, Canada

Clinique Neuro Rive-Sud

🇨🇦

Greenfield Park, Quebec, Canada

SMBD Jewish General Hospital

🇨🇦

Montreal, Quebec, Canada

Quebec Memory and Motor Skills Disorders Clinic

🇨🇦

Quebec, Canada

Molecular Neuroimaging, LLC

🇺🇸

New Haven, Connecticut, United States

University Of South Florida Movement Disorders Clinic

🇺🇸

Tampa, Florida, United States

Kentucky Neuroscience Research

🇺🇸

Louisville, Kentucky, United States

University of Florida

🇺🇸

Gainesville, Florida, United States

Hunter Holmes McGuire

🇺🇸

Richmond, Virginia, United States

Thomas Jefferson University

🇺🇸

Philadelphia, Pennsylvania, United States

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