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Toxicity Substudy of Evaluation of Subcutaneous Proleukin in a Randomised International Trial (ESPRIT): TOXIL-2 Substudy

Registration Number
NCT00147355
Lead Sponsor
Kirby Institute
Brief Summary

This substudy is an open-label, randomised study comparing the uptake of recombinant interleukin-2 (rIL-2) in HIV-1 infected individuals receiving different combinations of antiemetics and analgesic agents during rIL-2 dosing in ESPRIT. The design is a factorial one with 4 arms. All patients will receive regular ibuprofen and paracetamol from days 1-6 of the rIL-2 dosing cycle; in addition, patients will be randomised to receive one of two antiemetic combinations, i.e. ondansetron or metoclopramide with or without low dose codeine phosphate as an additional analgesic agent.

Detailed Description

The research is a randomised open-label substudy of ESPRIT. The substudy is exploring whether the amount of rIL-2 taken during a dosing cycle of rIL-2 can be increased through controlling the predictable side-effects of rIL-2 better. This is a four arm study with a factorial design; patients will be randomised to one of four arms. Each arm consists of different combinations of adjunctive agents. Each patient will receive paracetamol and ibuprofen prophylactically throughout the cycle, the other adjunctive agents prescribed will vary according to which arm the patient is randomised to, but the antiemetic used will be either ondansetron or metoclopramide with or without low dose codeine phosphate as an additional analgesic agent. The primary end-point is the percentage of planned rIL-2 actually taken during the cycle. Secondary end-points include safety, side-effects of rIL-2 and the adjunctive agents, CD4+ T-cell changes and quality of life measures.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
28
Inclusion Criteria

Patients participating in ESPRIT and randomised to the rIL-2 arm, who:

  1. Are not at CD4+ T-cell target for the protocol
  2. Have not received rIL-2 for > 2 months
  3. Have reported both GI upset and constitutional side-effects as one of the reasons for either dose modifying in prior cycles or unwillingness to receive further rIL-2
  4. Are considered by the Investigator as medically safe to receive further dosing with rIL-2
  5. Are willing to receive further dosing with rIL-2 at the dose specified by the Investigator
  6. Are willing to sign informed consent to participate in the substudy
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Exclusion Criteria
  1. All exclusions for the receipt of rIL-2 on ESPRIT
  2. Known allergy to non-steroidal anti-inflammatory drugs (NSAIDs), opiates, 5HT-3 (serotonin-3) inhibitors, anti-dopaminergic antiemetics, or any other components of the proposed adjunct regimens.
  3. Use of other NSAIDs (cyclooxygenase-2 [COX-2] inhibitors, corticosteroids) or opiate analgesics within two weeks of rIL-2 dosing. Use of low dose aspirin as a cardio-protective agent is allowed.
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Study & Design

Study Type
INTERVENTIONAL
Study Design
FACTORIAL
Arm && Interventions
GroupInterventionDescription
AOndansetron, ibuprofen, paracetamolOndansetron 4mg bid + Ibuprofen 200mg qds + paracetamol 1g qds days 1-6 inclusive of rIL-2 dosing cycle
BOndansetron, ibuprofen, paracetamolOndansetron 4mg bid + codeine phosphate 15mg tds + Ibuprofen 200mg qds + paracetamol 1g qds days 1-6 inclusive of rIL-2 dosing cycle
DMetoclopramide, codeine phosphate, ibuprofen, paracetamolmetoclopramide 10mg qds + codeine phosphate 15mg tds + Ibuprofen 200mg qds + paracetamol 1g qds days 1-6 inclusive of rIL-2 dosing cycle
Cmetoclopramide, ibuprofen, paracetamolmetoclopramide 10mg qds + Ibuprofen 200mg qds + paracetamol 1g qds days 1-6 inclusive of rIL-2 dosing cycle
Primary Outcome Measures
NameTimeMethod
percentage of planned rIL-2 taken during the first rIL-2 dosing cycle while participating in this substudy.6 months

we are comparing the percentage of planned rIL-2 taken when randomised to one of the four combinations used as adjunctive therapies to alleviate the known side-effects of rIL-2

Secondary Outcome Measures
NameTimeMethod
Patterns of rIL-2 cycling frequency in the six months after randomisation into the substudy6 months

to explore the patterns of rIL-2 and see if the different adjuntive regimens increase tolerability such that more rIL-2 is taken

Percentage of planned rIL-2 taken during the cycles after the first cycle6 mths

this is to assess whether the adjuncts to which the patient was randomised as part of this substudy impact on better tolerability of cycles of rIL-2 beyond the first

Mean difference in rIL-2 taken during each cycle in the six-month period following randomisation into this substudy and rIL-2 uptake during the last dosing cycle immediately prior to participation in the substudy6 months

to see if the adjuncts to which the patient is randomised improve amount of rIL-2 taken compared to the cycle taken prior to enrollment in this substudy

Number of patients with dose modifications during the cycle due to toxicity6 months

to assess whether the adjuncts to which they were randomised reduced the amount of rIL-2 dose modification during the rIL-2 cycle

Number of patients with grade 1-4 constitutional upset (defined as any or all of the following: flu-like illness/fever/myalgia/arthralgia/headache) and/or GI upset and/or evidence of capillary leak syndromes6 months

to assess the impact of the randomised adjuntive agents on the predictable side-effects of rIL-2

Grade 1-4 creatinine and sodium changes during and after rIL-2 dosing;6 months

to assess the impact of the randomised adjuntive agents on the predictable effects of rIL-2 in regards to salt and water homeostasis and renal function

Changes in quality of life during and after rIL-26 months

to assess whether the use of different adjunctive agents impacted on the tolerability of rIL-2 during the cycle and post as perceived by the patients qOL

Incidence of SAE and AE6 months

to assess the incidence of SAE and AEs that are rIL-2 (captured for the main study) and adjunctive agents

Trial Locations

Locations (16)

FUNCEI

🇦🇷

Buenos Aires, Argentina

Hospital Prof. Alejandro Posadas

🇦🇷

Buenos Aires, Argentina

Nambour Hospital

🇦🇺

Nambour, Queensland, Australia

AIDS Medical Unit

🇦🇺

Brisbane, Queensland, Australia

The Alfred Hospital

🇦🇺

Melbourne, Victoria, Australia

St. Vincent's Hospital

🇦🇺

Sydney, New South Wales, Australia

Hospital General de Agudos JM Ramos Mejia

🇦🇷

Buenos Aires, Argentina

Hospital Interzonal General de Agudos Oscar Alende

🇦🇷

Mar del Plata, Argentina

Hospital Italiano de Buenos Aires

🇦🇷

Buenos Aires, Argentina

Hospital Interzonal de Agudos San Juan de Dios

🇦🇷

La Plata, Argentina

Hospital Central

🇦🇷

Mendoza, Argentina

Cairns Base Hospital

🇦🇺

Cairns, Queensland, Australia

Gold Coast Sexual Health Clinic

🇦🇺

Gold Coast, Queensland, Australia

Kaplan Medical Center

🇮🇱

Rehovot, Israel

Carlton Clinic

🇦🇺

Melbourne, Victoria, Australia

CAICI

🇦🇷

Rosario, Argentina

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