MedPath

Cocaine and Zolmitriptan

Early Phase 1
Completed
Conditions
Cocaine Use Disorder
Interventions
Drug: Placebo oral capsule
Registration Number
NCT05019430
Lead Sponsor
William Stoops
Brief Summary

Cocaine potently inhibits the reuptake of serotonin (5-HT). Increased synaptic 5-HT resulting from this reuptake inhibition activates multiple 5-HT receptor subtypes. Some of these receptor subtypes have been implicated in the abuse-related effects of cocaine, including its primary reinforcing effects (i.e., cocaine taking behavior). 5-HT1b receptors, which are autoreceptors on 5-HT nerve endings that regulate 5-HT release and heteroreceptors that also mediate other neurotransmitter release, play a particularly important role in cocaine effects, likely because they are highly expressed in the mesocorticolimbic system. The 5-HT1b system displays profound dysregulation during both active cocaine use and abstinence. Initial preclinical research showed that selective 5-HT1b agonists enhanced the reinforcing and locomotor effects of cocaine during ongoing cocaine administration, but subsequent research showed that these agents robustly attenuated reinstatement of cocaine- and cue-primed cocaine seeking behavior. These findings have been replicated in rigorously conducted studies using multiple schedules of reinforcement and negative sucrose reinforcement controls across laboratories. Notably, though, these preclinical studies used compounds not approved for use in humans, hindering translation. Recently published data show that zolmitriptan, a commercially available selective 5-HT1b agonist migraine medication, also selectively attenuates the reinforcing and other abuse-related effects of cocaine, regardless of stage of use (i.e., ongoing or extinguished cocaine self-administration).

Although a robust preclinical literature supports the premise that 5-HT1b activation reduces a number of cocaine-associated behaviors (e.g., self-administration, cocaine seeking), this area remains unstudied in humans. The overarching goal of this project is to advance these promising preclinical findings, specifically those with zolmitriptan, to a clinical population, thereby demonstrating that the 5-HT1b system plays a key role in the effects of cocaine in humans

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
12
Inclusion Criteria
  • Recent cocaine use
Exclusion Criteria
  • Abnormal screening outcome (e.g., ECG, blood chemistry result) that study physicians deem clinically significant
  • Current or past histories of substance use disorder that are deemed by the study physicians to interfere with study completion
  • History of serious physical disease, current physical disease, impaired cardiovascular functioning, chronic obstructive pulmonary disease, history of seizure or current or past histories of serious psychiatric disorder that in the opinion of the study physician would interfere with study participation will be excluded from participation
  • Females not currently using effective birth control
  • Contraindications to cocaine or zolmitriptan

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
PlaceboPlacebo oral capsuleSubjects will be maintained on oral placebo. Cocaine will be administered acutely during placebo maintenance. Placebo will be administered acutely during placebo maintenance.
Zolmitriptan Dose 2ZolmitriptanSubjects will be maintained on oral zolmitriptan dose 2. Cocaine will be administered acutely during zolmitriptan dose 2 maintenance. Placebo will be administered acutely during zolmitriptan dose 2 maintenance.
PlaceboCocaineSubjects will be maintained on oral placebo. Cocaine will be administered acutely during placebo maintenance. Placebo will be administered acutely during placebo maintenance.
Zolmitriptan Dose 1CocaineSubjects will be maintained on oral zolmitriptan dose 1. Cocaine will be administered acutely during zolmitriptan dose 1 maintenance. Placebo will be administered acutely during zolmitriptan dose 1 maintenance.
Zolmitriptan Dose 2CocaineSubjects will be maintained on oral zolmitriptan dose 2. Cocaine will be administered acutely during zolmitriptan dose 2 maintenance. Placebo will be administered acutely during zolmitriptan dose 2 maintenance.
Zolmitriptan Dose 3CocaineSubjects will be maintained on oral zolmitriptan dose 3. Cocaine will be administered acutely during zolmitriptan dose 3 maintenance. Placebo will be administered acutely during zolmitriptan dose 3 maintenance.
Zolmitriptan Dose 3ZolmitriptanSubjects will be maintained on oral zolmitriptan dose 3. Cocaine will be administered acutely during zolmitriptan dose 3 maintenance. Placebo will be administered acutely during zolmitriptan dose 3 maintenance.
Primary Outcome Measures
NameTimeMethod
Reinforcing Effects of Cocaine Following Zolmitriptan Dose 3 Maintenance.Following at least 3 days of maintenance on zolmitriptan dose 3 during inpatient admission.

Number of cocaine doses earned by subjects on a progressive ratio schedule of reinforcement.

Reinforcing Effects of Cocaine Following Placebo Maintenance.Following at least 3 days of maintenance on placebo during inpatient admission

Number of cocaine doses earned by subjects on a progressive ratio schedule of reinforcement.

Reinforcing Effects of Cocaine Following Zolmitriptan Dose 1 Maintenance.Following at least 3 days of maintenance on zolmitriptan dose 1 during inpatient admission.

Number of cocaine doses earned by subjects on a progressive ratio schedule of reinforcement.

Reinforcing Effects of Cocaine Following Zolmitriptan Dose 2 Maintenance.Following at least 3 days of maintenance on zolmitriptan dose 2 during inpatient admission.

Number of cocaine doses earned by subjects on a progressive ratio schedule of reinforcement.

Secondary Outcome Measures
NameTimeMethod
TemperatureDaily over approximately 1 month inpatient admission

Degrees fahrenheit. Measured daily during inpatient admission.

Adjective Rating Scale-Sedative12 times over approximately 1 month inpatient admission

Subjects will complete the adjective rating scale during 12 sessions while they are admitted to our inpatient unit. Responses to 16 items are summed (total score=0-64; Higher values=more sedation) to calculate scores on a sedative subscale.

Adjective Rating Scale-Stimulant12 times over approximately 1 month inpatient admission

Subjects will complete the adjective rating scale during 12 sessions while they are admitted to our inpatient unit. Responses to 16 items are summed (total score=0-64; Higher values=more sedation) to calculate scores on a stimulant subscale.

Heart rateDaily over approximately four week inpatient admissions

Beats per minute. Measured daily during inpatient admission.

Blood pressureDaily over approximately 1 month inpatient admission.

mmHg. Measured daily during inpatient admission.

Drug Effect Questionnaire12 times over approximately 1 month inpatient admission

Subjects will complete the drug effect questionnaire during 12 sessions while they are admitted to our inpatient unit. The items (total scores=0-100; Higher scores=greater drug effect) on this scale categorize the constellation of drug effects endorsed by subjects.

Side EffectsDaily over approximately 1 month inpatient admission

Subjects will complete a side effects questionnaire daily while they reside on the inpatient unit. Side Effects questions will query subjects about common effects of centrally active medications.

n-back Task12 times over approximately 1 month inpatient admission

Subjects will complete the n-back task during 12 sessions while they are admitted to our inpatient unit. Percentage of correct responses will be the outcome.

Delay Discounting Task12 times over approximately 1 month inpatient admission

Subjects will complete the delay discounting task during 12 sessions while they are admitted to our inpatient unit. Responses will be used to calculate discounting slope (i.e., K).

Stop-Signal Task Inhibitory Failures12 times over approximately 1 month inpatient admission

Subjects will complete the stop-signal task during 12 sessions while they are admitted to our inpatient unit. Proportion of inhibitory failures will be the outcome variable.

Stop-Signal Task Reaction Time12 times over approximately 1 month inpatient admission

Subjects will complete the stop-signal task during 12 sessions while they are admitted to our inpatient unit. Reaction time in milliseconds and proportion of inhibitory failures will be the outcome variables.

Trial Locations

Locations (1)

University of Kentucky

🇺🇸

Lexington, Kentucky, United States

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