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CYP4A11 and CYP4F2 Gene Variants as Makers of Cardiovascular Adverse Events of Non-steroidal Anti-inflammatory Drugs

Phase 4
Completed
Conditions
Drug-Related Side Effects and Adverse Reactions
Interventions
Other: Placebo
Registration Number
NCT02779530
Lead Sponsor
Eduardo Barbosa Coelho
Brief Summary

Randomized, double-blinded, cross-over and placebo controlled clinical trial to evaluate the association between genetic polymorphism of CYP4F2 with cardiovascular adverse effects of non-steroidal anti-inflammatory drugs (NSAIDs). Two groups were included according the CYP4F2 V433M genetic polymorphism (control - MM, N=7 vs. VV or VM variants, N=13). According the sample size planned, a mean difference of total body water delta between groups (control vs. polymorphic) of at least allow 10% could be observed.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
20
Inclusion Criteria

Healthy volunteers 18-65 years-old -

Exclusion Criteria

Use of drugs and without clinical history of adverse effects of NSAIDS

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
PlaceboPlacebo-
DiclofenacDiclofenac-
Primary Outcome Measures
NameTimeMethod
Edemaafter 6 days of diclofenac and placebo

Presence of edema, measured by the estimative of total body water (deuterium oxide dilution technique). The measurements will be done in the end of 6 days of use of placebo and diclofenac, and the delta between diclofenac and placebo will be used as endpoint

Secondary Outcome Measures
NameTimeMethod
Blood Pressureafter 6 days of diclofenac and placebo

Variation (delta) of 24h diastolic blood pressure between placebo and diclofenac phases, measured by ambulatory blood pressure monitoring (ABPM)

Trial Locations

Locations (1)

Unidade de Pesquisa Clínica HCRP-USP

🇧🇷

Ribeirao Preto, Sao Paulo, Brazil

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