MedPath

Rilapladib

Generic Name
Rilapladib
Brand Names
-
Drug Type
Small Molecule
Chemical Formula
C40H38F5N3O3S
CAS Number
412950-08-4
Unique Ingredient Identifier
O14CWE893Z
Background

Rilapladib is the third genomics-derived small molecule drug arising from the Human Genome Sciences-GlaxoSmithKline collaboration to enter clinical development. It is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor. Lp-PLA2 is an enzyme associated with the formation of atherosclerotic plaques.

Indication

Investigated for use/treatment in atherosclerosis and cardiovascular disorders.

Associated Conditions
-
Associated Therapies
-
© Copyright 2025. All Rights Reserved by MedPath