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Fulvestrant and Ipatasertib for Advanced HER-2 Negative and Estrogen Receptor Positive (ER+) Breast Cancer Following Progression on First Line CDK 4/6 Inhibitor and Aromatase Inhibitor

Phase 3
Active, not recruiting
Conditions
Breast Cancer
Interventions
Registration Number
NCT04650581
Lead Sponsor
Canadian Cancer Trials Group
Brief Summary

The purpose of this study is to find out whether a new drug, Ipatasertib, can slow the growth of advanced breast cancer when added to standard therapy (Fulvestrant).

Detailed Description

Patients enrolled in this study will receive either Ipatasertib plus Fulvestrant or placebo (a substance that looks like the study drug but does not have any active or medicinal ingredient) plus Fulvestant. The study will provide information about the ability of Ipatasertib plus Fulvestrant to control the cancer, the side effects and safety of the treatment, how patients feel while taking the treatment and associated costs.

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
250
Inclusion Criteria
  • Histologically and/or cytologically confirmed ER positive, HER-2 negative breast cancer

  • Female patients must be post-menopausal; female patients who are pre-menopausal must have ovarian suppression using LHRH agonist while on study

  • Clinical and/or radiographic progression during treatment with or within 28 days after discontinuation of first line of treatment with a CDK 4/6 inhibitor and an aromatase inhibitor (AI) for advanced/metastatic disease

  • Evidence of clinically and/or radiologically documented disease

  • ≥ 18 years of age

  • ECOG performance status of 0 or 1

  • No concurrent anti-cancer therapy and must satisfy the following criteria for previous therapy

    • Must not have received more than one prior line of treatment with a CDK 4/6 inhibitor and an AI in the advanced disease setting.
    • Treatment with CDK 4/6 inhibitor and AI must have been the most recent treatment prior to registration for this study
  • Adequate hematology and organ function, in the absence of growth factors

    • Absolute neutrophils > 1.5 x 10^9/L
    • Platelets ≥ 100 x 10^9/L
    • Hemoglobin > 90 g/L
    • Total Bilirubin ≤ 1.5 x ULN (upper limit of normal) or ≤ 3 x ULN if confirmed Gilbert's Syndrome
    • ALT and AST ≤ 2.5 x ULN (or ≤ 5.0 x ULN if liver or bone metastasis)
    • Alkaline phosphatase ≤ 2.0 x ULN (or ≤ 5.0 x ULN if liver metastases, ≤ 7.0 x ULN if bone metastasis)
    • Fasting glucose ≤ 8.3 mmol/L
    • HbA1c ≤ 7.5%
    • Serum albumin ≥ 30 g/L
    • INR ≤ 1.2
    • Serum Creatinine or Creatinine clearance ≤ 1.5 x ULN or ≥ 50 mL/min; measured directly by 24-hour urine sampling or as calculated by Crockcroft and Gault equation
Read More
Exclusion Criteria
  • Untreated or symptomatic CNS metastases, radiation treatment for CNS metastases within 28 days
  • Active inflammatory bowel disease, bowel inflammation, inability to swallow oral medication or GI condition that alters oral absorption
  • Prior treatment with fulvestrant, selective estrogen receptor degraders (SERDs) or known inhibitors of the PI3K pathway including PI3K inhibitors, AKT inhibitors, or mTOR inhibitors
  • Mean QT interval corrected for heart rate (QTc) ≥ 480 msec by ECG or history of familial long QT syndrome
  • Active or uncontrolled infections or serious illnesses or medical conditions
  • Clinically significant liver diseases
  • History of lung disease or history of opportunistic infections
  • Type 1 or Type 2 diabetes mellitus requiring insulin
  • Grade ≥ 2 uncontrolled hypercholesterolemia or hypertriglyceridemia
  • Known abnormalities in coagulation
  • History of hypersensitivity to the study drugs or components
  • Pregnant or lactating women
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Ipatasertib + FulvestrantFulvestrant-
PlaceboPlacebo-
PlaceboFulvestrant-
Ipatasertib + FulvestrantIpatasertib-
Primary Outcome Measures
NameTimeMethod
Progression-free survival (PFS) using RECIST 1.15 years
Secondary Outcome Measures
NameTimeMethod
Clinical Benefit Rate (CBR);5 years
To compare the two treatment arms with respect to investigator assessed PFS (per RECIST 1.1) in the PIK3CA/AKT1/PTEN altered cohort5 years
Investigator assessed PFS (per RECIST 1.1) in the PIK3CA/AKT1/PTEN non-altered cohort5 years
Response rate (RR) (per RECIST 1.1)5 years
Economic Evaluation of health utilities measured using EQ-5D-5L5 years
Overall survival (OS)5 years
Quality of Life (QOL) as measured using EORTC QLQ-C30 questionnaire5 years
Duration of Response (DoR)5 years
Number of participants with treatment-related adverse events as assessed by CTCAE version 5.05 years
Adverse events as measured using NCI PRO-CTCAE questionnaire5 years
Time to commencement of subsequent line of systemic therapy or death (TSST)5 years
PFS as assessed by blinded central radiology review in all enrolled patients, PIK3CA/AKT1/PTEN altered and non-altered cohorts5 years
Economic Evaluation of healthcare utilization using average cost per study subject by treatment arm to estimate an overall mean cost per study arm.5 years

Trial Locations

Locations (39)

QEII Health Sciences Centre

🇨🇦

Halifax, Nova Scotia, Canada

Centre Integre de Sante et de Services Sociaux

🇨🇦

Greenfield Park, Quebec, Canada

CHUM-Centre Hospitalier de l'Universite de Montreal

🇨🇦

Montreal, Quebec, Canada

CHA-Hopital Du St-Sacrement

🇨🇦

Quebec City, Quebec, Canada

Allan Blair Cancer Centre

🇨🇦

Regina, Saskatchewan, Canada

Victorian Breast and Oncology Care

🇦🇺

East Melbourne, Victoria, Australia

Juravinski Cancer Centre at Hamilton Health Sciences

🇨🇦

Hamilton, Ontario, Canada

Algoma District Cancer Program

🇨🇦

Sault Ste. Marie, Ontario, Canada

Gosford Hospital

🇦🇺

Gosford, New South Wales, Australia

Southern Highlands Cancer Centre

🇦🇺

Bowral, New South Wales, Australia

Lake Macquarie Private Hospital

🇦🇺

Gateshead, New South Wales, Australia

Macquarie University Hospital

🇦🇺

Macquarie University, New South Wales, Australia

Toowoomba Hospital

🇦🇺

Toowoomba, Queensland, Australia

Shoalhaven Cancer Care Centre

🇦🇺

Nowra, New South Wales, Australia

Sunshine Coast University Hospital

🇦🇺

Birtinya, Queensland, Australia

The Northern Hospital

🇦🇺

Epping, Victoria, Australia

Frankston Hospital

🇦🇺

Frankston, Victoria, Australia

Alfred Hospital

🇦🇺

Melbourne, Victoria, Australia

St John of God Bunbury

🇦🇺

Bunbury, Western Australia, Australia

Fiona Stanley Hospital

🇦🇺

Murdoch, Western Australia, Australia

Canberra Hospital

🇦🇺

Garran, Australia

Sunshine Hospital

🇦🇺

St. Albans, Victoria, Australia

Royal Brisbane and Womens Hospital

🇦🇺

Herston, Australia

BCCA - Fraser Valley Cancer Centre

🇨🇦

Surrey, British Columbia, Canada

BCCA - Cancer Centre for the Southern Interior

🇨🇦

Kelowna, British Columbia, Canada

BCCA - Vancouver Cancer Centre

🇨🇦

Vancouver, British Columbia, Canada

Regional Health Authority B, Zone 2

🇨🇦

Saint John, New Brunswick, Canada

William Osler Health System

🇨🇦

Brampton, Ontario, Canada

Royal Victoria Regional Health Centre

🇨🇦

Barrie, Ontario, Canada

Ottawa Hospital Research Institute

🇨🇦

Ottawa, Ontario, Canada

Stronach Regional Health Centre at Southlake

🇨🇦

Newmarket, Ontario, Canada

Kingston Health Sciences Centre

🇨🇦

Kingston, Ontario, Canada

London Regional Cancer Program

🇨🇦

London, Ontario, Canada

Thunder Bay Regional Health Sciences Centre/

🇨🇦

Thunder Bay, Ontario, Canada

University Health Network

🇨🇦

Toronto, Ontario, Canada

Windsor Regional Cancer Centre

🇨🇦

Windsor, Ontario, Canada

Saskatoon Cancer Centre

🇨🇦

Saskatoon, Saskatchewan, Canada

Auckland City Hospital

🇳🇿

Auckland, New Zealand

Wellington Cancer Centre, Wellington Hospital

🇳🇿

Wellington, New Zealand

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