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Rechallenge of BRAF +/- MEK Inhibitors Following an Adverse Event in Patients With Cancer

Conditions
Cancer
Interventions
Drug: BRAF inhibitor
Registration Number
NCT05080361
Lead Sponsor
University Hospital, Caen
Brief Summary

Very little data are published on the safety of a rechallenge with a BRAF inhibitor or combination of BRAF and MEK inhibitor (BRAFi and MEKi) after an adverse event (AE). This study aimed at identifying the recurrence rate of the same AE after a BRAFi +/- MEKi rechallenge in patients with cancer and the factors associated to the recurrence.

Detailed Description

This is an observational, cross-sectional, pharmacovigilance cohort study. AEs were extracted from safety reports from the World Health Organization database VigiBase®, to evaluate the safety of a rechallenge with a BRAF inhibitor or combination of BRAF and MEK inhibitor (BRAFi and MEKi) after an adverse event (AE) in patients with cancer.

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
16000
Inclusion Criteria
  • All consecutive AE cases associated with BRAFi and MEKi therapy. Combination therapy cases, where BRAFi were concurrently reported with MEKi will be identified, as well as the combination therapy regimen (V+C, D+T, E+B). We will not study MEKi monotherapy cases
Exclusion Criteria
  • MEKi monotherapy cases
  • Cases concurrently reporting on immune checkpoint inhibitor therapies

Study & Design

Study Type
OBSERVATIONAL
Study Design
Not specified
Arm && Interventions
GroupInterventionDescription
Reports of adverse events associated with the use of BRAF +/- MEK inhibitorsBRAF inhibitorReports of adverse event (individual case safety reports) from Vigibase, the World Health Organization pharmacovigilance database related to the use of BRAF +/- MEK inhibitors from inception (1986) until March, 1, 2021 will be extracted. Cases concurrently reporting on immune checkpoint inhibitor therapies will be excluded.
Primary Outcome Measures
NameTimeMethod
Recurrence rateUp to the date of the individual case safety report notification in VigiBase(r), assessed up to 10 years

The primary outcome is the rate of recurrence of the same AE after a BRAFi+/- MEKi rechallenge among informative rechallenges The recurrence rate will be obtained by dividing the number of cases with an AE recurrence by the number of informative rechallenges and will be expressed as a percentage

Secondary Outcome Measures
NameTimeMethod
Comparison of rechallenge and non-rechallenge casesUp to 10 years

Baseline characteristics (initial adverse event, cancer indication, age, sex) Measurements are the Medical Dictionary for Regulatory Activities preferred terms for adverse events and cancer indications, the Anatomical and Therapeutical Class for drugs. Age is categorized (18-45, 45-64, 65-74, \> 75y.o.), sex (male, female).

Factors associated with the recurrence after a rechallenge among informative rechallenges (i.e. variables associated with a higher recurrence rate, in a regression model)Up to 10 years

Across baseline characteristics (initial adverse event, cancer indication, age, sex). Measurements are the Medical Dictionary for Regulatory Activities preferred terms for adverse events and cancer indications, the Anatomical and Therapeutical Class for drugs. Age is categorized (18-45, 45-64, 65-74, \> 75y.o.), sex (male, female).

The recurrence is defined as a second occurrence of an initial adverse event after the treatment was reintroduced. It is a dichotomous outcome.

Data will be analyzed through a regression model, so as to determinate which of these covariates are associated with a higher recurrence rate.

Rate of occurrence of a different AE after a monotherapy or combination therapy rechallenge (among informative rechallenges)Up to the date of the individual case safety report notification in VigiBase(r), assessed up to 10 years

The occurrence rate will be obtained by dividing the number of cases with another AE that occurred following a treatment rechallenge by the number of informative rechallenges and will be expressed as a percentage

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