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Ph1b/2 Study of the Safety and Efficacy of T-DXd Combinations in Advanced HER2-expressing Gastric Cancer (DESTINY-Gastric03)

Registration Number
NCT04379596
Lead Sponsor
AstraZeneca
Brief Summary

DESTINY-Gastric03 will investigate the safety, tolerability, pharmacokinetics, immunogenicity, and preliminary antitumor activity of trastuzumab deruxtecan (T-DXd) alone or in combination with chemotherapy and/or immunotherapy in HER2-expressing advanced/metastatic gastric/gastroesophageal junction (GEJ) and esophageal adenocarcinoma patients.

Study hypotheses: Combination of T-DXd with cytotoxic chemotherapy and/or immunotherapy administered to subjects at the recommended phase 2 dose will show manageable safety and tolerability and preliminary anti-tumor efficacy so as to permit further clinical testing. T-DXd in combination with cytotoxic chemotherapy or immune checkpoint inhibitor administered to HER2-expressing gastric, GEJ and esophageal cancer patients who have not received prior treatment for advanced/metastatic disease will show preliminary evidence of anti-tumour activity and the potential to become a therapeutic option for this patient population.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
413
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Arm 3BFluorouracil (5-FU)T-DXd, Volrustomig and 5-FU or capecitabine
Arm 1CDurvalumabT-DXd and durvalumab
Arm 1CTrastuzumab deruxtecanT-DXd and durvalumab
Arm 1AFluorouracil (5-FU)T-DXd and 5-fluorouracil (5-FU)
Arm 1E(b)CapecitabineT-DXd, capecitabine, and durvalumab
Arm 1BCapecitabineT-DXd and capecitabine
Arm 1BTrastuzumab deruxtecanT-DXd and capecitabine
Arm 1D(b)CapecitabineT-DXd, capecitabine, and oxaliplatin
Arm 1E(a)Fluorouracil (5-FU)T-DXd, 5-FU, and durvalumab
Arm 1E(b)DurvalumabT-DXd, capecitabine, and durvalumab
Arm 2AFluorouracil (5-FU)Trastuzumab, 5-FU or capecitabine, and cisplatin or oxaliplatin
Arm 3AFluorouracil (5-FU)T-DXd, Volrustomig and 5-FU or capecitabine
Arm 2ACisplatinTrastuzumab, 5-FU or capecitabine, and cisplatin or oxaliplatin
Arm 2CCapecitabineT-DXd, 5-FU or capecitabine
Arm 2DPembrolizumabT-DXd, pembrolizumab and 5-FU or capecitabine
Arm 2FCapecitabineT-DXd, pembrolizumab and 5-FU or capecitabine
Arm 2DFluorouracil (5-FU)T-DXd, pembrolizumab and 5-FU or capecitabine
Arm 2EPembrolizumabT-DXd and pembrolizumab
Arm 2DTrastuzumab deruxtecanT-DXd, pembrolizumab and 5-FU or capecitabine
Arm 2ATrastuzumabTrastuzumab, 5-FU or capecitabine, and cisplatin or oxaliplatin
Arm 2BTrastuzumab deruxtecanT-DXd monotherapy
Arm 2CFluorouracil (5-FU)T-DXd, 5-FU or capecitabine
Arm 2DCapecitabineT-DXd, pembrolizumab and 5-FU or capecitabine
Arm 3ACapecitabineT-DXd, Volrustomig and 5-FU or capecitabine
Arm 3BCapecitabineT-DXd, Volrustomig and 5-FU or capecitabine
Arm 2CTrastuzumab deruxtecanT-DXd, 5-FU or capecitabine
Arm 2FFluorouracil (5-FU)T-DXd, pembrolizumab and 5-FU or capecitabine
Arm 3ATrastuzumab deruxtecanT-DXd, Volrustomig and 5-FU or capecitabine
Arm 4BTrastuzumab deruxtecanT-DXd, Rilvegostomig and 5-FU or capecitabine
Arm 2FTrastuzumab deruxtecanT-DXd, pembrolizumab and 5-FU or capecitabine
Arm 2FPembrolizumabT-DXd, pembrolizumab and 5-FU or capecitabine
Arm 3AVolrustomigT-DXd, Volrustomig and 5-FU or capecitabine
Arm 3BVolrustomigT-DXd, Volrustomig and 5-FU or capecitabine
Arm 4ATrastuzumab deruxtecanT-DXd, Rilvegostomig and 5-FU or capecitabine
Arm 4AFluorouracil (5-FU)T-DXd, Rilvegostomig and 5-FU or capecitabine
Arm 4ACapecitabineT-DXd, Rilvegostomig and 5-FU or capecitabine
Arm 4BRilvegostomigT-DXd, Rilvegostomig and 5-FU or capecitabine
Arm 4BFluorouracil (5-FU)T-DXd, Rilvegostomig and 5-FU or capecitabine
Arm 4ARilvegostomigT-DXd, Rilvegostomig and 5-FU or capecitabine
Arm 1ATrastuzumab deruxtecanT-DXd and 5-fluorouracil (5-FU)
Arm 1D(b)OxaliplatinT-DXd, capecitabine, and oxaliplatin
Arm 1D(b)Trastuzumab deruxtecanT-DXd, capecitabine, and oxaliplatin
Arm 1E(a)DurvalumabT-DXd, 5-FU, and durvalumab
Arm 1E(a)Trastuzumab deruxtecanT-DXd, 5-FU, and durvalumab
Arm 2AOxaliplatinTrastuzumab, 5-FU or capecitabine, and cisplatin or oxaliplatin
Arm 1E(b)Trastuzumab deruxtecanT-DXd, capecitabine, and durvalumab
Arm 2ACapecitabineTrastuzumab, 5-FU or capecitabine, and cisplatin or oxaliplatin
Arm 2ETrastuzumab deruxtecanT-DXd and pembrolizumab
Arm 3BTrastuzumab deruxtecanT-DXd, Volrustomig and 5-FU or capecitabine
Arm 4BCapecitabineT-DXd, Rilvegostomig and 5-FU or capecitabine
Primary Outcome Measures
NameTimeMethod
Part 1: Occurrence of adverse events (AEs) and serious adverse events (SAEs), graded according to NCI CTCAE v5.0Safety will be assessed up to the follow-up period, approximately 24 months.

Occurrence of AEs and SAEs graded according to NCI CTCAE v5.0

Part 1: Changes from baseline in electrocardiogram (ECG) resultsSafety will be assessed up to the follow-up period, approximately 24 months.

Changes in ECG results compared to baseline results.

Part 1: Changes from baseline in laboratory parametersSafety will be assessed up to the follow-up period, approximately 24 months.

Changes in laboratory parameters (every in appropriate units) compared to baseline results.

Part 1: Changes from baseline in vital signsSafety will be assessed up to the follow-up period, approximately 24 months.

Changes in vital signs results compared to baseline results.

Part 1: Ocurrence of dose-limiting toxicities (DLTs)Safety will be assessed up to the follow-up period, approximately 24 months.

Occurrence of dose limiting toxicities

Part 2, Part 3 and Part 4: Endpoint assessed by Investigator per RECIST v1.1: Confirmed Objective Response Rate (ORR)(Endpoint: ORR) Efficacy will be assessed at an average of approximately 12 months

Confirmed ORR per RECIST 1.1 is the percentage of patients with Complete Response or Partial Response that is subsequently confirmed.

Secondary Outcome Measures
NameTimeMethod
Part 2, Part 3 and Part 4: Changes from baseline in laboratory parametersSafety will be assessed up to follow-up period, approximately 24 months

Changes in laboratory parameters (every in appropriate units) compared to baseline results.

Part 1: Objective Response Rate (ORR)Efficacy will be assessed at an average of approximately 12 months

Confirmed ORR per RECIST 1.1 is the percentage of patients with Complete Response or Partial Response that is subsequently confirmed.

Part 2, Part 3 and Part 4: Changes from baseline in electrocardiogram (ECG) resultsSafety will be assessed up to follow-up period, approximately 24 months

Changes in ECG results compared to baseline results.

Disease Control Rate (DCR)Efficacy will be assessed at an average of approximately 12 months

DCR is the percentage of subjects who have a best overall response of complete response (CR) or partial response (PR) or stable disease (SD)

Comparison of PFSWhile on study drug up to study completion, approximately 24 months

Comparison of progression-free survival between participants using local HER2 test results and central HER2 test results from tumor samples with evaluable results

Part 2, Part 3 and Part 4: Changes from baseline in vital signsSafety will be assessed up to follow-up period, approximately 24 months

Changes in vital signs results compared to baseline results.

Duration of Response (DoR)Until progression or death, efficacy (DoR) will be assessed up to approximately 24 months

DOR is defined as the time from the date of first documented response until the date of documented progression or death

Serum concentration of T-DXd, total anti-HER2 antibody, and MAAA-1181a in all armsWhile on study drug up to study completion, approximately 24 months

Individual participant data and descriptive statistics will be provided for serum concentration data at each time point for each dose level for T-DXd, total anti-HER2 antibody, MAAA-1181a

Comparison of ORRWhile on study drug up to study completion, approximately 24 months

Comparison of objective response rate between participants using local HER2 test results and central HER2 test results from tumor samples with evaluable results

Comparison of DoRWhile on study drug up to study completion, approximately 24 months

Comparison of duration of response between participants using local HER2 test results and central HER2 test results from tumor samples with evaluable results

Part 2, Part 3 and Part 4: Occurrence of adverse events (AEs) and serious adverse events (SAEs)Safety will be assessed up to follow-up period, approximately 24 months

Occurrence of AEs and SAEs graded according to NCI CTCAE v5.0

Part 2, Part 3 and Part 4: Changes from baseline in body weightSafety will be assessed up to follow-up period, approximately 24 months

Changes in body weight in kilograms compared to baseline results.

Progression Free Survival (PFS)Until progression or death, efficacy (PFS) will be assessed up to approximately 24 months

PFS is the time from date of first dose until the date of objective disease progression or death

Serum concentration of durvalumab in study arms including T-DXd in combination with durvalumabWhile on study drug up to study completion, approximately 24 months

Individual participant data and descriptive statistics will be provided for serum concentration data at each time point for durvalumab.

Comparison of OSWhile on study drug up to study completion, approximately 24 months

Comparison of overall survival between participants using local HER2 test results and central HER2 test results from tumor samples with evaluable results

Overall survival (OS)Until death, efficacy (OS) will be assessed up to approximately 24 months

OS is the time from date of first dose until death due to any cause

Presence of ADAs for T-DXD, durvalumab, volrustomig and rilvegostomig (in study arms including T-DXd and durvalumab, and T-DXd and volrustomig, and T-DXd and rilvegostomig respectively)While on study drug up to study completion, approximately 24 months

Individual participant data and descriptive statistics will be provided for data at each time point for each dose level for T-DXd and durvalumab.

Serum concentrations of volrustomig and rilvegostomig in study arms including T-DXd in combination with volrustomig and T-DXd in combination with rilvegostomigWhile on study drug up to study completion, approximately 24 months

Individual participant data and descriptive statistics will be provided for data at each time point for rilvegostomig and volrustomig

Comparison of DCRWhile on study drug up to study completion, approximately 24 months

Comparison of disease control rate between participants using local HER2 test results and central HER2 test results from tumor samples with evaluable results

Trial Locations

Locations (1)

Research Site

🇬🇧

Sutton, United Kingdom

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