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A Study to Investigate Safety and Effect of Sparsentan in Combination With SGLT2 Inhibition in Participants With IgAN

Phase 2
Completed
Conditions
Immunoglobulin A Nephropathy
Interventions
Registration Number
NCT05856760
Lead Sponsor
Travere Therapeutics, Inc.
Brief Summary

This is a 28-week, open-label, multicenter, single-group Phase 2 exploratory study to determine the safety and effect of sparsentan in participants with IgAN who are at risk of disease progression to kidney failure despite being on both stable RAASi and SGLT2 inhibitor treatment for at least 12 weeks prior to study entry

Detailed Description

This is a 28-week, open-label, multicenter, single-group Phase 2 exploratory study to determine the safety and effect of sparsentan in participants with Immunoglobulin A Nephropathy (IgAN) who are at risk of disease progression to kidney failure (KF) despite being on both stable renin angiotensin aldosterone system inhibitor (RAASi) and sodium glucose cotransporter-2 (SGLT2) inhibitor treatment for at least 12 weeks prior to study entry.

Participants who provide written informed consent will be assessed for eligibility and will undergo baseline evaluations including clinical laboratory tests. Per the eligibility criteria, all participants are required to be on a stable dose(s) of angiotensin converting enzyme inhibitor (ACEI) and/or angiotensin receptor blocker (ARB) and on a stable dose of a SGLT2 inhibitor at screening and will continue their stable treatments through the screening period. Eligible participants will discontinue ACEI and/or ARB therapy the day before the Day 1 visit and remain on stable SGLT2 inhibitor dosing for the duration of the study.

Study intervention will be administered daily for a treatment period of 24 weeks with study visits conducted at weeks 2-, 4-, 12-, and 24- following Day 1. Following the 24-week treatment period, study intervention will be discontinued for 4 weeks and standard of care RAASi treatment resumed, with a safety visit at Week 28.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
48
Inclusion Criteria
  • Aged ≥18 years at the time of signing the informed consent.

  • Biopsy-proven IgAN. The biopsy may have been performed at any time in the past.

  • UA/C ≥0.3 g/g at screening

  • An eGFR value of ≥25 mL/min/1.73m2 at screening.

  • On a stable dose of an SGLT2 inhibitor for at least 12 weeks prior to screening.

  • On a stable dose of ACEI and/or ARB therapy for at least 12 weeks prior to screening that is:

    • The participant's maximum tolerated dose (MTD), and
    • at least one half of the maximum labeled dose (MLD)
Exclusion Criteria
  • IgAN secondary to another condition or immunoglobulin A (IgA) vasculitis.
  • Undergone any organ transplant, with the exception of corneal transplants.
  • Documented history of heart failure, clinically significant cardiovascular or liver disease.
  • Taking high dose (defined as >10 mg/day prednisone) or other any systemic immunosuppressive medications within 12 weeks of prior to screening.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
sparsentanSparsentanSparsentan will be administered daily as a 200-mg oral tablet. The goal is to titrate from the initial dose of 200 mg (Day 1) to the target dose of 400 mg at Week 2.
Primary Outcome Measures
NameTimeMethod
Change in urine albumin-creatinine ratio (UA/C) at Week 24Week 24

The change from baseline in UA/C at Week 24 based on first morning void (FMV) samples

Secondary Outcome Measures
NameTimeMethod
Estimated glomerular filtration rate (eGFR) at each visitWeek 24

Change from baseline eGFR at each visit

UA/C <0.2 g/g at Week 24Week 24

Achievement of UA/C of \<0.2 g/g at Week 24 based on FMV samples

UA/C and Urine protein-to-creatinine ratio (UP/C) at each visitWeek 24

Change from baseline in UA/C and UP/C at each visit based on FMV samples

30% and 50% reduction from baseline in UA/C at Week 24Week 24

Achievement of 30% and 50% reduction from baseline in UA/C at Week 24 based on FMV samples

Blood pressure (BP) at each visitWeek 24

Change from baseline systolic and diastolic BP at each visit.

Trial Locations

Locations (2)

Travere Investigational Site

🇭🇰

Tsuen Wan, Hong Kong

Travere Investigation SIte

🇺🇸

Clifton Park, New York, United States

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