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The Role of Theophylline Plus Low-dose Formoterol-budesonide in Treatment of Bronchiectasis

Phase 4
Completed
Conditions
Bronchiectasis
Interventions
Drug: Formoterol-budesonide
Drug: Placebo
Registration Number
NCT01769898
Lead Sponsor
The First Affiliated Hospital of Guangzhou Medical University
Brief Summary

The purpose of this study is to examine the efficacy and safety of 24 weeks treatment with theophylline plus low-dose formoterol-budesonide in subjects with bronchiectasis.

Detailed Description

Non-cystic fibrosis bronchiectasis is an orphan disease caused by the pathogenic vicious circle including infection, inflammation and airway repair. Today's principle of treatment is to break the cycle of inflammation and infection. Nowadays, most clinical trials are anti-infective treatment by antibiotics trying to break this cycle by reducing the bacterial load, which may cause bacterial resistance. There were still some anti-inflammation trials by using inhaled corticosteroids(ICS). Tsang and Martínez-García showed that inhaled corticosteroids reduced IL-1,IL-8 levels and sputum inflammation cells, and improved sputum volume as well as quality of life, though the corticosteroid must be high dose or medium dose combined with long-acting ß2 adrenergic agonists. As described in asthma and chronic obstructive pulmonary disease(COPD), theophylline can improve the activity of histone deacetylase (HDAC) and then enhanced the anti-inflammatory effect of steroids. We hypothesis that theophylline may have the same effect in subjects with bronchiectasis. Theophylline plus inhaled low-dose formoterol-budesonide may improve quality of life and reduce airway inflammation.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
50
Inclusion Criteria
  • Patients between 18-70 years old with non-cystic fibrosis(CF) bronchiectasis, free from acute exacerbations for at least 3 months.Stable phase of the disease.
Exclusion Criteria
  • Patients with a cigarette smoking history of more than 10 packs-year. Patients with COPD. Patients with traction bronchiectasis due to advanced fibrosis. Patients with known intolerance for theophylline. Patients with asthma. Patients with other disease disturbing outcomes of the trials. Patients without consent.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placebo+formoterol-budesonideFormoterol-budesonidePlacebo(for Theophylline sustained-release tablet) tablet by mouth 100mg every 12hours for 24weeks. Inhaled Formoterol-budesonide combined treatment 4.5µg/160µg every 12hours for 24weeks.
Placebo+formoterol-budesonidePlaceboPlacebo(for Theophylline sustained-release tablet) tablet by mouth 100mg every 12hours for 24weeks. Inhaled Formoterol-budesonide combined treatment 4.5µg/160µg every 12hours for 24weeks.
Theophylline+formoterol-budesonideFormoterol-budesonideTheophylline sustained-release tablet by mouth 100mg every 12hours for 24weeks. Inhaled formoterol-budesonide combined treatment 4.5µg/160µg every 12hours for 24weeks.
Theophylline+formoterol-budesonideTheophyllineTheophylline sustained-release tablet by mouth 100mg every 12hours for 24weeks. Inhaled formoterol-budesonide combined treatment 4.5µg/160µg every 12hours for 24weeks.
Primary Outcome Measures
NameTimeMethod
Quality of Life Assessment with St George's Respiratory Questionnaire(SGRQ) and Leicester Cough Questionnaire(LCQ)Baseline and 24 weeks
Secondary Outcome Measures
NameTimeMethod
Changes of sputum characteristics from baseline to 24 weeksBaseline and 24 weeks
Changes of 24 hour sputum volume from baseline to 24 weeksBaseline and 24 weeks
Changes of forced expiratory volume in 1 second(FEV1) from baseline to 24 weeksBaseline and 24 weeks
Mean number of exacerbations per patient per 24 weeksBaseline and 24 weeks

Exacerbations defined by persistent (≥ 24 h) deterioration in at least three respiratory symptoms, including cough, dyspnea, hemoptysis, increased sputum purulence or volume, chest pain (with or without fever).

Changes of peak expiratory flow(PEF) from baseline to 24 weeksBaseline and 24 weeks
Induced sputum cytology countBaseline and 24 weeks
Changes of sputum culture from baseline to 24 weeksBaseline and 24 weeks
Tumor necrosis factor(TNF)αBaseline and 24 weeks

Test TNF-α both in blood and sputum.

Activity of histone deacetylase(HDAC)Baseline and 24 weeks

HDACs are extracted from cells in blood.

Activity of histone acetyltransferase(HAT)Baseline and 24 weeks

HATs are extracted from cells in blood.

8-IsoprostaneBaseline and 24 weeks
Neutrophilic granulocytes in blood routine examinationBaseline and 24 weeks
White blood cells in blood routine examinationBaseline and 24 weeks
Monocytes in blood routine examinationBaseline and 24 weeks
Eosinophilic granulocytes in blood routine examinationBaseline and 24 weeks
Number of participants with Adverse events as a measure of safety and tolerability24 weeks

Adverse events may contain symptoms such as nausea, sickness, headache, insomnia, palpitation, arrhythmia and so on. Record the symptoms and times of the patients.

Plasma Concentration of Theophylline24 weeks

Venous blood was taken for plasma theophylline at the end of the treatment period. (At the very time of 2 hours after patients taken the pills)

IL-6Baseline and 24 weeks

Test IL-6 both in blood and sputum.

IL-8Baseline and 24 weeks

Test IL-8 both in blood and sputum.

IL-10At 24 weeks

Test IL-10 both in blood and sputum.

Changes of mean forced expiratory flow between 25% and 75% of the FVC(FEF25-75)from baseline to 24 weeksBaseline and 24 weeks
Changes of forced vital capacity(FVC) from baseline to 24 weeksBaseline and 24 weeks

Trial Locations

Locations (2)

State Key Laboratory of Respiratory Research Institute.

🇨🇳

Guangzhou City, Guangdong, China

The First Affiliated Hospital of Guangzhou Medical University

🇨🇳

Guangzhou, Guangdong, China

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