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Efficacy, Safety, Tolerability And Actual Use Study Of Bococizumab And An Autoinjector (Pre-Filled Pen) In Subjects With Hyperlipidemia Or Dyslipidemia

Phase 3
Completed
Conditions
Hyperlipidemia
Interventions
Biological: Bococizumab 150mg
Biological: Bococizumab 75mg
Biological: Bococizumab 150mg placebo
Biological: Bococizumab 75mg placebo
Registration Number
NCT02458287
Lead Sponsor
Pfizer
Brief Summary

This study is a multicenter, randomized study in subjects with high cholesterol receiving statins to assess the efficacy to lower LDL-C, the safety, tolerability and actual use of bococizumab and an autoinjector (pre-filled pen).

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
299
Inclusion Criteria
  • Treated with a statin - Fasting LDL-C >=70mg/dL and triglycerides <=400mg/dL
Exclusion Criteria
  • Pregnant or breastfeeding females - Cardiovascular or cerebrovascular event or procedures during the past 90 days - Congestive heart failure NYHA class IV - Poorly controlled hypertension

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Bococizumab 150mgBococizumab 150mgBococizumab 150mg autoinjector (pre-filled pen)
Bococizumab 75mgBococizumab 75mgBococizumab 75mg autoinjector (pre-filled pen)
Bococizumab 150mg placeboBococizumab 150mg placeboBococizumab 150mg placebo autoinjector (pre-filled pen)
Bococizumab 75mg placeboBococizumab 75mg placeboBococizumab 75mg autoinjector (pre-filled pen)
Primary Outcome Measures
NameTimeMethod
Percentage of Injections That Met the Definition for Successful Assessment Using the Participant Assessment Tool (PAT) for Bococizumab 150 mg Dose Group at Week 4Week 4

A successful injection based on PAT was an injection where the participant answered "yes" to all the three questions: "Were you able to inject your medicine?" "Has the blue bar moved across the window?" Was the medicine not flowing after needle withdrawn?"

Percentage of Injections That Met the Definition for Successful Assessment Using the Participant Assessment Tool (PAT) for Bococizumab 150 mg Dose Group at Week 2Week 2

A successful injection based on PAT was an injection where the participant answered "yes" to all the three questions: "Were you able to inject your medicine?" "Has the blue bar moved across the window?" Was the medicine not flowing after needle withdrawn?"

Percentage of Injections That Met the Definition for Successful Assessment Using the Participant Assessment Tool (PAT) for Bococizumab 150 mg Dose Group at Week 8Week 8

A successful injection based on PAT was an injection where the participant answered "yes" to all the three questions: "Were you able to inject your medicine?" "Has the blue bar moved across the window?" Was the medicine not flowing after needle withdrawn?"

Percent Change From Baseline at Week 12 in Fasting Low Density Lipoprotein Cholesterol (LDL-C) Level for Bococizumab 150 mg Dose Group and Matched PlaceboBaseline, Week 12
Percentage of Injections That Met the Definition for Successful Assessment Using the Participant Assessment Tool (PAT) for Bococizumab 150 mg Dose Group at Week 0 (Day 1)Week 0 (Day 1)

A successful injection based on PAT was an injection where the participant answered "yes" to all the three questions: "Were you able to inject your medicine?" "Has the blue bar moved across the window?" Was the medicine not flowing after needle withdrawn?"

Percentage of Injections That Met the Definition for Successful Assessment Using the Participant Assessment Tool (PAT) for Bococizumab 150 mg Dose Group at Week 10Week 10

A successful injection based on PAT was an injection where the participant answered "yes" to all the three questions: "Were you able to inject your medicine?" "Has the blue bar moved across the window?" Was the medicine not flowing after needle withdrawn?"

Percentage of Injections That Met the Definition for Successful Assessment Using the Participant Assessment Tool (PAT) for Bococizumab 150 mg Dose Group at Week 6Week 6

A successful injection based on PAT was an injection where the participant answered "yes" to all the three questions: "Were you able to inject your medicine?" "Has the blue bar moved across the window?" Was the medicine not flowing after needle withdrawn?"

Secondary Outcome Measures
NameTimeMethod
Percent Change From Baseline in Fasting Non- High Density Lipoprotein Cholesterol (Non HDL-C) at Week 12Baseline, Week 12
Percentage of Injections That Met the Definition for Successful Assessment Using the Participant Assessment Tool (PAT) for Bococizumab 75 mg Dose Group and Combined Bococizumab 150 mg and 75 mg Dose Group at Week 0 (Day 1), 2, 4, 6, 8 and 10Week 0 (Day 1), 2, 4, 6, 8, 10

A successful injection based on PAT was an injection where the participant answered "yes" to all the three questions: "Were you able to inject your medicine?" "Has the blue bar moved across the window?" Was the medicine not flowing after needle withdrawn?"

Percent Change From Baseline in Apolipoprotein B (ApoB) at Week 12Baseline, Week 12
Percent Change From Baseline at Week 12 in Fasting Low Density Lipoprotein Cholesterol (LDL-C) Level for Bococizumab 75 mg Dose Group and Matched PlaceboBaseline, Week 12
Percentage of Participants With Anti-Drug Antibodies (ADA) and Neutralizing Antibodies (nAb)Baseline up to 18 weeks

Percentage of participants with at least 1 positive ADA titer or 1 positive nAb titer were reported. Participants with their ADA titer levels \>=6.23 were considered as ADA positive and participants with their nAb titer level \>=1.58 were considered as nAb positive.

Plasma Concentration of Bococizumab at Week 12Week 12
Plasma Concentration of Proprotein Convertase Subtilisin Kexin Type 9 (PCSK9) at Week 12Week 12

PCSK9 is an enzyme encoded by the PCSK9 gene in humans on chromosome. It is the 9th member of the proprotein convertase family of proteins that activate other proteins.

Percent Change From Baseline in Fasting Total Cholesterol (TC) at Week 12Baseline, Week 12
Percentage of Injections That Met the Definition for Successful Assessment Using the Observer Assessment Tool (OAT) for Bococizumab 150 mg Dose, Bococizumab 75 mg Dose Group and Combined Bococizumab 150 mg and 75 mg Dose Group at Week 0 (Day 1), 4 and 8Week 0 (Day 1), 4, 8

As per the OAT, a 'successful' injection was based on observer's response for the question - "Was the administration successful?''. Observer's response being 'Yes' corresponded to a successful injection.

Number of Participants With Treatment-Emergent Adverse Events (AEs) and Serious Adverse Events (SAEs)Baseline up to 18 weeks

An AE was any untoward medical occurrence in a participant who received study drug without regard to possibility of causal relationship. SAE was an AE resulting in any of the following outcomes or deemed significant for any other reason: death; Initial or prolonged inpatient hospitalization; life threatening experience (immediate risk of dying); persistent or significant disability/incapacity; congenital anomaly. Treatment-emergent were events between first dose of study drug up to the follow up visit (up to 18 weeks), that were absent before treatment or that worsened relative to pretreatment state. AEs included both SAEs and non-SAEs.

Trial Locations

Locations (30)

Omega Clinical Research Center

🇺🇸

Metairie, Louisiana, United States

National Research Institute

🇺🇸

Los Angeles, California, United States

A & R Research Group LLC

🇺🇸

Pembroke Pines, Florida, United States

Evanston Premier Healthcare Research,LLC

🇺🇸

Evanston, Illinois, United States

North Georgia Internal Medicine

🇺🇸

Woodstock, Georgia, United States

PMG Research Of Charleston

🇺🇸

Mount Pleasant, South Carolina, United States

Rainier Clinical Research Center, Inc.

🇺🇸

Renton, Washington, United States

Heart Care Associates, P.C.

🇺🇸

Hopewell, Virginia, United States

ACRC - Cardiology

🇺🇸

Atlantis, Florida, United States

Clinical Research of South Florida

🇺🇸

Coral Gables, Florida, United States

Palmetto Clinical Research

🇺🇸

Summerville, South Carolina, United States

Invesclinic, LLC

🇺🇸

Fort Lauderdale, Florida, United States

California Medical Research Associates Inc.

🇺🇸

Northridge, California, United States

Clinical Trial Research

🇺🇸

Lincoln, California, United States

Texas Center for Drug Development, Inc.

🇺🇸

Houston, Texas, United States

Diablo Clinical Research, Inc.

🇺🇸

Walnut Creek, California, United States

Manassas Clinical Research Center

🇺🇸

Manassas, Virginia, United States

North Georgia Clinical Research

🇺🇸

Woodstock, Georgia, United States

Radiant Research Incorporated

🇺🇸

Chandler, Arizona, United States

Clinical Research Atlanta

🇺🇸

Stockbridge, Georgia, United States

Solaris Clinical Research

🇺🇸

Meridian, Idaho, United States

PharmQuest

🇺🇸

Greensboro, North Carolina, United States

Buynak Clinical Research, P.C.

🇺🇸

Valparaiso, Indiana, United States

Northern California Research

🇺🇸

Sacramento, California, United States

Clinical Research of Miami, Inc.

🇺🇸

Miami, Florida, United States

Prestige Clinical Research Center, Inc.

🇺🇸

Miami, Florida, United States

Midwest Institute For Clinical Research

🇺🇸

Indianapolis, Indiana, United States

L-MARC Research Center

🇺🇸

Louisville, Kentucky, United States

Sterling Research Group, Ltd.

🇺🇸

Cincinnati, Ohio, United States

National Clinical Research-Richmond, Inc.

🇺🇸

Richmond, Virginia, United States

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