MedPath

Study BT8009-230 in Participants With Locally Advanced or Metastatic Urothelial Cancer (Duravelo-2)

Phase 2
Recruiting
Conditions
Metastatic Urothelial Cancer
Interventions
Registration Number
NCT06225596
Lead Sponsor
BicycleTx Limited
Brief Summary

This is a global, multicenter, randomized, open-label study, with an adaptive design. The main objective of the study is to measure the efficacy and safety of BT8009 (zelenectide pevedotin) as monotherapy and in combination with pembrolizumab in participants with locally advanced or metastatic urothelial cancer (UC). The study includes a dose selection phase followed by an adaptive design continuation. The study is comprised of 2 cohorts. Cohort 1 will include participants who have not received any prior systemic therapy for locally advanced or metastatic UC and are eligible to receive platinum-based chemotherapy, whereas Cohort 2 will include participants who have received ≥ 1 prior systemic therapy for locally advanced or metastatic UC.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
956
Inclusion Criteria
  • Life expectancy ≥ 12 weeks.

  • Measurable disease as defined by RECIST v1.1.

  • Histologically or cytologically confirmed locally advanced (unresectable) or metastatic UC of the renal pelvis, ureter, bladder, or urethra.

  • Archival or fresh tumor tissue comprising muscle-invasive UC or locally advanced or metastatic UC should be available for submission to central laboratory.

  • Negative pregnancy test for women of childbearing potential (WOCBP) (negative serum test at Screening and negative urine or serum test within 72 hours prior to the first dose).

  • Cohort 1: Previously Untreated: Eligible to receive platinum-based chemotherapy (either cisplatin- or carboplatin-based chemotherapy based on Investigator decision.

  • Cohort 1: Participants must not have received prior systemic therapy for locally advanced or metastatic UC with the following exceptions:

    1. Prior local intravesical chemotherapy, local surgery when full resection is not achieved, local immunotherapy, and radiotherapy are permitted if completed at least 4 weeks prior to the initiation of study treatment and all acute toxicities have resolved.
    2. Prior neoadjuvant/adjuvant chemotherapy or monomethyl auristatin E (MMAE)-based therapy with recurrence >12 months from completion of therapy.
    3. Prior neoadjuvant/adjuvant immune checkpoint inhibitor therapy with recurrence >12 months from completion of therapy.
  • Cohort 2: Previously Treated: Participants must have received ≥ 1 prior systemic treatment for locally advanced or metastatic UC. This includes neoadjuvant/adjuvant platinum-based chemotherapy if recurrence occurred within 12 months of completing therapy.

  • Cohort 2: Progression or recurrence of UC during or following receipt of most recent therapy.

Key

Exclusion Criteria
  • Active keratitis or corneal ulcerations.
  • Requirement, while on study, for treatment with strong inhibitors or strong inducers of human cytochrome P450 3A (CYP3A) or inhibitors of P-glycoprotein (P-gp) including herbal- or food-based inhibitors.
  • Any condition requiring current treatment with high dose corticosteroids (> 10 mg daily prednisone or equivalent).
  • Known hypersensitivity or allergy to any of the ingredients of any of the study interventions, or to MMAE.
  • Has not adequately recovered from recent major surgery (excluding placement of vascular access).
  • Receipt of live or attenuated vaccine within 30 days of first dose.
  • Cohort 1: Previously Untreated: Prior treatment with a checkpoint inhibitor (CPI) for any other malignancy within the last 12 months.
  • Cohort 2: Previously Treated: Received more than 1 prior platinum-based chemotherapy regimen for locally advanced or metastatic UC. This includes neoadjuvant/adjuvant platinum-based chemotherapy if recurrence occurred within 12 months of completing therapy.
  • Cohort 2: Prior treatment with enfortumab vedotin or any other MMAE-based therapy

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Cohort 1: BT8009 Arm 1PembrolizumabParticipants will receive BT8009 and a standard dose of pembrolizumab.
Cohort 1: BT8009 Arm 1BT8009Participants will receive BT8009 and a standard dose of pembrolizumab.
Cohort 2: BT8009 Arm 1BT8009Participants will receive BT8009.
Cohort 1: Arm 3Gemcitabine + cisplatin Or carboplatinParticipants will receive Platinum-based combination chemotherapy +/- avelumab maintenance
Cohort 1: BT8009 Arm 2BT8009Participants will receive BT8009 and a standard dose of pembrolizumab.
Cohort 2: BT8009 Arm 2BT8009Participants will receive BT8009.
Cohort 2: Arm 3: BT8009 (Not Recruiting)BT8009Participants will receive BT8009 and a standard dose of pembrolizumab.
Cohort 1: BT8009 Arm 2PembrolizumabParticipants will receive BT8009 and a standard dose of pembrolizumab.
Cohort 2: Arm 3: BT8009 (Not Recruiting)PembrolizumabParticipants will receive BT8009 and a standard dose of pembrolizumab.
Cohort 1: Arm 3AvelumabParticipants will receive Platinum-based combination chemotherapy +/- avelumab maintenance
Primary Outcome Measures
NameTimeMethod
Cohort 1: Progression-free survival (PFS) per Response Evaluation Criteria in Solid Tumors, version 1.1 (RECIST v1.1) assessed by blinded central independent review (BICR)Up to approximately 6 years

The time from randomization to date of first documentation of disease progression or death.

Cohort 2: Objective response rate (ORR) per RECIST 1.1 assessed by BICRUp to approximately 6 years

The time from randomization to date of first documentation of disease progression or death.

Secondary Outcome Measures
NameTimeMethod
Cohort 2: PFS per RECIST v1.1 assessed by BICRUp to approximately 6 years

The time from randomization to date of first documentation of disease progression or death.

Cohorts 1 and 2: Number of participants reporting adverse events (AEs) and Serious adverse events (SAEs)Until 30 days post last dose, up to approximately 6 years
Cohorts 1 and 2: DCR per RECIST 1.1 assessed by InvestigatorUp to approximately 6 years

The time from Cycle 1 Day 1 to date of first documentation of disease progression or death

Cohorts 1 and 2: PFS per RECIST v1.1 assessed by InvestigatorUp to approximately 6 years

The time from randomization to date of first documentation of disease progression or death.

Cohorts 1 and 2: ORR per RECIST 1.1 assessed by InvestigatorUp to approximately 6 years

The time from randomization to date of first documentation of disease progression or death.

Cohorts 1 and 2: Overall survival (OS) rateUp to approximately 7 years

The time from randomization to date of death from any cause.

Cohorts 1 and 2: Duration of response (DoR) per RECIST 1.1 assessed by BICRUp to approximately 6 years

The time from time of first documentation of objective response that is subsequently confirmed to date of first documentation of objective tumor progression or death.

Cohorts 1 and 2: DoR per RECIST 1.1 assessed by InvestigatorUp to approximately 6 years

The time from time of first documentation of objective response that is subsequently confirmed to date of first documentation of objective tumor progression or death.

Cohorts 1 and 2: Number of Participants with Clinically Significant Changes in vital signsUntil the end of treatment, up to approximately 6 years
Cohort 1: ORR per RECIST 1.1 assessed by BICRUp to approximately 6 years

The time from randomization to date of first documentation of disease progression or death.

Cohorts 1 and 2: Disease control rate (DCR) per RECIST 1.1 assessed by BICRUp to approximately 6 years

The time from randomization to date of first documentation of disease progression or death.

Cohorts 1 and 2: Number of Participants with Clinically Significant Changes in Laboratory ResultsUntil the end of treatment, up to approximately 6 years
Cohorts 1 and 2: Number of Participants with Clinically Significant Changes in Electrocardiogram (ECG)Until the end of treatment, up to approximately 6 years
Cohorts 1 and 2: Change from Baseline in European Organization for Research and Treatment of Cancer Quality of Life Questionnaire Core 30 (EORTC QLQ-C30)Until the end of treatment, up to approximately 6 years
Cohorts 1 and 2: Change from Baseline in Euroqol-5 Dimensions (EQ-5D) QuestionnaireUntil the end of treatment, up to approximately 6 years

Trial Locations

Locations (169)

University of Arkansas for Medical Sciences

🇺🇸

Little Rock, Arkansas, United States

Virginia K. Crosson Cancer Center at St. Jude Medical Center

🇺🇸

Fullerton, California, United States

University of California - Irvine Medical Center

🇺🇸

Orange, California, United States

Adventist Health St. Helena

🇺🇸

Saint Helena, California, United States

University of California, San Francisco (UCSF)

🇺🇸

San Francisco, California, United States

Rocky Mountain Cancer Center

🇺🇸

Denver, Colorado, United States

Yale University School of Medicine - Yale Cancer Center

🇺🇸

New Haven, Connecticut, United States

Medical Oncology Hematology Consultants

🇺🇸

Newark, Delaware, United States

Cancer Specialists of North Florida

🇺🇸

Jacksonville, Florida, United States

Mount Sinai Medical Center of Florida, Inc.

🇺🇸

Miami Beach, Florida, United States

University of Miami - Sylvester Comprehensive Cancer Center

🇺🇸

Miami, Florida, United States

AP Medical Research

🇺🇸

Miami, Florida, United States

Moffitt

🇺🇸

Tampa, Florida, United States

Southern Illinois University (SIU) - Simmons Cancer Institute

🇺🇸

Springfield, Illinois, United States

Mission Cancer + Blood

🇺🇸

Des Moines, Iowa, United States

University of Kansas Cancer Center

🇺🇸

Westwood, Kansas, United States

UofL Health Brown Cancer Center

🇺🇸

Louisville, Kentucky, United States

Mary Bird Perkins Cancer Center

🇺🇸

Baton Rouge, Louisiana, United States

Princess Margaret Hospital

🇨🇦

Toronto, Canada

Nebraska Cancer Specialists

🇺🇸

Omaha, Nebraska, United States

XCancer Omaha/Urology Cancer Center

🇺🇸

Omaha, Nebraska, United States

Astera Cancer Care

🇺🇸

East Brunswick, New Jersey, United States

Summit Health (New Jersey Urology)

🇺🇸

Voorhees, New Jersey, United States

Montefiore Medical Center

🇺🇸

Bronx, New York, United States

Columbia University Irving Medical Center

🇺🇸

New York, New York, United States

University Hospitals Cleveland Medical Center

🇺🇸

Cleveland, Ohio, United States

Medical University of South Carolina (MUSC) - Hollings Cancer Center

🇺🇸

Charleston, South Carolina, United States

Carolina Urologic Research Center

🇺🇸

Myrtle Beach, South Carolina, United States

SCRI Oncology Partners

🇺🇸

Nashville, Tennessee, United States

The Center for Cancer and Blood Disorders

🇺🇸

Fort Worth, Texas, United States

MD Anderson Cancer Center

🇺🇸

Houston, Texas, United States

University of Texas Health Science Center at San Antonio

🇺🇸

San Antonio, Texas, United States

Centro de Diagnostico Urologico S.R.L.

🇦🇷

Buenos Aires, Argentina

Hospital Britanico de Buenos Aires

🇦🇷

Buenos Aires, Argentina

Hospital Sirio Libanes de Buenos Aires

🇦🇷

Buenos Aires, Argentina

Instituto Alexander Fleming

🇦🇷

Buenos Aires, Argentina

Fundacion Medica Rio Negro y Neuquen

🇦🇷

Cipolletti, Argentina

Centro Medico Privado (CEMAIC)

🇦🇷

Córdoba, Argentina

Fundación CORI para la investigación y Prevención del Cancer

🇦🇷

La Rioja, Argentina

Centro De Investigacion Pergamino S.A.

🇦🇷

Pergamino, Argentina

Instituto de Oncologia de Rosario

🇦🇷

Santa Fe, Argentina

Clinica Viedma S.A.

🇦🇷

Viedma, Argentina

Cancer Research SA

🇦🇺

Adelaide, Australia

Mater Misericordiae Ltd, South Brisbane

🇦🇺

Brisbane, Australia

Townsville Hospital and Health Service

🇦🇺

Douglas, Australia

Barwon Health

🇦🇺

Geelong, Australia

Calvary Mater Newcastle

🇦🇺

Hunter, Australia

Sir Charles Gairdner Hospital

🇦🇺

Nedlands, Australia

Blacktown Hospital

🇦🇺

New South Wales, Australia

Prince of Wales Hospital

🇦🇺

Randwick, Australia

Icon Cancer Centre

🇦🇺

South Brisbane, Australia

Gold Coast University Hospital

🇦🇺

Southport, Australia

Princess Alexandra Hospital

🇦🇺

Woolloongabba, Australia

Urologie und Andrologie Ordensklinikum Linz GmbH Elisabethinen

🇦🇹

Linz, Austria

Krankenhaus der Barmherzigen Brüder Wien

🇦🇹

Wien, Austria

Medizinische Universitaet Wien

🇦🇹

Wien, Austria

ASBL Grand Hôpital de Charleroi (GHdC), Site Notre Dame

🇧🇪

Charleroi, Belgium

General Hospital Maria Middelares

🇧🇪

Gent, Belgium

University Hospital Gent

🇧🇪

Gent, Belgium

Universitaire Ziekenhuizen Leuven

🇧🇪

Leuven, Belgium

Fundacao PIO XII - Hospital de Amor

🇧🇷

Barretos, Brazil

CEPEN - Centro de Pesquisa e Ensino em Oncologia de Santa Catarina

🇧🇷

Florianópolis, Brazil

Oncosite - Centro de Pesquisa Clinica Em Oncologia

🇧🇷

Ijuí, Brazil

Centro Gaucho Integrado de Oncologia, Hematologia, Ensino e Pesquisa

🇧🇷

Porto Alegre, Brazil

Hospital Sao Lucas - Pontificia Universidade Catolica do Rio Grande do Sul (PUCRS)

🇧🇷

Porto Alegre, Brazil

Hospital Alemao Oswaldo Cruz

🇧🇷

São Paulo, Brazil

Hospital A.C. Camargo Cancer Center

🇧🇷

São Paulo, Brazil

British Columbia Cancer Agency- Centre for the Southern Interior

🇨🇦

Kelowna, Canada

McGill University Health Center

🇨🇦

Québec, Canada

Cancer Care Manitoba

🇨🇦

Winnipeg, Canada

Fundación Arturo López Pérez (FALP)

🇨🇱

Santiago, Chile

Centro de Investigacion Clinica Bradford Hill

🇨🇱

Santiago, Chile

Oncocentro APYS

🇨🇱

Viña Del Mar, Chile

Aalborg University Hospital

🇩🇰

Aalborg, Denmark

Service d'Oncologie Medicale - CHRU Besancon

🇫🇷

Besançon, France

Institut Bergonie

🇫🇷

Bordeaux Cedex, France

CHU Bordeaux - Hopital Saint-Andre

🇫🇷

Bordeaux, France

Groupement de Cooperation Sanitaire (GCS) ELSAN - Clinique Victor Hugo

🇫🇷

Le Mans, France

CHU de Limoges - Hopital Dupuytren 1

🇫🇷

Limoges, France

Centre Leon Berard

🇫🇷

Lyon, France

Institut Paoli-Calmettes

🇫🇷

Marseille, France

ICM - Institut Regional du Cancer de Montpellier

🇫🇷

Montpellier Cedex 5, France

Centre d'Oncologie de Gentilly

🇫🇷

Nancy, France

Centre Antoine-Lacassagne

🇫🇷

Nice, France

Institut Mutualiste Montsouris

🇫🇷

Paris, France

AP-HP Hopital Europeen Georges Pompidou

🇫🇷

Paris, France

HCL Centre Hospitalier Lyon Sud

🇫🇷

Pierre-Benite Cedex, France

CHU Poitiers - Pole Regional de Cancerologie de Poitiers (PRC)

🇫🇷

Poitiers, France

Institut Gustave Roussy

🇫🇷

Villejuif, France

LTD High Technology Hospital Medcenter

🇬🇪

Batumi, Georgia

The First University Clinic of Tbilisi State Medical University

🇬🇪

Tbilisi, Georgia

New Vision University Hospital

🇬🇪

Tbilisi, Georgia

Multiprofile Clinic Consilium Medulla LTD

🇬🇪

Tbilisi, Georgia

Universitaetsklinikum Carl Gustav Carus Dresden

🇩🇪

Dresden, Germany

Universitaetsklinikum Essen

🇩🇪

Essen, Germany

Krankenhaus Nordwest GmbH

🇩🇪

Frankfurt, Germany

Universitaetsklinikum Frankfurt - Klinikum der Johann Wolfgang Goethe Universitaet

🇩🇪

Frankfurt, Germany

Universitaetsklinikum Freiburg

🇩🇪

Freiburg, Germany

Georg-August-Universitaet Goettingen Stiftung oeffentlichen Rechts Universitaetsmedizin Goettingen

🇩🇪

Göttingen, Germany

Marien Hospital Herne - Universitaetsklinikum der Ruhr-Universitaet Bochum

🇩🇪

Herne, Germany

Universitaetsmedizin Mannheim

🇩🇪

Mannheim, Germany

Universitaetsklinikum Muenster

🇩🇪

Münster, Germany

Studienpraxis Urologie

🇩🇪

Nürtingen, Germany

Universitaetsklinikum Tuebingen

🇩🇪

Tübingen, Germany

Orszagos Onkologiai Intezet

🇭🇺

Budapest, Hungary

Budapesti Uzsoki Utcai Korhaz

🇭🇺

Budapest, Hungary

Somogy Varmegyei Kaposi Mor Oktato Korhaz

🇭🇺

Kaposvár, Hungary

Bacs-Kiskun Varmegyei Oktatokorhaz

🇭🇺

Kecskemét, Hungary

Shamir Medical Center

🇮🇱

Be'er Ya'aqov, Israel

Rambam Health Care Campus

🇮🇱

Haifa, Israel

Hadassah Hebrew University Medical Center

🇮🇱

Jerusalem, Israel

Meir Medical Center

🇮🇱

Kfar Saba, Israel

Rabin Medical Center - Beilinson Hospital

🇮🇱

Petach Tikva, Israel

Sourasky Medical Center

🇮🇱

Tel Aviv, Israel

Centro Riferimento Oncologico - Aviano

🇮🇹

Aviano, Italy

Ospedale Policlinico San Martino IRCCS

🇮🇹

Genova, Italy

Istituto Europeo di Oncologia

🇮🇹

Milano, Italy

Istituto Nazionale Tumori IRCCS "Fondazione G. Pascale"

🇮🇹

Napoli, Italy

Azienda Ospedaliera Santa Maria di Terni

🇮🇹

Terni, Italy

Chungnam National University Hospital

🇰🇷

Daejeon, Korea, Republic of

National Cancer Center

🇰🇷

Goyang, Korea, Republic of

Chonnam National University Hwasun Hospital

🇰🇷

Gwangju, Korea, Republic of

Korea University Anam Hospital

🇰🇷

Seoul, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Asan Medical Center

🇰🇷

Seoul, Korea, Republic of

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

Severance Hospital, Yonsei University Health System

🇰🇷

Seoul, Korea, Republic of

Copernicus PL Sp. z o.o., Wojewodzkie Centrum Onkologii

🇵🇱

Gdańsk, Poland

Spitale Pomorskie Sp.z.o.o ODDZIAL ONKOLOGII KLINICZNEJ

🇵🇱

Gdynia, Poland

SCM Sp. z o.o.

🇵🇱

Kraków, Poland

Mazowiecki Szpital Onkologiczny

🇵🇱

Wieliszew, Poland

University Clinical Center of Serbia, Clinic of Urology

🇷🇸

Belgrade, Serbia

National University Hospital

🇸🇬

Singapore, Singapore

National Cancer Centre Singapore

🇸🇬

Singapore, Singapore

Hospital de la Santa Creu i Sant Pau

🇪🇸

Barcelona, Spain

Hospital Clinic Barcelona

🇪🇸

Barcelona, Spain

Institut Catala d'Oncologia - L'Hospitalet

🇪🇸

Barcelona, Spain

Hospital Universitario Insular de Gran Canaria

🇪🇸

Las Palmas De Gran Canaria, Spain

Hospital General Universitario Gregorio Maranon

🇪🇸

Madrid, Spain

Clinica Universidad de Navarra - Madrid

🇪🇸

Madrid, Spain

Hospital Fundacion Jimenez Diaz

🇪🇸

Madrid, Spain

Hospital Universitario 12 de Octubre

🇪🇸

Madrid, Spain

Hospital Universitario La Paz

🇪🇸

Madrid, Spain

Clinica Universidad de Navarra - Pamplona

🇪🇸

Pamplona, Spain

Hospital Universitario Donostia

🇪🇸

San Sebastián, Spain

Hospital Universitario Marques de Valdecilla

🇪🇸

Santander, Spain

Hospital Clinico Universitario de Santiago

🇪🇸

Santiago De Compostela, Spain

Instituto Valenciano de Oncologia

🇪🇸

Valencia, Spain

Kaohsiung Medical University Chung-Ho Memorial Hospital

🇨🇳

Kaohsiung, Taiwan

China Medical University Hospital

🇨🇳

Taichung, Taiwan

National Cheng Kung University Hospital

🇨🇳

Tainan, Taiwan

Chi Mei Medical Center

🇨🇳

Tainan, Taiwan

National Taiwan University Hospital

🇨🇳

Taipei, Taiwan

Linkou Chang Gung Memorial Hospital (CGMHLK)

🇨🇳

Taoyuan city, Taiwan

Liv Hospital Ankara

🇹🇷

Ankara, Turkey

Trakya University Medical Faculty

🇹🇷

Edirne, Turkey

Goztepe Prof. Dr. Suleyman Yalcin City Hospital

🇹🇷

Istanbul, Turkey

Istinye Universitesi VM Medical Park Pendik Hastanesi

🇹🇷

Istanbul, Turkey

Medical Point Izmir Hospital

🇹🇷

İzmir, Turkey

Kocaeli University Faculty of Medicine

🇹🇷

Kocaeli, Turkey

Bristol Haematology and Oncology Centre

🇬🇧

Bristol, United Kingdom

Addenbrooke's Hospital

🇬🇧

Cambridge, United Kingdom

St. Bartholomew's Hospital

🇬🇧

London, United Kingdom

University College London Hospital

🇬🇧

London, United Kingdom

Royal Free London NHS Foundation Trust

🇬🇧

London, United Kingdom

Charing Cross Hospital

🇬🇧

London, United Kingdom

The Christie NHS Foundation Trust

🇬🇧

Manchester, United Kingdom

Derriford Hospital

🇬🇧

Plymouth, United Kingdom

The Royal Marsden Hospital

🇬🇧

Sutton, United Kingdom

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