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Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Atrosimab (ATM001) in Healthy Volunteers

Phase 1
Completed
Conditions
Healthy Volunteers
Registration Number
NCT04650126
Lead Sponsor
Baliopharm Pty Ltd
Brief Summary

This is a double-blind, parallel group and placebo-controlled clinical study to assess safety tolerability, pharmacokinetics and pharmacodynamics of Atrosimab in healthy volunteers

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
42
Inclusion Criteria
  • healthy male subjects
  • body mass index 18-32 kg/m2
  • normal physical examination, clinical laboratory values and ECG
  • additional inclusion criteria apply
Exclusion Criteria
  • febrile or infectious illness at least 7 days prior to the first administration
  • any active physical disease, acute or chronic
  • history of alcohol or drug abuse
  • history of chronic or recurrent metabolic, renal, hepatic, pulmonary, gastrointestinal, neurological, endocrinological, immunological, psychiatric, or cardio-vascular disease, myopathies and bleeding tendency
  • additional exclusion criteria apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Primary Outcome Measures
NameTimeMethod
Any adverse event, serious adverse event (SAE)4 weeks
PK: Area under the plasma concentration curve from administration until the last quantifiable sampling point (AUC 0-t)8 days
PK: Apparent terminal elimination rate constant (λz)8 days
PK: Apparent volume of distribution (Vz)8 days
PK: Maximum Plasma Concentration [Cmax]8 days
PK: Clearance (CL)8 days
pharmacokinetic (PK): Area under the analyte concentration-time curve from time 0 and extrapolated to infinite time (AUC 0-∞)8 days
PK: Terminal half life (t1/2)8 days
PK: Mean residence time (MRT)8 days
Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (1)

Q-Pharm

🇦🇺

Herston, Brisbane, Australia

Q-Pharm
🇦🇺Herston, Brisbane, Australia

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