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Safety, Tolerability and Relative Bioavailability Study of BMS-986195 in Healthy Subjects

Phase 1
Completed
Conditions
Rheumatoid Arthritis
Interventions
Other: Placebo
Registration Number
NCT02705989
Lead Sponsor
Bristol-Myers Squibb
Brief Summary

The purpose of this study is to evaluate the safety profile, tolerability, pharmacokinetics, and pharmacodynamics following single and multiple ascending oral doses of BMS-986195 in healthy subjects, and to assess the relative bioavailability of two formulations of BMS-986195 with or without food.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
439
Inclusion Criteria
  • Body Mass Index(BMI) of 18 to 32 kilograms/meter^2
  • Healthy male and female, first generation Japanese with confirmed paternal and maternal Japanese ancestry, 18-55 years old, whose residency outside of Japan does not exceed 10 years with a BMI of 18-30 kilograms/meter^2 inclusive.
  • Women must not be pregnant or breastfeeding
  • Women of Childbearing Potential (WOCBP) must agree to follow instructions for method(s) of contraception for the duration of treatment with study drug plus 14 days or longer if required.
  • Males who are sexually active with WOCBP must agree to follow instructions for method(s) of contraception for the duration of treatment with study drug plus 14 days or longer if required.
Exclusion Criteria
  • Any significant acute or chronic medical illness
  • Known or suspected autoimmune disorder, including but not limited to rheumatoid arthritis, fibromyalgia, systemic lupus erythematosis, polymyalgia rheumatica, giant cell arteritis, Behcet's disease, dermatomyositis, multiple sclerosis, moderate to severe asthma, any autoimmune vasculitis, autoimmune hepatitis, or any other active autoimmune disease for which a subject requires medical follow-up or medical treatment
  • Any history of known or suspected congenital or acquired immunodeficiency state or condition that would compromise the subject's immune status (example: history of splenectomy)
  • Presence of any factors that would predispose the subject to develop infection e.g., rectal fissures, poor dentition, open skin lesions, and presence of preexisting skin conditions that increase risks for injection site complications e.g. Behcet's Disease, Psoriasis, pustular dermatoses
  • Any history or risk for tuberculosis (TB)

Other protocol defined inclusion/exclusion criteria could apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Multiple Ascending Dose(MAD)PlaceboMultiple ascending dose of BMS-986195 or Placebo matching BMS-986195
Single Ascending Dose (SAD)PlaceboSingle ascending dose of BMS-986195 or Placebo matching BMS-986195
Japanese-Multiple Ascending Dose(MAD)PlaceboMultiple ascending dose of BMS-986195 or Placebo matching BMS-986195 in subjects with Japanese heritage
Single Ascending Dose (SAD)BMS-986195Single ascending dose of BMS-986195 or Placebo matching BMS-986195
Japanese-Multiple Ascending Dose(MAD)BMS-986195Multiple ascending dose of BMS-986195 or Placebo matching BMS-986195 in subjects with Japanese heritage
Multiple Ascending Dose(MAD)BMS-986195Multiple ascending dose of BMS-986195 or Placebo matching BMS-986195
Relative Bioavailability with Food Effects (Open Label)BMS-986195-
Primary Outcome Measures
NameTimeMethod
Safety and tolerability of single oral dose of BMS-986195 as determined by medical review of adverse event reports, vital sign measurements, electrocardiograms (ECGs), and results of physical examination and laboratory testsUp to 8 days during and after last dose
Safety and tolerability of multiple oral doses of BMS-986195 as determined by medical review of adverse event reports, vital sign measurements, electrocardiograms (ECGs), and results of physical examination and laboratory testsUp to 21 days during and after last dose
Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (1)

Local Institution

🇦🇺

Melbourne, Victoria, Australia

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