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Clinical Trials/NL-OMON48728
NL-OMON48728
Completed
Not Applicable

A single center, randomized study investigating the safety, tolerability, and pharmacokinetics of AZ-009 (Staccato apomorphine) in healthy volunteers and the safety, tolerability, pharmacokinetics, and pharmacodynamics of AZ-009 in subjects with established Parkinson*s Disease. - SAD study of AZ-009 in HV and PD patients

Alexza Pharmaceuticals Inc.0 sites56 target enrollmentTBD

Overview

Phase
Not Applicable
Intervention
Not specified
Conditions
Parkinson's disease
Sponsor
Alexza Pharmaceuticals Inc.
Enrollment
56
Status
Completed
Last Updated
2 years ago

Overview

Brief Summary

No summary available.

Registry
who.int
Start Date
TBD
End Date
TBD
Last Updated
2 years ago
Study Type
Interventional

Investigators

Eligibility Criteria

Inclusion Criteria

  • \* Healthy adult males and females between 18 and 60 years of age, inclusive at the time of signing the informed consent document.
  • \* Female subjects, who are:
  • o Surgically sterile (including bilateral tubal ligation) for at least 3 months prior to screening
  • o Postmenopausal, defined as 1 of the following:
  • \* Last menstrual sequence greater than 12 months prior to screening
  • \* Last menstrual sequence greater than 6 months prior to screening and a serum follicle\-stimulating hormone (FSH) concentration \> 40 mIU/mL
  • o Of childbearing potential (i.e. do not meet the criteria outlined above); subjects must:
  • \* Have a negative urine pregnancy test at Screening and Day \-1, as verified by the study doctor prior to starting study therapy.
  • \* Either commit to true abstinence from heterosexual contact or agree to use, and be able to comply with, effective contraception without interruption with one of the following methods during the study participation up until 90 days after administration of study drug:
  • \* Oral contraceptive medications

Exclusion Criteria

  • \* Any significant medical condition, psychiatric illness or history of depression that could, in the investigator\*s opinion, compromise the subject\*s safety or interfere with the completion of this protocol.
  • \* Any condition including the presence of laboratory abnormalities, which according to the investigator places the subject at unacceptable risk if he/she were to participate in the study.
  • \* Any condition that according to the investigator confounds the ability to interpret data from the study such as a virus, seasonal allergy, concurrent skin rash, etc. on screening or prior to drug treatment phase that may be difficult to discern from further health status changes from an investigational product.
  • \* History of clinically significant central nervous system (e.g., seizures), cardiac, pulmonary (e.g., asthma, COPD), metabolic, renal, hepatic, or gastrointestinal (GI) conditions including gastric bypass or other weight loss surgical procedure; or history of such conditions that, in the opinion of the investigator, may place the subject at an unacceptable risk as a participant in this trial, may interfere with the interpretation of safety and/or tolerability data obtained in the trial, or may interfere with the absorption, distribution, metabolism, or excretion of the study drugs.
  • \* Use of 5HT3 antagonists, drugs known to prolong QTc and use of antihypertensives.
  • \* PR interval \> 220 msec or QRS duration \> 120 msec or QTcF interval \> 450 msec for men and 470 msec for women obtained at screening visit or prior to the first dose of study drug.
  • \* Aspartate transaminase (AST), alanine transaminase (ALT), gamma\-glutamyl transferase (GGT), serum creatinine, or total bilirubin \> 1\.5 upper limit of normal (ULN) at screening or prior to the first dose of study drug. These laboratory tests may be repeated once, if they are abnormal on first screening, and if there is a medical reason to believe the results may be inaccurate. If the repeat test is within the reference range, the subject may be included only if the investigator considers that the previous finding will not compromise the subject\*s safety and will not interfere with the interpretation of safety data.
  • \* Use of non\-prescription medications, including herbal and dietary supplements within 5 days or 5 half\-lives (whichever is longer) prior to the first dose of study drug, (The subject may take paracetamol (\* 2 grams/day) or ibuprofen (\* 1600 mg/day) for up to 48 hours prior to the first dose of study drug. Females may take oral contraceptives. The investigator and study team may review medication use on a case\-by\-case basis to determine if its use would compromise subject safety or interfere with study procedures or data interpretation.
  • \* Use of medication that is inhibitor or inducer of CYP450\-3A4/5 within 3 days of dosing and during the course of the study.
  • \* Consumption of grapefruit, grapefruit juice, star fruit, oranges, orange juice, Seville oranges within 3 days prior to administration of study drug.

Outcomes

Primary Outcomes

Not specified

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