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A Study of SHR-A1811 in Subjects With Advanced Malignant Solid Tumors

Phase 1
Recruiting
Conditions
Advanced Solid Tumors
Interventions
Registration Number
NCT04446260
Lead Sponsor
Jiangsu HengRui Medicine Co., Ltd.
Brief Summary

This is an open-label, two-part study to evaluate the safety, tolerability, pharmacokinetics and immunogenicity of SHR-A1811 and preliminary anti-tumor efficacy in HER2 expressing or mutated advanced malignant solid tumor subjects.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
226
Inclusion Criteria
  • Advanced/unresectable or metastatic solid tumor with HER2 expression or mutation that is refractory to or intolerable with standard treatment, or for which no standard treatment is available
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
  • LVEF β‰₯ 50% by either ECHO or MUGA
  • Has adequate renal and hepatic function
  • Female subjects agree not to be pregnant or lactating from beginning of the study screening until 6 months after receiving the last treatment
Exclusion Criteria
  • History of clinically significant lung diseases (e.g., interstitial pneumonia, pneumonitis, pulmonary fibrosis, and severe radiation pneumonitis) or suspected to have these diseases by imaging at screening period
  • Known hereditary or acquired bleeding and thrombotic tendency

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Part 1 Dose escalationSHR-A1811-
Part 2 PK expansionSHR-A1811-
Part 3 Indication expansionSHR-A1811-
Primary Outcome Measures
NameTimeMethod
Incidence and severity of adverse events (AEs)From Day1 to 90 days after last dose

Frequency and seriousness of treatment emergent adverse events (TEAEs)

Secondary Outcome Measures
NameTimeMethod
Tumor response using RECIST 1.1From first dose to disease progression or death, whichever comes first, up to 30 months

RECIST=Response Evaluation Criteria in Solid Tumors Assessment of tumor response until disease progression or death to evaluate the efficacy of SHR-A1811 up to 30 months

PK parameter: Tmax of SHR-A1811Through study completion, an average of 1 year

Time to maximal concentration (Tmax) of SHR-A1811

Immunogenicity of SHR-A1811Through study completion, an average of 1 year

Including anti-drug antibody and/or neutralizing antibody

PK parameter: AUC0-t of SHR-A1811Through study completion, an average of 1 year

AUC computed from time zero to the time of the last quantifiable concentration (AUC0-t) of SHR-A1811

PK parameter: Cmax of SHR-A1811Through study completion, an average of 1 year

Maximal concentration (Cmax) of SHR-A1811

Trial Locations

Locations (35)

Gabrail Cancer Center

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Canton, Ohio, United States

Seoul National University Hospital

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Seoul, Korea, Republic of

Macquarie University Hospital

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Macquarie, New South Wales, Australia

Sun Yat-Sen Memorial Hospital, Sun Yat-sen University

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Guangzhou, Guangdong, China

Shengjing Hospital of China medical university

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Shengyang, Liaoning, China

The second affiliated hospital Zhejiang university school of medicine

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Hangzhou, Zhejiang, China

Fudan University Shanghai cancer center

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Shanghai, Shanghai, China

National Cheng Kung University Hospital

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Tainan, Taiwan

Hunan cancer hospital

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Changsha, Hunan, China

The First Hospital of Jilin University

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Changchuan, Jilin, China

Sichuan Cancer Hospital

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Chengdu, Sichuan, China

Tianjin medical university cancer institute&hoospital

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Tianjin, Tianjin, China

Chang Gung Memorial Hospital, Linkou

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Taoyuan, Taiwan

Prisma-Health Cancer Institute

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Greenville, South Carolina, United States

Xiangya hospital central south university

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Changsha, Hunan, China

China Medical University Hospital

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Taichung, Taiwan

Asan Medical Center

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Seoul, Korea, Republic of

Hubei cancer hospital

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Wuhan, Hubei, China

Greenville Hospital System

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Greenville, South Carolina, United States

The first affiliated hospital of bengbu medical college

πŸ‡¨πŸ‡³

Bengbu, Anhui, China

Henan cancer Hospital

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Zhengzhou, Henan, China

Seoul National University Bundang Hospital

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Seongnam, Gyeonggi-do, Korea, Republic of

Fudan Unversity Zhongshan Hospital

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Shanghai, Shanghai, China

Zhongnan hospital of Wuhan university

πŸ‡¨πŸ‡³

Wuhan, Hubei, China

Nanjing Drum Tower Hospital

πŸ‡¨πŸ‡³

Nanjing, Jiangsu, China

Montefiore-Einstein Center for Cancer Care

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Bronx, New York, United States

Mary Crowley Cancer Research

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Dallas, Texas, United States

Center for Oncology and Blood Disorders

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Houston, Texas, United States

Nucleus Network

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Melbourne, Victoria, Australia

Nanfang Hospital

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Guangzhou, Guangdong, China

Zhejiang provincial people's hospital

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Hangzhou, Zhejiang, China

Alfred Hospital

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Melbourne, Australia

Southern Oncology Clinical Research Unit

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Bedford Park, South Australia, Australia

Cancer Hospital Chinese Academy of Medical Sciences

πŸ‡¨πŸ‡³

Beijing, Beijing, China

Peninsula and South Eastern Haematology & Oncology Group

πŸ‡¦πŸ‡Ί

Frankston, Victoria, Australia

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