MedPath

Targeting ER Stress in Vascular Dysfunction

Early Phase 1
Terminated
Conditions
Vasodilation
Arterial Stiffness
Interventions
Registration Number
NCT04001647
Lead Sponsor
Colorado State University
Brief Summary

Aging and obesity are both risk factors for cardiovascular disease (CVD). One process that links both of these conditions to CVD is vascular dysfunction. Data from animal studies indicate that endoplasmic reticulum (ER) stress may play an important role in the development of endothelial dysfunction in aging and obesity. Therefore, the goal of this study is to investigate the relative contributions of aging and obesity on vascular dysfunction and ER stress. Additionally, this study will determine if taking an oral supplement for 8 weeks will improve vascular dysfunction and ER stress. Results from this study have the potential to identify a safe treatment option for improving vascular function in aging and obese populations.

Detailed Description

Aging is the primary risk factor for cardiovascular disease (CVD). One critical process that links aging to CVD is the development of vascular dysfunction, characterized by endothelial dysfunction and arterial stiffness. Both endothelial dysfunction and arterial stiffness predict cardiovascular events in older individuals. Aging often coincides with obesity, another independent risk factor for CVD. Although vascular function is well characterized in both aging and obesity, it's unclear how these two conditions interact to modulate vascular function, and whether the combination of aging and obesity has additive or compounding effects on endothelial dysfunction and arterial stiffness.

Currently, it is unknown whether vascular dysfunction is driven by the same underlying cellular mechanisms in aging and obesity. Accumulating data in experimental animals suggest that ER stress may be an important factor in aging- and obesity-related vascular dysfunction. Additionally, middle-aged and older obese adults with endothelial dysfunction display evidence of ER stress within biopsied endothelial cells. In light of these data, the overall goal of this proposal is to test the hypothesis that ER stress is associated with human vascular dysfunction in the settings of aging and obesity, and to determine the efficacy of the chemical chaperone tauroursodeoxycholic acid (TUDCA), an established inhibitor of ER stress, to reduce endothelial cell ER stress and improve vascular function in these at-risk individuals. Results from this study have the potential to identify a novel, safe, and clinically relevant intervention strategy for the treatment of vascular dysfunction in an aging population at high-risk for the development of CVD.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
17
Inclusion Criteria
  • Young, healthy weight adults (age: 18-35; BMI 18.5-24.9 kg/m2)
  • Young, obese adults (age: 18-35; BMI 30- 39.9 kg/m2)
  • Older, healthy weight adults (age: 60-80; 18.5-24.9 kg/m2)
  • Older, obese adults (age: 60-80; 30-39.9 kg/m2)
Exclusion Criteria
  • blood pressure >140/90 mmHg
  • triglycerides >500 mg/dL or LDL cholesterol >190 mg/dL
  • current smoking or history of smoking in the last 12 months
  • diagnosed chronic disease including cancer, cardiovascular, diabetes, kidney, liver, and pancreatic disease
  • weight change >3 kg in the past 3 months or actively trying to lose weight
  • >12 alcoholic drinks/week
  • hormone replacement therapy

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
TUDCASodium NitroprussideYoung and older healthy weight and obese participants will visit the lab for assessment of vascular function prior to the intervention. Aortic stiffness will be evaluated non-invasively using carotid-femoral pulse-wave velocity. A physician will place a catheter in the brachial artery for endothelial cell biopsies and local vasodilator infusions. A venous catheter will also be placed for the systemic ascorbic acid infusion. Aortic stiffness measures and vascular responses to vasodilator infusions will be performed before and after the ascorbic acid infusion. Following the completion of the vascular assessments, participants will receive 1750 mg/day of the dietary supplement tauroursodeoxycholic acid (TUDCA) for 8 weeks. Participants will return to the lab after the 8 week intervention and the vascular assessments described above will be repeated.
PlaceboSodium NitroprussideOlder obese participants will visit the lab for assessment of vascular function prior to the intervention. Aortic stiffness will be evaluated non-invasively using carotid-femoral pulse-wave velocity. A physician will place a catheter in the brachial artery for endothelial cell biopsies and local vasodilator infusions. A venous catheter will also be placed for the systemic ascorbic acid infusion. Aortic stiffness measures and vascular responses to vasodilator infusions will be performed before and after the ascorbic acid infusion. Following the completion of the vascular assessments, participants will receive oral capsules containing a placebo treatment for 8 weeks. Participants will return to the lab after the 8 week intervention and the vascular assessments described above will be repeated.
TUDCAAscorbic AcidYoung and older healthy weight and obese participants will visit the lab for assessment of vascular function prior to the intervention. Aortic stiffness will be evaluated non-invasively using carotid-femoral pulse-wave velocity. A physician will place a catheter in the brachial artery for endothelial cell biopsies and local vasodilator infusions. A venous catheter will also be placed for the systemic ascorbic acid infusion. Aortic stiffness measures and vascular responses to vasodilator infusions will be performed before and after the ascorbic acid infusion. Following the completion of the vascular assessments, participants will receive 1750 mg/day of the dietary supplement tauroursodeoxycholic acid (TUDCA) for 8 weeks. Participants will return to the lab after the 8 week intervention and the vascular assessments described above will be repeated.
PlaceboAscorbic AcidOlder obese participants will visit the lab for assessment of vascular function prior to the intervention. Aortic stiffness will be evaluated non-invasively using carotid-femoral pulse-wave velocity. A physician will place a catheter in the brachial artery for endothelial cell biopsies and local vasodilator infusions. A venous catheter will also be placed for the systemic ascorbic acid infusion. Aortic stiffness measures and vascular responses to vasodilator infusions will be performed before and after the ascorbic acid infusion. Following the completion of the vascular assessments, participants will receive oral capsules containing a placebo treatment for 8 weeks. Participants will return to the lab after the 8 week intervention and the vascular assessments described above will be repeated.
TUDCAAcetylcholineYoung and older healthy weight and obese participants will visit the lab for assessment of vascular function prior to the intervention. Aortic stiffness will be evaluated non-invasively using carotid-femoral pulse-wave velocity. A physician will place a catheter in the brachial artery for endothelial cell biopsies and local vasodilator infusions. A venous catheter will also be placed for the systemic ascorbic acid infusion. Aortic stiffness measures and vascular responses to vasodilator infusions will be performed before and after the ascorbic acid infusion. Following the completion of the vascular assessments, participants will receive 1750 mg/day of the dietary supplement tauroursodeoxycholic acid (TUDCA) for 8 weeks. Participants will return to the lab after the 8 week intervention and the vascular assessments described above will be repeated.
PlaceboAcetylcholineOlder obese participants will visit the lab for assessment of vascular function prior to the intervention. Aortic stiffness will be evaluated non-invasively using carotid-femoral pulse-wave velocity. A physician will place a catheter in the brachial artery for endothelial cell biopsies and local vasodilator infusions. A venous catheter will also be placed for the systemic ascorbic acid infusion. Aortic stiffness measures and vascular responses to vasodilator infusions will be performed before and after the ascorbic acid infusion. Following the completion of the vascular assessments, participants will receive oral capsules containing a placebo treatment for 8 weeks. Participants will return to the lab after the 8 week intervention and the vascular assessments described above will be repeated.
Primary Outcome Measures
NameTimeMethod
Endothelium-independent vasodilationChange in baseline vasodilation at 8 weeks

Blood flow response to increasing doses of sodium nitroprusside

Aortic stiffnessChange in baseline pulse-wave velocity at 8 weeks

Carotid-femoral pulse-wave velocity

Endothelial cell oxidative stress marker p47phoxChange in baseline endothelial p47phox at 8 weeks

Protein expression of nicotinamide adenine dinucleotide phosphate (NADPH) oxidase subunit p47phox

Endothelial cell oxidative stress marker MnSODChange in baseline endothelial MnSOD at 8 weeks

Protein expression of manganese superoxide dismutase (MnSOD)

Endothelial cell oxidative stress marker CuZnSODChange in baseline endothelial CuZnSOD at 8 weeks

Protein expression of copper-zinc SOD (CuZnSOD)

Endothelial cell ER stress marker IRE1αChange in baseline endothelial IRE1α at 8 weeks

Protein expression of inositol-requiring ER-to-nucleus signaling protein 1(IRE1α)

Endothelium-dependent vasodilationChange in baseline vasodilation at 8 weeks

Blood flow response to increasing doses of acetycholine

Endothelial cell inflammatory marker p65Change in baseline endothelial p65 at 8 weeks

Protein expression of nuclear factor kappa B phosphorylated p65 subunit

Endothelial cell inflammatory marker IL-6Change in baseline endothelial IL-6 at 8 weeks

Protein expression of interleukin-6 (IL-6)

Endothelial cell ER stress marker ATF6Change in baseline endothelial ATF6 at 8 weeks

Protein expression of activating transcription factor 6 (ATF6)

Endothelial cell ER stress marker GRP78Change in baseline endothelial GRP78 at 8 weeks

Protein expression of glucose-regulated protein 78 (GRP78)

Endothelial cell ER stress marker GADD34Change in baseline endothelial GADD34 at 8 weeks

Protein expression of growth arrest and DNA damage-inducible 34 (GADD34)

Endothelial cell oxidative stress marker NTChange in baseline endothelial NT at 8 weeks

Protein expression of nitrotyrosine (NT)

Endothelial cell inflammatory marker IκBαChange in baseline endothelial IκBα at 8 weeks

Protein expression of phosphorylated inhibitor of kappa B (IκBα)

Endothelial cell ER stress marker PERKChange in baseline endothelial PERK at 8 weeks

Protein expression of RNA-dependent protein kinase- like ER eukaryotic initiation factor-2α kinase (PERK)

Endothelial cell ER stress marker CHOPChange in baseline endothelial CHOP at 8 weeks

Protein expression of CCAAT-enhancer-binding protein homologous protein (CHOP)

Endothelial cell inflammatory marker TNFαChange in baseline endothelial TNFα at 8 weeks

Protein expression of tumor necrosis factor-alpha (TNFα)

Secondary Outcome Measures
NameTimeMethod
Circulating CRPChange in baseline CRP at 8 weeks

Blood levels of C-reactive protein (CRP)

Circulating triglyceridesChange in baseline triglycerides at 8 weeks

Blood levels of triglycerides

Circulating IL-6Change in baseline IL-6 at 8 weeks

Blood levels of interleukin (IL)-6

Circulating IL-10Change in baseline IL-10 at 8 weeks

Blood levels of interleukin (IL)-10

Circulating TNFαChange in baseline TNFα at 8 weeks

Blood levels of tumor necrosis factor-alpha (TNFα)

Circulating insulinChange in baseline insulin at 8 weeks

Blood levels of insulin

Circulating IL-1βChange in baseline IL-1β at 8 weeks

Blood levels of interleukin (IL)-1 beta (β)

Circulating glucoseChange in baseline blood glucose at 8 weeks

Blood glucose

Circulating cholesterolChange in baseline total cholesterol, LDL cholesterol, and HDL cholesterol at 8 weeks

Blood levels of total cholesterol, LDL cholesterol, and HDL cholesterol

Circulating IL-18Change in baseline IL-18 at 8 weeks

Blood levels of interleukin (IL)-18

Trial Locations

Locations (1)

Colorado State University

🇺🇸

Fort Collins, Colorado, United States

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