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Preoperative Window Opportunity Study With Giredestrant or Tamoxifen in Premenopausal Women With ER+/HER2[-] & Ki67≥10%

Phase 2
Completed
Conditions
Breast Cancer
Breast Cancer, Early-Onset
Interventions
Registration Number
NCT05659563
Lead Sponsor
MedSIR
Brief Summary

This study is a window of opportunity clinical trial to evaluate the efficacy of giredestrant (GDC-9545) or tamoxifen in estrogen receptor-positive (ER\[+\])/human epidermal growth factor receptor 2-negative (HER2\[-\]) primary invasive adenocarcinoma of the breast with Ki67 level ≥ 10%.

A total of 92 patients will be enrolled in this trial and randomized 1:1 in the arm A with giredestrant (GDC-9545) and the arm B with tamoxifen, with a total duration of treatment of 15 days.

This study will analyze the efficacy of giredestrant (GDC-9545) as determined by Ki67 expression between baseline tumor biopsy samples and post-treatment biopsy samples.

Detailed Description

This is a multicenter, international, open-label, two-arms, one stage, phase II, preoperative window of opportunity clinical trial to evaluate the efficacy of giredestrant (GDC-9545) as single agent in ER\[+\]/HER2\[-\] early breast cancer patients with Ki67 ≥ 10%.

Upon meeting all selection criteria, 92 patients enrolled in the study will receive either giredestrant (GDC-9545) 30 mg or tamoxifen .

A total of 92 patients will be enrolled as follows:

* 46 patients in the investigational Arm A will receive giredestrant \[GDC-9545\] 30 mg. It will be administered orally once a day during 15 days.

* 46 patients in the control Arm B will receive tamoxifen 20 mg. It will be administered orally once a day during 15 days.

Patients can take both treatments at home.

The main objective is to analyze the efficacy of giredestrant (GDC-9545) according to changes in tumor cell proliferation. This analysis will compare absolute changes for Ki67 expression between baseline score and the evaluation after 15 days of treatment.

Total study duration is 15 days of treatment and until 28 days after the last dose of the study treatment (or discontinuation) of follow up.

Recruitment & Eligibility

Status
COMPLETED
Sex
Female
Target Recruitment
92
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Arm BTamoxifenTamoxifen: 20mg, orally (PO), daily (QD) during 15 days
Arm AGiredestrantGiredestrant (GDC-9545): 30mg, orally (PO), daily (QD) during 15 days
Primary Outcome Measures
NameTimeMethod
Change in proliferative index (Ki67 expression)Baseline up to 15 days

To assess changes in tumor cell proliferation as measured by Ki67 expression between baseline and D15 (+1 day) post-treatment tumor biopsy samples by central assessment in patients with centrally confirmed Ki67 ≥10% (Arm A: giredestrant vs Arm B: tamoxifen)

Secondary Outcome Measures
NameTimeMethod
Complete cell cycle arrest (CCCA)Baseline up to 15 days

To measure complete cell cycle arrest in all arms, defined as the percentage of participants with centrally assessed Ki67 scores ≤2.7% stained nuclei upon treatment

Changes in molecular profiles of tumor tissue samplesBaseline up to 15 days

To analyze gene expression profiles in tumor tissue samples obtained at baseline and after treatment using the HTG EdgeSeq Oncology Biomarker Panel

Changes in expression levels of estrogen receptor and progesterone receptor in tumor tissue samplesBaseline up to 15 days

To analyze the expression of estrogen receptor and progesterone receptor in tumor tissue samples obtained at baseline and post-therapy

Trial Locations

Locations (18)

Hôpital Tenon AP-HP

🇫🇷

Paris, France

Hopital Europeen Georges Pompidou

🇫🇷

Paris, France

Institut Català d' Oncologia Badalona

🇪🇸

Badalona, Barcelona, Spain

Hospital Universitari Sant Joan de Reus

🇪🇸

Reus, Tarragona, Spain

Hospital General Universitario Dr. Balmis

🇪🇸

Alicante, Spain

Hospital Clínic i Provincial de Barcelona

🇪🇸

Barcelona, Spain

Hospital Universitari Dexeus

🇪🇸

Barcelona, Spain

Hospital Universitario Reina Sofía

🇪🇸

Cordoba, Spain

Hospital Universitario Clínico San Cecilio de Granada

🇪🇸

Granada, Spain

Hospital Universitario de León

🇪🇸

León, Spain

Hospital Beata Maria Ana

🇪🇸

Madrid, Spain

Hospital Universitario La Paz

🇪🇸

Madrid, Spain

Hospital Universitario Ramón y Cajal

🇪🇸

Madrid, Spain

Hospital Clínico Universitario Virgen de la Arrixaca

🇪🇸

Murcia, Spain

Hospital Universitario Virgen del Rocío

🇪🇸

Sevilla, Spain

Hospital Arnau de Vilanova de Valencia

🇪🇸

Valencia, Spain

Hospital Clinico Universitario de Valencia

🇪🇸

Valencia, Spain

Instituto Valenciano de Oncología

🇪🇸

Valencia, Spain

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