MedPath

A Study Evaluating the Safety and Efficacy of Targeted Therapies in Subpopulations of Patients With Metastatic Colorectal Cancer (INTRINSIC)

Phase 1
Recruiting
Conditions
Metastatic Colorectal Cancer
Interventions
Registration Number
NCT04929223
Lead Sponsor
Hoffmann-La Roche
Brief Summary

This open-label, exploratory study is designed to evaluate the safety and efficacy of targeted therapies or immunotherapy as single agents or combinations, in participants with metastatic colorectal cancer (mCRC) whose tumors are biomarker positive as per treatment arm-specific definition. Eligible participants with mCRC will be enrolled into specific treatment arms based on their biomarker assay results.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
542
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Inavolisib + CetuximabCetuximabParticipants will receive 9 milligrams (mg) of inavolisib by mouth once daily (QD) on Days 8-28 of Cycle 1, then QD on Days 1-28 from Cycle 2 onwards (1 cycle=28 days). Participants will also receive cetuximab intravenous (IV) infusion 400 mg/m2 body surface area on Day 1 of Cycle 1. All subsequent weekly (QW) doses will be 250 mg/m2 each. This arm is active, and not recruiting participants.
Inavolisib + BevacizumabBevacizumabParticipants will receive 9 mg of inavolisib by mouth QD combined with bevacizumab 15 milligram/kilogram (mg/kg) IV once every three weeks (Q3W) on Day 1 of each cycle (1 cycle=21 days). This arm is active, and not recruiting participants.
Atezolizumab + Tiragolumab + BevacizumabBevacizumabParticipants in this randomized cohort will receive 1200 mg of atezolizumab by IV infusion on Day 1 of each cycle, combined with tiragolumab at a dose of 600 mg IV infusion on Day 1 of each cycle and bevacizumab IV infusion at a dose of 15 mg/kg on Day 1 of each cycle. (Cycle length=21 days) This arm is active, and not recruiting participants.
Atezolizumab + Tiragolumab + BevacizumabAtezolizumabParticipants in this randomized cohort will receive 1200 mg of atezolizumab by IV infusion on Day 1 of each cycle, combined with tiragolumab at a dose of 600 mg IV infusion on Day 1 of each cycle and bevacizumab IV infusion at a dose of 15 mg/kg on Day 1 of each cycle. (Cycle length=21 days) This arm is active, and not recruiting participants.
Atezolizumab + Tiragolumab + BevacizumabTiragolumabParticipants in this randomized cohort will receive 1200 mg of atezolizumab by IV infusion on Day 1 of each cycle, combined with tiragolumab at a dose of 600 mg IV infusion on Day 1 of each cycle and bevacizumab IV infusion at a dose of 15 mg/kg on Day 1 of each cycle. (Cycle length=21 days) This arm is active, and not recruiting participants.
Atezolizumab + TiragolumabAtezolizumabParticipants in this randomized cohort will receive 1200 mg of atezolizumab by IV infusion on Day 1 of each cycle combined with tiragolumab 600 mg IV infusion on Day 1 of each cycle. (Cycle length=21 days) This arm is active, and not recruiting participants.
Atezolizumab + TiragolumabTiragolumabParticipants in this randomized cohort will receive 1200 mg of atezolizumab by IV infusion on Day 1 of each cycle combined with tiragolumab 600 mg IV infusion on Day 1 of each cycle. (Cycle length=21 days) This arm is active, and not recruiting participants.
Atezolizumab + SY-5609AtezolizumabParticipants will receive 1680 mg of atezolizumab by IV infusion on Day 1 of each cycle Q4W in repeated 28-day cycles combined with SY-5609 at a dose of 3, 4, 5, 6, 7 or 10 mg by mouth for 7 days, followed by 7 days off. (Cycle length=28 days) This arm is closed.
Atezolizumab + SY-5609SY-5609Participants will receive 1680 mg of atezolizumab by IV infusion on Day 1 of each cycle Q4W in repeated 28-day cycles combined with SY-5609 at a dose of 3, 4, 5, 6, 7 or 10 mg by mouth for 7 days, followed by 7 days off. (Cycle length=28 days) This arm is closed.
Divarasib + Cetuximab + FOLFOXCetuximabParticipants will receive cetuximab IV 500 mg/m2 body surface area on Days 1 and 15 and FOLFOX on Days 1 and 15 with divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Divarasib + Cetuximab + FOLFOXFOLFOXParticipants will receive cetuximab IV 500 mg/m2 body surface area on Days 1 and 15 and FOLFOX on Days 1 and 15 with divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Divarasib + CetuximabCetuximabParticipants will receive cetuximab IV 500 mg/m2 body surface area on Days 1 and 15 with divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is active, and not recruiting participants.
Divarasib + Cetuximab + FOLFIRICetuximabParticipants will receive cetuximab IV 500 mg/m2 body surface area on Days 1 and 15 and FOLFIRI on Days 1 and 15 with divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is active, and not recruiting participants.
Divarasib + Cetuximab + FOLFIRIFOLFIRIParticipants will receive cetuximab IV 500 mg/m2 body surface area on Days 1 and 15 and FOLFIRI on Days 1 and 15 with divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is active, and not recruiting participants.
Divarasib + Bevacizumab + FOLFOXBevacizumabParticipants will receive Bevacizumab 5 mg/kg by IV infusion on Days 1 and 15 and FOLFOX on Days 1 and 15 with Divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Divarasib + Bevacizumab + FOLFOXFOLFOXParticipants will receive Bevacizumab 5 mg/kg by IV infusion on Days 1 and 15 and FOLFOX on Days 1 and 15 with Divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Divarasib + Bevacizumab + FOLFIRIBevacizumabParticipants will receive Bevacizumab 5 mg/kg by IV infusion on Days 1 and 15 and FOLFIRI on Days 1 and 15 with Divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Divarasib + Bevacizumab + FOLFIRIFOLFIRIParticipants will receive Bevacizumab 5 mg/kg by IV infusion on Days 1 and 15 and FOLFIRI on Days 1 and 15 with Divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Divarasib + Cetuximab + FOLFOXDivarasibParticipants will receive cetuximab IV 500 mg/m2 body surface area on Days 1 and 15 and FOLFOX on Days 1 and 15 with divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Divarasib + CetuximabDivarasibParticipants will receive cetuximab IV 500 mg/m2 body surface area on Days 1 and 15 with divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is active, and not recruiting participants.
Divarasib + Cetuximab + FOLFIRIDivarasibParticipants will receive cetuximab IV 500 mg/m2 body surface area on Days 1 and 15 and FOLFIRI on Days 1 and 15 with divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is active, and not recruiting participants.
Divarasib + Bevacizumab + FOLFOXDivarasibParticipants will receive Bevacizumab 5 mg/kg by IV infusion on Days 1 and 15 and FOLFOX on Days 1 and 15 with Divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Divarasib + Bevacizumab + FOLFIRIDivarasibParticipants will receive Bevacizumab 5 mg/kg by IV infusion on Days 1 and 15 and FOLFIRI on Days 1 and 15 with Divarasib PO QD on Days 1-28. (Cycle length=28 days) This arm is recruiting participants.
Inavolisib + CetuximabInavolisibParticipants will receive 9 milligrams (mg) of inavolisib by mouth once daily (QD) on Days 8-28 of Cycle 1, then QD on Days 1-28 from Cycle 2 onwards (1 cycle=28 days). Participants will also receive cetuximab intravenous (IV) infusion 400 mg/m2 body surface area on Day 1 of Cycle 1. All subsequent weekly (QW) doses will be 250 mg/m2 each. This arm is active, and not recruiting participants.
Inavolisib + BevacizumabInavolisibParticipants will receive 9 mg of inavolisib by mouth QD combined with bevacizumab 15 milligram/kilogram (mg/kg) IV once every three weeks (Q3W) on Day 1 of each cycle (1 cycle=21 days). This arm is active, and not recruiting participants.
Primary Outcome Measures
NameTimeMethod
Objective Response RateApproximately 84 months

Defined as the proportion of participants with a complete response or partial response, as determined by the investigator according to RECIST v1.1

Secondary Outcome Measures
NameTimeMethod
Duration of ResponseApproximately 84 months

Defined as the time from the first occurrence of a documented objective response to disease progression or death from any cause (whichever occurs first), as determined by the investigator according to RECIST v1.1

Disease Control RateApproximately 84 months

Defined as the proportion of participants with stable disease, or a complete or partial response, as determined by the investigator according to RECIST v1.1

Percentage of Participants with Adverse Events (AEs)Approximately 84 months

Percentage of participants with adverse events.

Plasma Concentrations of DivarasibAt pre-defined intervals from first administration of study drug up to approximately 84 months

Plasma concentration of divarasib for divarasib + cetuximab + FOLFOX, divarasib + cetuximab, and divarasib + cetuximab+ FOLFIRI, Divarasib + Bevacizumab + FOLFOX, Divarasib + Bevacizumab + FOLFIRI treatment arms.

Recommended Dose of Divarasib in Combination with Bevacizumab and FOLFOXApproximately 84 months

Recommended dose of divarasib in combination with bevacizumab and FOLFOX based on the totality of safety, efficacy and PK data.

Recommended Dose of Divarasib in Combination with Bevacizumab and FOLFIRIApproximately 84 months

Recommended dose of divarasib in combination with bevacizumab and FOLFIRI based on the totality of safety, efficacy and PK data.

Trial Locations

Locations (73)

UAB Comprehensive Cancer Center

🇺🇸

Birmingham, Alabama, United States

Mayo Clinic Arizona

🇺🇸

Phoenix, Arizona, United States

City of Hope Comprehensive Cancer Center

🇺🇸

Duarte, California, United States

cCare

🇺🇸

Encinitas, California, United States

USC Norris Cancer Center

🇺🇸

Los Angeles, California, United States

Cedars-Sinai Medical Center

🇺🇸

Los Angeles, California, United States

UCLA

🇺🇸

Los Angeles, California, United States

Hoag Memorial Hospital Presbyterian

🇺🇸

Newport Beach, California, United States

Stanford Cancer Center

🇺🇸

Stanford, California, United States

University of Colorado Cancer Center

🇺🇸

Aurora, Colorado, United States

Yale Cancer Center

🇺🇸

New Haven, Connecticut, United States

Eastern Ct Hema/Onco Assoc

🇺🇸

Norwich, Connecticut, United States

Mayo Clinic in Florida

🇺🇸

Jacksonville, Florida, United States

Moffitt Cancer Center

🇺🇸

Tampa, Florida, United States

Mary Bird Perkins Cancer Ctr

🇺🇸

Baton Rouge, Louisiana, United States

Massachusetts General Hospital

🇺🇸

Boston, Massachusetts, United States

Karmanos Cancer Institute

🇺🇸

Detroit, Michigan, United States

Mayo Clinic Rochester

🇺🇸

Rochester, Minnesota, United States

New York Cancer & Blood Specialists - Bronx

🇺🇸

Bronx, New York, United States

New York Cancer & Blood Specialists - New Hyde Park

🇺🇸

New Hyde Park, New York, United States

New York Cancer and Blood Specialists-Central Park Hematology & Oncology

🇺🇸

New York, New York, United States

New York Cancer & Blood Specialists

🇺🇸

Port Jefferson Station, New York, United States

Duke University Medical Center

🇺🇸

Durham, North Carolina, United States

Hematology Oncology Salem

🇺🇸

Salem, Oregon, United States

UPMC - Hillman Cancer Center

🇺🇸

Pittsburgh, Pennsylvania, United States

Sarah Cannon Research Institute / Tennessee Oncology

🇺🇸

Nashville, Tennessee, United States

Vanderbilt University Medical Center

🇺🇸

Nashville, Tennessee, United States

Lumi Research

🇺🇸

Kingwood, Texas, United States

Swedish Cancer Inst.

🇺🇸

Seattle, Washington, United States

Medical Oncology Associates

🇺🇸

Spokane, Washington, United States

Peter Maccallum Cancer Centre

🇦🇺

Melbourne, Victoria, Australia

Princess Margaret Cancer Center

🇨🇦

Toronto, Ontario, Canada

Jewish General Hospital

🇨🇦

Montreal, Quebec, Canada

McGill University Health Center

🇨🇦

Montreal, Quebec, Canada

Rigshospitalet, Onkologisk Klinik

🇩🇰

København Ø, Denmark

Charité Universitätsmedizin Berlin

🇩🇪

Berlin, Germany

Katholisches Klinikum Bochum gGmbH - St. Josef-Hospital

🇩🇪

Bochum, Germany

Universitätsklinik Carl Gustav Carus der Technischen Universität Dresden

🇩🇪

Dresden, Germany

Universitätsklinikum Düsseldorf

🇩🇪

Düsseldorf, Germany

Asklepios Klinik Altona

🇩🇪

Hamburg, Germany

SLK-Kliniken Heilbronn GmbH;Klinik für Innere Medizin III

🇩🇪

Heilbronn, Germany

Klinikum der Universität München, Campus Großhadern

🇩🇪

München, Germany

Universitätsklinikum Ulm

🇩🇪

Ulm, Germany

Università degli Studi della Campania Luigi Vanvitelli

🇮🇹

Napoli, Campania, Italy

Policlinico Universitario Agostino Gemelli IRCCS

🇮🇹

Roma, Lazio, Italy

Irccs Istituto Nazionale Dei Tumori (Int)

🇮🇹

Milano, Lombardia, Italy

Azienda Socio Sanitaria Territoriale Niguarda (Ospedale Niguarda Ca' Granda)

🇮🇹

Milano, Lombardia, Italy

IRCCS Istituto Oncologico Veneto (IOV)

🇮🇹

Padova, Veneto, Italy

National Cancer Center

🇰🇷

Goyang-si, Korea, Republic of

Chonnam National University Hwasun Hospital

🇰🇷

Jeollanam-do, Korea, Republic of

Seoul National University Bundang Hospital

🇰🇷

Seongnam-si, Korea, Republic of

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Severance Hospital, Yonsei University Health System

🇰🇷

Seoul, Korea, Republic of

Asan Medical Center

🇰🇷

Seoul, Korea, Republic of

Szpital Uniwersytecki w Krakowie, Oddzia? Kliniczny Kliniki Onkologii

🇵🇱

Kraków, Poland

Uniwersytecki Szpital Kliniczny w Poznaniu

🇵🇱

Poznan, Poland

Narodowy Instytut Onkologii im. M. Sklodowskiej-Curie

🇵🇱

Warszawa, Poland

Vall d?Hebron Institute of Oncology (VHIO), Barcelona

🇪🇸

Barcelona, Spain

START Madrid-FJD, Hospital Fundacion Jimenez Diaz

🇪🇸

Madrid, Spain

START Madrid. Centro Integral Oncologico Clara Campal

🇪🇸

Madrid, Spain

Hospital Clínico Universitario de Valencia

🇪🇸

Valencia, Spain

National Cheng Kung University Hospital

🇨🇳

Tainan, Taiwan

Taipei Veterans General Hospital

🇨🇳

Taipei City, Taiwan

National Taiwan University Hospital

🇨🇳

Zhongzheng Dist., Taiwan

Addenbrookes Hospital

🇬🇧

Cambridge, United Kingdom

Velindre Cancer Centre

🇬🇧

Cardiff, United Kingdom

Royal Free Hospital

🇬🇧

London, United Kingdom

Royal Marsden Hospital;Dept of Med-Onc

🇬🇧

London, United Kingdom

Sarah Cannon Research Institute

🇬🇧

London, United Kingdom

Imperial College Healthcare NHS Trust

🇬🇧

London, United Kingdom

The Christie NHS Foundation Trust

🇬🇧

Manchester, United Kingdom

Royal Marsden Hospital

🇬🇧

Sutton, United Kingdom

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